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Compound Name:

Compounds Sorted by Binding Data per Compound

1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29
30 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55
56 57 58 59 60 61 62 63 64 65 66 67 68 69 70 71 72 73 74 75 76 77 78 79 80 81
82 83 84 85 86 87 88 89 90 91 92 93 94 95 96 97 98 99 100 101 102 103 104 105
106 107 108 109 110 111 112 113 114 115 116 117 118 119 120 121 122 123 124
125 127 128 129 130 132 133 134 135 136 137 138 139 140 141 143 144 145 146
147 148 149 150 151 153 154 155 156 159 160 161 163 164 165 168 170 171 173
174 176 178 179 183 184 186 188 189 190 191 192 193 196 198 199 200 203 204
205 206 207 208 209 210 216 220 224 226 227 229 232 237 238 241 243 248 252
253 259 261 270 274 276 277 285 291 303 304 313 318 323 325 328 333 335 337
339 341 353 360 361 365 389 393 398 401 413 433 442 444 445 446 447 448 451
453 454 455 457 458 460 463 465 467 473 477 478 482 484 499 504 505 506 517
521 525 543 549 551 554 591 606 663 691 708 796 804 821 825 833 842 847 854
855 861 873 879 883 887 913 914 925 926 938 947 1010 1027 1050 1052 1081 1082
1099 1115 1130 1133 1206 1262 1543 1639 1903 2029
Compounds Sorted Alphabetically
Compound Name (alphabetical)
Enz. Inhib. Data
ITC Data
Binding Targets
Alternate Compound Names
1 Ki 11 IC50
  • Caspase-1
  • Caspase-3
  • Caspase-6
  • Caspase-7
  • Caspase-8
  • (S)-1-(4-Methoxybenzyl)-5-(2-phenoxymethyl-pyrrolidine-1-sulfonyl)-1H-indole-2,3-dione
  • 1-[(4-methoxyphenyl)methyl]-5-{[(2S)-2-(phenoxymethyl)pyrrolidine-1-]sulfonyl}-2,3-dihydro-1H-indole-2,3-dione
  • CHEMBL200677
  • Pyrrolidine Isatin Analogue 11b
1 Ki 11 IC50
  • Caspase-1
  • Caspase-3
  • Caspase-6
  • Caspase-7
  • Caspase-8
  • (S)-1-(4-Hydroxybenzyl)-5-(2-phenoxymethyl-pyrrolidine-1-sulfonyl)-1H-indole-2,3-dione
  • 1-[(4-hydroxyphenyl)methyl]-5-{[(2S)-2-(phenoxymethyl)pyrrolidine-1-]sulfonyl}-2,3-dihydro-1H-indole-2,3-dione
  • CHEMBL200927
  • Pyrrolidine Isatin Analogue 11f
4 Ki 8 IC50
  • Caspase-1
  • Caspase-3
  • hIL-1beta
  • (3S)-3-[(2S)-2-[(2S)-2-[(2S)-2-acetamido-3-(4-hydroxyphenyl)propanamido]-3-methylbutanamido]propanamido]-4-oxobutanoic acid
  • Ac-YVAD-CHO
  • CHEMBL37630
9 Ki 3 EC50
  • Beta-2 adrenergic receptor
  • Muscarinic acetylcholine receptor M3
  • US8551978, 322
  • US8551978, 323
  • US8816088, I-66
  • US8816088, I-67
  • US9394275, I-66
  • US9572802, Compound I-67
  • US9682957, I-67
12 IC50
  • Serine/threonine-protein kinase PIM-3
  • Serine/threonine-protein kinase pim-1
  • Serine/threonine-protein kinase pim-2
  • US8575145, 120
  • US8575145, 121
  • US8575145, 150
  • US8575145, 151
  • US8575145, 90
  • US8575145, 91
4 Ki 6 IC50 1 Kd 1 EC50
  • Acetylcholinesterase
  • Carboxylic ester hydrolase
  • Choline transporter
  • Plasminogen
  • Potassium voltage-gated channel subfamily H member 2
  • Prothrombin
  • Pteridine reductase 1
  • Trypsin
  • Twik-RElated Potassium (K+) channel 1 (TREK1)
  • Voltage-gated potassium channel
  • Voltage-gated potassium channel subfamily A member 1/beta-1
  • 4-AP
  • 4-Aminopyridine 10
  • CHEMBL284348
  • DALFAMPRIDINE
  • pyridin-4-amine
12 IC50
  • Nitric oxide synthase, brain
  • Nitric oxide synthase, endothelial
  • Nitric oxide synthase, inducible
  • Sodium-dependent noradrenaline transporter
  • CHEMBL2036264
  • US8586620, 114
9 Ki 3 IC50
  • Serine/threonine-protein kinase pim-1
  • Serine/threonine-protein kinase pim-2
  • Serine/threonine-protein kinase pim-3
  • US8592455, 96
12 IC50
  • CDK2/CycE
  • Cyclin-Dependent Kinase 1 (CDK1)
  • Cyclin-Dependent Kinase 2 (CDK2)
  • Cyclin-Dependent Kinase 5 (CDK5)
  • Cyclin-Dependent Kinase 7 (CDK7)
  • Cyclin-Dependent Kinase 9 (CDK9)
  • Cyclin-dependent kinase 2
  • Cyclin-dependent kinase 4/G1/S-specific cyclin-E1
  • Cyclin-dependent kinase 9
  • Cyclin-dependent-like kinase 5
  • US8592581, 1
12 IC50
  • 11-beta-hydroxysteroid dehydrogenase 1
  • Cytochrome P450 2C19
  • Cytochrome P450 2C9
  • Cytochrome P450 3A
  • US8575157, 200
  • US8592410, Comparator 12
  • US8598163, 70
12 IC50
  • Axin-1/Glycogen synthase kinase-3 beta
  • Cyclin-Dependent Kinase 1 (CDK1)
  • Cyclin-Dependent Kinase 5 (CDK5)
  • Dual specificty protein kinase CLK1
  • Dual-specificity tyrosine-(Y)-phosphorylation regulated kinase 1A
  • Dual-specificity tyrosine-phosphorylation regulated kinase 1A
  • Glycogen Synthase Kinase-3, beta
  • Mitogen-activated protein kinase kinase kinase 14
  • cAMP-Dependent Protein Kinase (PKA)
  • cGMP-Dependent Protein Kinase
  • 4-(1H-indol-3-yl)pyrimidin-2-amine
  • Meridianin G
1 Ki 3 IC50 8 Kd
  • Chitinase 1
  • Chitinase B
  • Chitinase Mutant (A217G)
  • Chitinase Mutant (D175A)
  • Chitinase Mutant (E322A)
  • Chitinase Mutant (M243A)
  • Chitinase Mutant (R301K)
  • Chitinase Mutant (T138A)
  • Chitinase Mutant (Y245F)
  • Endochitinase B1
  • 4-[(1S,4R,10S,13S,16S,18R)-10-{3-[(acetamidomethanimidoyl)amino]propyl}-18-hydroxy-16-(1H-imidazol-4-ylmethyl)-3,9,12,15,20-pentaoxo-2,8,11,14,17-pentaazatricyclo[15.2.1.0^{4,8}]icosan-13-yl]butanoic acid
  • Argadin
  • CHEMBL445236
12 IC50
  • Activin receptor type-1
  • Activin receptor type-1B
  • Activin receptor type-1B/Activin receptor-like kinase 4 (ALK-4)
  • Activin receptor-like kinase 3 (ALK-3)
  • Bone morphogenetic protein receptor type-1B (BMPR1B) aa 168-495
  • Serine/threonine-protein kinase receptor R3
  • Serine/threonine-protein kinase receptor R3 (ALK1)
  • TGF-beta receptor type-1
  • US10017516, Compound 48
  • US9682983, 48
12 IC50
  • Dipeptidyl peptidase 2 (DPP II)
  • Dipeptidyl peptidase 4
  • Dipeptidyl peptidase 9
  • Dipeptidyl peptidase VIII
  • (1S,2S)-1-(dimethylcarbamoyl)-1-[4-(4-fluorophenyl)phenyl]-3-[(3S)-3-fluoropyrrolidin-1-yl]-3-oxopropan-2-aminium; 2,2,2-trifluoroacetate
  • beta-dimethylamide 4
  • beta-substituted phenylalanine deriv. 22
  • phenylalanine derived inhibitor, 3
12 IC50
  • Dipeptidyl peptidase 2 (DPP II)
  • Dipeptidyl peptidase 4
  • Dipeptidyl peptidase 9
  • Dipeptidyl peptidase VIII
  • (2S,3S)-3-[4-(4-fluorophenyl)phenyl]-1-[(3S)-3-fluoropyrrolidin-1-yl]-1-oxobutan-2-aminium; 2,2,2-trifluoroacetate
  • 3-(S)-fluoropyrrolidide 25
  • beta-substituted phenylalanine deriv. 14
  • phenylalanine derived inhibitor, 4
10 Ki 2 IC50
  • 72 kDa type IV collagenase
  • Carbonic Anhydrase IV
  • Carbonic anhydrase 1
  • Carbonic anhydrase 2
  • Collagenase (ChC)
  • Interstitial collagenase
  • Matrix metalloproteinase 12
  • Matrix metalloproteinase-9
  • Neutrophil collagenase
  • (2S)-2-[benzyl(4-methoxybenzene)sulfonamido]-N-hydroxy-3-methylbutanamide
  • Hydroxamate 24
  • N-4-Methoxyphenylsulfonyl-N-benzyl-L-valine hydroxamate
11 Ki 1 IC50
  • 72 kDa type IV collagenase
  • Carbonic Anhydrase IV
  • Carbonic anhydrase 1
  • Carbonic anhydrase 2
  • Collagenase (ChC)
  • Interstitial collagenase
  • Matrix metalloproteinase-9
  • Neutrophil collagenase
  • 2-{[(2-chlorophenyl)methyl](1,1,2,2,3,3,4,4,4-nonafluorobutane)sulfonamido}-N-hydroxypropanamide
  • Hydroxamate 43
  • hydroxamate deriv. B4
11 Ki 1 IC50
  • 72 kDa type IV collagenase
  • Carbonic Anhydrase IV
  • Carbonic anhydrase 1
  • Carbonic anhydrase 2
  • Collagenase (ChC)
  • Interstitial collagenase
  • Matrix metalloproteinase-9
  • Neutrophil collagenase
  • 2-{[(2-chlorophenyl)methyl](2,3,4,5,6-pentafluorobenzene)sulfonamido}-N-hydroxypropanamide
  • Hydroxamate 44
  • hydroxamate deriv. B21
11 Ki 1 IC50
  • 72 kDa type IV collagenase
  • Carbonic Anhydrase IV
  • Carbonic anhydrase 1
  • Carbonic anhydrase 2
  • Collagenase (ChC)
  • Interstitial collagenase
  • Matrix metalloproteinase-9
  • Neutrophil collagenase
  • 2-{[(2-chlorophenyl)methyl](4-methoxybenzene)sulfonamido}-N-hydroxypropanamide
  • Hydroxamate 45
  • hydroxamate deriv. B24
12 IC50
  • Dipeptidyl peptidase 2 (DPP II)
  • Dipeptidyl peptidase 4
  • Dipeptidyl peptidase 9
  • Dipeptidyl peptidase VIII
  • Fibroblast Activation Protein (FAP)
  • Fibroblast activation protein alpha
  • (2S)-1-(2-{[4-(2,3-dihydro-1H-isoindol-2-yl)-2-methyl-4-oxobutan-2-yl]amino}acetyl)pyrrolidine-2-carbonitrile
  • (2S)-Cyanopyrrolidine analogue 21d
  • (2S)-cyanopyrrolidine 4
  • 2-[3-[2-[2-Cyano-(S)-pyrrolidin-1-yl]-2-oxoethylamino]-3-methyl-1-oxobutyl]-1,3-dihydroisoindole
12 IC50
  • Activin receptor type-1
  • Activin receptor type-1B
  • Activin receptor type-1B/Activin receptor-like kinase 4 (ALK-4)
  • Activin receptor-like kinase 3 (ALK-3)
  • Bone morphogenetic protein receptor type-1B (BMPR1B) aa 168-495
  • Serine/threonine-protein kinase receptor R3
  • Serine/threonine-protein kinase receptor R3 (ALK1)
  • TGF-beta receptor type-1
  • US10017516, Compound 3
  • US9682983, 3
12 IC50
  • Activin receptor type-1
  • Activin receptor type-1B
  • Activin receptor type-1B/Activin receptor-like kinase 4 (ALK-4)
  • Activin receptor-like kinase 3 (ALK-3)
  • Bone morphogenetic protein receptor type-1B (BMPR1B) aa 168-495
  • Serine/threonine-protein kinase receptor R3
  • Serine/threonine-protein kinase receptor R3 (ALK1)
  • TGF-beta receptor type-1
  • US10017516, Compound 4
  • US9682983, 4
5 Ki 7 IC50
  • 72 kDa type IV collagenase
  • Collagenase 3
  • Interstitial collagenase
  • Matrix metalloproteinase-14 (MMP14)
  • Matrix metalloproteinase-9
  • Neutrophil collagenase
  • Stromelysin-1
  • 4-{[4-(4-Chlorophenoxy)phenyl]sulfonyl}-N-hydroxy tetrahydro-2H-pyran-4-carboxamide
  • 4-{[4-(4-chlorophenoxy)benzene]sulfonyl}-N-hydroxyoxane-4-carboxamide
  • alpha-sulfone 21
1 Ki 11 IC50
  • Cereblon/Histone deacetylase 6
  • Histone deacetylase 1
  • Histone deacetylase 10
  • Histone deacetylase 11
  • Histone deacetylase 2
  • Histone deacetylase 3
  • Histone deacetylase 4
  • Histone deacetylase 5
  • Histone deacetylase 7
  • Histone deacetylase 8
  • Histone deacetylase 9
  • Prostaglandin E2 receptor EP2 subtype
  • BDBM119696
  • US8685986, 15
4 Ki 4 IC50 4 Kd
  • Cytochrome P450 2C9
  • Cytochrome P450 2D6 (2D6)
  • Cytochrome P450 3A
  • Orexin receptor type 1
  • Orexin receptor type 2
  • Potassium voltage-gated channel subfamily H member 2
  • US8742106, 1.4
3 Ki 9 IC50
  • Cytochrome P450 2A6
  • Cytochrome P450 2B6
  • Cytochrome P450 2C19
  • Cytochrome P450 2C9
  • Cytochrome P450 2D6 (2D6)
  • Cytochrome P450 2E1
  • Cytochrome P450 3A
  • 3-(thiophen-3-yl)pyridine
  • CHEMBL361153
  • US8609708,11
  • nicotine 3-heteroaromatic analogue 8
12 IC50
  • High affinity nerve growth factor receptor
  • JAK2 (aa 808-1132)
  • Tyrosine-protein kinase JAK2
  • US10251889, Example 17
  • US10758542, Example 17
  • US8791123, 17
  • US9782415, Example 17
  • US9796724, Example 17
12 IC50
  • High affinity nerve growth factor receptor
  • Non-receptor tyrosine-protein kinase TYK2
  • Tyk2
  • Tyrosine-protein kinase JAK1
  • Tyrosine-protein kinase JAK2
  • Tyrosine-protein kinase JAK3
  • US8791123, 181
  • US9782415, Example 181
12 IC50
  • Activin receptor type-1
  • Activin receptor type-1B
  • Activin receptor type-1B/Activin receptor-like kinase 4 (ALK-4)
  • Activin receptor-like kinase 3 (ALK-3)
  • Bone morphogenetic protein receptor type-1B (BMPR1B) aa 168-495
  • Serine/threonine-protein kinase receptor R3
  • Serine/threonine-protein kinase receptor R3 (ALK1)
  • TGF-beta receptor type-1
  • US10017516, Compound 6
  • US9682983, 6
12 IC50
  • 3',5'-cyclic phosphodiesterase
  • Lipopolysaccharide-induced tumor necrosis factor-alpha factor
  • Tumor necrosis factor
  • cAMP-specific 3',5'-cyclic phosphodiesterase 4B
  • cAMP-specific 3',5'-cyclic phosphodiesterase 4B (PDE4B2)
  • cAMP-specific 3',5'-cyclic phosphodiesterase 4D
  • phosphodiesterase 4B2
  • phosphodiesterase 4D
  • US10085990, Example 30
  • US10568888, Example 30
  • US8853226, 30
  • US9393245, 30
  • US9833457, 30
12 IC50
  • 3',5'-cyclic phosphodiesterase
  • Lipopolysaccharide-induced tumor necrosis factor-alpha factor
  • Tumor necrosis factor
  • cAMP-specific 3',5'-cyclic phosphodiesterase 4B
  • cAMP-specific 3',5'-cyclic phosphodiesterase 4B (PDE4B2)
  • cAMP-specific 3',5'-cyclic phosphodiesterase 4D
  • phosphodiesterase 4B2
  • phosphodiesterase 4D
  • US10085990, Example 32
  • US10568888, Example 32
  • US8853226, 32
  • US9393245, 32
  • US9833457, 32
12 IC50
  • 3',5'-cyclic phosphodiesterase
  • Lipopolysaccharide-induced tumor necrosis factor-alpha factor
  • Tumor necrosis factor
  • cAMP-specific 3',5'-cyclic phosphodiesterase 4B
  • cAMP-specific 3',5'-cyclic phosphodiesterase 4B (PDE4B2)
  • cAMP-specific 3',5'-cyclic phosphodiesterase 4D
  • phosphodiesterase 4B2
  • phosphodiesterase 4D
  • US10085990, Example 33
  • US10568888, Example 33
  • US8853226, 33
  • US9393245, 33
  • US9833457, 33
12 IC50
  • 3',5'-cyclic phosphodiesterase
  • Lipopolysaccharide-induced tumor necrosis factor-alpha factor
  • Tumor necrosis factor
  • cAMP-specific 3',5'-cyclic phosphodiesterase 4B
  • cAMP-specific 3',5'-cyclic phosphodiesterase 4B (PDE4B2)
  • cAMP-specific 3',5'-cyclic phosphodiesterase 4D
  • phosphodiesterase 4B2
  • phosphodiesterase 4D
  • US10085990, Example 51
  • US10568888, Example 51
  • US8853226, 51
  • US9393245, 51
  • US9833457, 51
12 IC50
  • 3',5'-cyclic phosphodiesterase
  • Lipopolysaccharide-induced tumor necrosis factor-alpha factor
  • Tumor necrosis factor
  • cAMP-specific 3',5'-cyclic phosphodiesterase 4B
  • cAMP-specific 3',5'-cyclic phosphodiesterase 4B (PDE4B2)
  • cAMP-specific 3',5'-cyclic phosphodiesterase 4D
  • phosphodiesterase 4B2
  • phosphodiesterase 4D
  • US10085990, Example 54
  • US10568888, Example 54
  • US8853226, 54
  • US9393245, 54
  • US9833457, 54
12 IC50
  • 3',5'-cyclic phosphodiesterase
  • Lipopolysaccharide-induced tumor necrosis factor-alpha factor
  • Tumor necrosis factor
  • cAMP-specific 3',5'-cyclic phosphodiesterase 4B
  • cAMP-specific 3',5'-cyclic phosphodiesterase 4B (PDE4B2)
  • cAMP-specific 3',5'-cyclic phosphodiesterase 4D
  • phosphodiesterase 4B2
  • phosphodiesterase 4D
  • US10085990, Example 84
  • US10568888, Example 84
  • US8853226, 84
  • US9393245, 84
  • US9833457, 84
12 IC50
  • 3',5'-cyclic phosphodiesterase
  • Lipopolysaccharide-induced tumor necrosis factor-alpha factor
  • Tumor necrosis factor
  • cAMP-specific 3',5'-cyclic phosphodiesterase 4B
  • cAMP-specific 3',5'-cyclic phosphodiesterase 4B (PDE4B2)
  • cAMP-specific 3',5'-cyclic phosphodiesterase 4D
  • phosphodiesterase 4B2
  • phosphodiesterase 4D
  • US10085990, Example 92
  • US10568888, Example 92
  • US8853226, 92
  • US9393245, 92
  • US9833457, 92
12 IC50
  • 3',5'-cyclic phosphodiesterase
  • Lipopolysaccharide-induced tumor necrosis factor-alpha factor
  • Tumor necrosis factor
  • cAMP-specific 3',5'-cyclic phosphodiesterase 4B
  • cAMP-specific 3',5'-cyclic phosphodiesterase 4B (PDE4B2)
  • cAMP-specific 3',5'-cyclic phosphodiesterase 4D
  • phosphodiesterase 4B2
  • phosphodiesterase 4D
  • US10085990, Example 115
  • US10568888, Example 115
  • US8853226, 115
  • US9393245, 115
  • US9833457, 115
12 IC50
  • 3',5'-cyclic phosphodiesterase
  • Lipopolysaccharide-induced tumor necrosis factor-alpha factor
  • Tumor necrosis factor
  • cAMP-specific 3',5'-cyclic phosphodiesterase 4B
  • cAMP-specific 3',5'-cyclic phosphodiesterase 4B (PDE4B2)
  • cAMP-specific 3',5'-cyclic phosphodiesterase 4D
  • phosphodiesterase 4B2
  • phosphodiesterase 4D
  • US10085990, Example 118
  • US10568888, Example 118
  • US8853226, 118
  • US9393245, 118
  • US9833457, 118
12 IC50
  • 3',5'-cyclic phosphodiesterase
  • Lipopolysaccharide-induced tumor necrosis factor-alpha factor
  • Tumor necrosis factor
  • cAMP-specific 3',5'-cyclic phosphodiesterase 4B
  • cAMP-specific 3',5'-cyclic phosphodiesterase 4B (PDE4B2)
  • cAMP-specific 3',5'-cyclic phosphodiesterase 4D
  • phosphodiesterase 4B2
  • phosphodiesterase 4D
  • US10085990, Example 127
  • US10568888, Example 127
  • US8853226, 127
  • US9393245, 127
  • US9833457, 127
12 IC50
  • Beta-secretase 1
  • Cathepsin D
  • Cytochrome P450 1A
  • Cytochrome P450 2C19
  • Cytochrome P450 2C8
  • Cytochrome P450 2D6 (2D6)
  • Cytochrome P450 3A
  • Potassium voltage-gated channel subfamily H member 2
  • US8865706, 9
12 IC50
  • Cereblon/Histone deacetylase 1
  • Cereblon/Histone deacetylase 2
  • Cereblon/Histone deacetylase 6
  • Histone deacetylase 1
  • Histone deacetylase 2
  • Histone deacetylase 3
  • US10858323, Compound 1
  • US8614223, 73
12 Ki
  • Coagulation factor X
  • Prothrombin
  • Trypsin
  • Urokinase-type plasminogen activator
  • 2-(3-HYDROXY-PYRIDIN-2-YL)-1H-BENZOIMIDAZOLE-5-CARBOXAMIDINE
  • APC-1801
  • {amino[2-(3-hydroxypyridin-2-yl)-1H-1,3-benzodiazol-5-yl]methylidene}azanium
12 IC50
  • Androgen Receptor
  • Baculoviral IAP repeat-containing protein 2/Estrogen receptor
  • Estrogen receptor
  • Glucocorticoid receptor
  • Mineralocorticoid receptor
  • Progesterone receptor
  • US8916600, 2
  • US8916600, 3
  • US9738632, Example 2
12 Ki
  • Coagulation factor X
  • Plasminogen
  • Prothrombin
  • Tissue-type plasminogen activator
  • Trypsin
  • Urokinase (uPA) Mutant (S190A)
  • Urokinase-type plasminogen activator
  • 2-{5-[amino(iminiumyl)methyl]-1H-1,3-benzodiazol-2-yl}-6-(cyclopentyloxy)benzen-1-olate
  • APC-10655
  • CA-06
5 Ki 4 IC50 2 Kd 0 Other
  • Beta-secretase 1
  • Coagulation factor III/Factor VIIa (fVIIa)
  • Neutrophil cytosol factor 1
  • Nitric oxide synthase, brain
  • Nitric oxide synthase, endothelial
  • Nitric oxide synthase, inducible
  • Trypsin
  • Tryptase
  • Tyrosine-protein kinase TEC
  • Urokinase-type plasminogen activator
  • 1-amino-isoquinoline
  • CHEMBL62083
  • Fragment 17
  • fragment 1 (J. med. chem.,50,1116)
  • isoquinolin-1-amine
12 IC50
  • Activin receptor type-1
  • Activin receptor type-1B
  • Activin receptor type-1B/Activin receptor-like kinase 4 (ALK-4)
  • Activin receptor-like kinase 3 (ALK-3)
  • Bone morphogenetic protein receptor type-1B (BMPR1B) aa 168-495
  • Serine/threonine-protein kinase receptor R3
  • Serine/threonine-protein kinase receptor R3 (ALK1)
  • TGF-beta receptor type-1
  • US10017516, Compound 7
  • US9682983, 7
12 IC50
  • Activin receptor type-1
  • Activin receptor type-1B
  • Activin receptor type-1B/Activin receptor-like kinase 4 (ALK-4)
  • Activin receptor-like kinase 3 (ALK-3)
  • Bone morphogenetic protein receptor type-1B (BMPR1B) aa 168-495
  • Serine/threonine-protein kinase receptor R3
  • Serine/threonine-protein kinase receptor R3 (ALK1)
  • TGF-beta receptor type-1
  • US10017516, Compound 8
  • US9682983, 8
12 IC50
  • Activin receptor type-1
  • Activin receptor type-1B
  • Activin receptor type-1B/Activin receptor-like kinase 4 (ALK-4)
  • Activin receptor-like kinase 3 (ALK-3)
  • Bone morphogenetic protein receptor type-1B (BMPR1B) aa 168-495
  • Serine/threonine-protein kinase receptor R3
  • Serine/threonine-protein kinase receptor R3 (ALK1)
  • TGF-beta receptor type-1
  • US10017516, Compound 10
  • US9682983, 10
12 IC50
  • Activin receptor type-1
  • Activin receptor type-1B
  • Activin receptor type-1B/Activin receptor-like kinase 4 (ALK-4)
  • Activin receptor-like kinase 3 (ALK-3)
  • Bone morphogenetic protein receptor type-1B (BMPR1B) aa 168-495
  • Serine/threonine-protein kinase receptor R3
  • Serine/threonine-protein kinase receptor R3 (ALK1)
  • TGF-beta receptor type-1
  • US10017516, Compound 11
  • US9682983, 11
12 Ki
  • Coagulation factor X
  • Plasminogen
  • Prothrombin
  • Tissue-type plasminogen activator
  • Trypsin
  • Trypsin-1
  • Tryptase
  • Urokinase (uPA) Mutant (S190A)
  • Urokinase-type plasminogen activator
  • 2-{5-[amino(iminiumyl)methyl]-6-fluoro-1H-1,3-benzodiazol-2-yl}-6-phenylbenzen-1-olate
  • CA-09
  • CRA-10818
12 IC50
  • Anandamide amidohydrolase
  • Cytochrome P450 1A
  • Cytochrome P450 2C19
  • Cytochrome P450 2C9
  • Cytochrome P450 2D6
  • Cytochrome P450 3A
  • Fatty-acid amide hydrolase 1
  • US9682953, 20.A-1
12 IC50
  • Anandamide amidohydrolase
  • Cytochrome P450 1A
  • Cytochrome P450 2C19
  • Cytochrome P450 2C9
  • Cytochrome P450 2D6
  • Cytochrome P450 3A
  • Fatty-acid amide hydrolase 1
  • US9682953, 20.A-3
12 IC50
  • Activin receptor type-1
  • Activin receptor type-1B
  • Activin receptor type-1B/Activin receptor-like kinase 4 (ALK-4)
  • Activin receptor-like kinase 3 (ALK-3)
  • Bone morphogenetic protein receptor type-1B (BMPR1B) aa 168-495
  • Serine/threonine-protein kinase receptor R3
  • Serine/threonine-protein kinase receptor R3 (ALK1)
  • TGF-beta receptor type-1
  • US10017516, Compound 13
  • US9682983, 13
12 Ki
  • Orexin receptor type 1 (OX1)
  • Orexin receptor type 2
  • Orexin receptor type 2 (OX2)
  • US10183953, Example 4
  • US8969352, 4
  • US9611277, Example 4
  • US9845333, 4
12 Ki
  • Orexin receptor type 1 (OX1)
  • Orexin receptor type 2
  • Orexin receptor type 2 (OX2)
  • US10183953, Example 21
  • US8969352, 21
  • US9611277, Example 21
  • US9845333, 21
12 Ki
  • Orexin receptor type 1 (OX1)
  • Orexin receptor type 2
  • Orexin receptor type 2 (OX2)
  • US10183953, Example 31
  • US8969352, 31
  • US9611277, Example 31
  • US9845333, 31
12 Ki
  • Orexin receptor type 1
  • Orexin receptor type 1 (OX1)
  • Orexin receptor type 2
  • Orexin receptor type 2 (OX2)
  • US10183953, Example 32
  • US8969352, 32
  • US9845333, 32
12 Ki
  • Orexin receptor type 1 (OX1)
  • Orexin receptor type 2
  • Orexin receptor type 2 (OX2)
  • US10183953, Example 41
  • US8969352, 41
  • US9611277, Example 41
  • US9845333, 41
12 Ki
  • Orexin receptor type 1 (OX1)
  • Orexin receptor type 2
  • Orexin receptor type 2 (OX2)
  • US10183953, Example 51
  • US8969352, 51
  • US9611277, Example 51
  • US9845333, 51
12 Ki
  • Orexin receptor type 1 (OX1)
  • Orexin receptor type 2
  • Orexin receptor type 2 (OX2)
  • US10183953, Example 52
  • US8969352, 52
  • US9611277, Example 52
  • US9845333, 52
12 Ki
  • Orexin receptor type 1
  • Orexin receptor type 1 (OX1)
  • Orexin receptor type 2
  • Orexin receptor type 2 (OX2)
  • US8969352, 54
  • US9611277, Example 54
  • US9845333, 54
12 Ki
  • 5-lipoxygenase-activating protein (FLAP)
  • 5-lipoxygenase/FLAP
  • US8952177, 1
  • US8952177, 5
  • US8952177, 6
  • US9089569, 7
  • US9695149, 6
12 IC50
  • Coagulation factor III/Factor VIIa (fVIIa)
  • Coagulation factor VII
  • Coagulation factor X
  • Prothrombin
  • Thrombin and coagulation factor VII
  • 2-[3-Amino-3-fluoro-4-(isopropylamino)-1,1-biphenyl-2-yl]-N-{4-[amino(imino)methyl]benzyl}acetamide
  • 2-[6-(3-aminophenyl)-2-fluoro-3-(propan-2-ylamino)phenyl]-N-[(4-carbamimidoylphenyl)methyl]acetamide
  • CHEMBL125781
  • Substituted Benzene Analog 50c
12 IC50
  • Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B
  • Mitogen-activated protein kinase 14
  • Phosphodiesterase 8
  • Phosphodiesterase Type 10 (PDE10A)
  • Phosphodiesterase Type 11 (PDE11A)
  • Phosphodiesterase Type 2 (PDE2A)
  • Phosphodiesterase Type 3 (PDE3B)
  • Phosphodiesterase Type 4 (PDE4B)
  • Phosphodiesterase Type 4 (PDE4D)
  • Phosphodiesterase Type 5 (PDE5A)
  • Phosphodiesterase Type 7 (PDE7B)
  • Phosphodiesterase Type 9 (PDE9A)
  • (E)-{1-[3-(cyclopentyloxy)-4-methoxyphenyl]ethylidene}amino carbamate
  • Filaminast
  • [1-(3-cyclopentyloxy-4-methoxy-phenyl)ethylideneamino] carbamate
12 IC50
  • Activin receptor type-1
  • Activin receptor type-1B
  • Activin receptor type-1B/Activin receptor-like kinase 4 (ALK-4)
  • Activin receptor-like kinase 3 (ALK-3)
  • Bone morphogenetic protein receptor type-1B (BMPR1B) aa 168-495
  • Serine/threonine-protein kinase receptor R3
  • Serine/threonine-protein kinase receptor R3 (ALK1)
  • TGF-beta receptor type-1
  • US10017516, Compound 24
  • US9682983, 24
12 IC50
  • Activin receptor type-1
  • Activin receptor type-1B
  • Activin receptor type-1B/Activin receptor-like kinase 4 (ALK-4)
  • Activin receptor-like kinase 3 (ALK-3)
  • Bone morphogenetic protein receptor type-1B (BMPR1B) aa 168-495
  • Serine/threonine-protein kinase receptor R3
  • Serine/threonine-protein kinase receptor R3 (ALK1)
  • TGF-beta receptor type-1
  • US10017516, Compound 27
  • US9682983, 27
12 IC50
  • Activin receptor type-1
  • Activin receptor type-1B
  • Activin receptor type-1B/Activin receptor-like kinase 4 (ALK-4)
  • Activin receptor-like kinase 3 (ALK-3)
  • Bone morphogenetic protein receptor type-1B (BMPR1B) aa 168-495
  • Serine/threonine-protein kinase receptor R3
  • Serine/threonine-protein kinase receptor R3 (ALK1)
  • TGF-beta receptor type-1
  • US10017516, Compound 28
  • US9682983, 28
12 IC50
  • Activin receptor type-1
  • Activin receptor type-1B
  • Activin receptor type-1B/Activin receptor-like kinase 4 (ALK-4)
  • Activin receptor-like kinase 3 (ALK-3)
  • Bone morphogenetic protein receptor type-1B (BMPR1B) aa 168-495
  • Serine/threonine-protein kinase receptor R3
  • Serine/threonine-protein kinase receptor R3 (ALK1)
  • TGF-beta receptor type-1
  • US10017516, Compound 31
  • US9682983, 31
12 IC50
  • Activin receptor type-1
  • Activin receptor type-1B
  • Activin receptor type-1B/Activin receptor-like kinase 4 (ALK-4)
  • Activin receptor-like kinase 3 (ALK-3)
  • Bone morphogenetic protein receptor type-1B (BMPR1B) aa 168-495
  • Serine/threonine-protein kinase receptor R3
  • Serine/threonine-protein kinase receptor R3 (ALK1)
  • TGF-beta receptor type-1
  • US10017516, Compound 33
  • US9682983, 33
12 IC50
  • Activin receptor type-1
  • Activin receptor type-1B
  • Activin receptor type-1B/Activin receptor-like kinase 4 (ALK-4)
  • Activin receptor-like kinase 3 (ALK-3)
  • Bone morphogenetic protein receptor type-1B (BMPR1B) aa 168-495
  • Serine/threonine-protein kinase receptor R3
  • Serine/threonine-protein kinase receptor R3 (ALK1)
  • TGF-beta receptor type-1
  • US10017516, Compound 35
  • US9682983, 35
12 IC50
  • Activin receptor type-1
  • Activin receptor type-1B
  • Activin receptor type-1B/Activin receptor-like kinase 4 (ALK-4)
  • Activin receptor-like kinase 3 (ALK-3)
  • Bone morphogenetic protein receptor type-1B (BMPR1B) aa 168-495
  • Serine/threonine-protein kinase receptor R3
  • Serine/threonine-protein kinase receptor R3 (ALK1)
  • TGF-beta receptor type-1
  • US10017516, Compound 36
  • US9682983, 36
12 IC50
  • Activin receptor type-1
  • Activin receptor type-1B
  • Activin receptor type-1B/Activin receptor-like kinase 4 (ALK-4)
  • Activin receptor-like kinase 3 (ALK-3)
  • Bone morphogenetic protein receptor type-1B (BMPR1B) aa 168-495
  • Serine/threonine-protein kinase receptor R3
  • Serine/threonine-protein kinase receptor R3 (ALK1)
  • TGF-beta receptor type-1
  • US10017516, Compound 37
  • US9682983, 37
2 Ki 10 IC50
  • Beta-secretase 1
  • Potassium voltage-gated channel subfamily H member 2
  • US8975415, RP111
  • US8975415, RP52a
  • US9242973, RP111
12 IC50
  • Protein kinase B (Akt 1)
  • Protein kinase C (PKC)
  • Protein kinase C, gamma
  • RAC-alpha serine/threonine-protein kinase
  • Serine/threonine-protein kinase AKT
  • Serine/threonine-protein kinase AKT2
  • cAMP-Dependent Protein Kinase (PKA)
  • 3-[(2S)-2-amino-3-({5-[(E)-2-(pyridin-4-yl)ethenyl]pyridin-3-yl}oxy)propyl]-1H-indole
  • bispyridinylethylene, 2
  • pyridine-base inhibitor 1b
  • trans-bispyridinylethylene analog 2q
2 Ki 10 IC50
  • Protein kinase B (Akt 1)
  • Protein kinase C (PKC)
  • Protein kinase C, gamma
  • RAC-alpha serine/threonine-protein kinase
  • Serine/threonine-protein kinase AKT
  • Serine/threonine-protein kinase AKT2
  • Serine/threonine-protein kinase Chk1/2
  • cAMP-Dependent Protein Kinase (PKA)
  • (2S)-1-(1H-indol-3-yl)-3-(5-isoquinolin-6-ylpyridin-3-yl)oxy-propan-2-amine
  • 13a (S-)
  • 5-isoquinolinyl pyridine 2
  • 6-{5-[(2S)-2-amino-3-(1H-indol-3-yl)propoxy]pyridin-3-yl}isoquinoline
  • isoquinoline-pyridine, 1
  • isoquinoline-pyridine, 3
  • pyridine-base inhibitor 13a
12 IC50
  • Aldehyde dehydrogenase, mitochondrial
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] A
  • Amine oxidase [flavin-containing] B
  • US10507215, Compound 7
  • US9000015, 7
  • US9610299, Example 7
12 IC50
  • Aldehyde dehydrogenase, mitochondrial
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] A
  • Amine oxidase [flavin-containing] B
  • US10507215, Compound 14
  • US9000015, 14
  • US9610299, Example 14
10 IC50 2 Kd
  • Chromobox protein homolog 7 (CBX7)
  • E3 ubiquitin-protein ligase (UHRF1)
  • Lethal(3)malignant brain tumor-like protein 1 (L3MBTL1)
  • Lysine-specific demethylase 5A
  • MBT domain-containing protein 1 (MBTD1)
  • Methyl-lysine binding protein (53BP1)
  • PHD finger protein 1 (PHF1)
  • PHD finger protein 19 (PHF19)
  • PHD finger protein 23 (PHF23)
  • Tumor suppressor p53-binding protein 1
  • 3-Bromo-N-(3-(tert-butylamino)propyl)benzamide (UNC2170, 1)
12 IC50
  • Cytochrome P450 1A
  • Cytochrome P450 1A1
  • Cytochrome P450 2C19
  • Cytochrome P450 2C8
  • Cytochrome P450 2C9
  • Cytochrome P450 2D6
  • Cytochrome P450 2D6 (2D6)
  • H3K27me2
  • H3K27me3
  • US10098888, Compound 1
  • US9006242, 1
12 IC50
  • Cytochrome P450 1A
  • Cytochrome P450 1A1
  • Cytochrome P450 2C19
  • Cytochrome P450 2C8
  • Cytochrome P450 2C9
  • Cytochrome P450 2D6
  • Cytochrome P450 2D6 (2D6)
  • H3K27me2
  • H3K27me3
  • US10098888, Compound 2
  • US9006242, 2
6 Ki 6 IC50
  • Mitogen-activated protein kinase 10
  • Mitogen-activated protein kinase 8
  • Mitogen-activated protein kinase 9
  • Aminopyridine-Based Inhibitor 6o
  • N-(4-Amino-5-cyano-6-ethoxypyridin-2-yl)-2-(2,5-dimethoxyphenyl)acetamide
  • aminopyridine deriv. 2
12 IC50
  • Sodium-dependent dopamine transporter
  • Sodium-dependent noradrenaline transporter
  • Sodium-dependent serotonin transporter
  • US9034899, 36
  • US9173879, 1 (-) - enantiomer
  • US9604960, 36
12 IC50
  • Non-receptor tyrosine-protein kinase TYK2
  • Tyrosine-protein kinase JAK1
  • Tyrosine-protein kinase JAK2
  • Tyrosine-protein kinase JAK3
  • PF-02384554
  • US9035074, 8
4 Ki 8 IC50
  • P2X purinoceptor 7
  • P2X purinoceptor 7 (P2X7)
  • P2X7 rat
  • US10047092, 15
  • US10053463, 15
  • US9040534, 15
6 Ki 6 IC50
  • P2X purinoceptor 7
  • P2X purinoceptor 7 (P2X7)
  • P2X7 rat
  • US10047092, 19
  • US10053463, 19
  • US9040534, 19
6 Ki 6 IC50
  • P2X purinoceptor 7
  • P2X purinoceptor 7 (P2X7)
  • P2X7 rat
  • US10047092, 20
  • US10053463, 20
  • US9040534, 20
6 Ki 6 IC50
  • P2X purinoceptor 7
  • P2X purinoceptor 7 (P2X7)
  • P2X7 rat
  • US10047092, 21
  • US10053463, 21
  • US9040534, 21
6 Ki 6 IC50
  • P2X purinoceptor 7
  • P2X purinoceptor 7 (P2X7)
  • P2X7 rat
  • US10047092, 22
  • US10053463, 22
  • US9040534, 22
6 Ki 6 IC50
  • P2X purinoceptor 7
  • P2X purinoceptor 7 (P2X7)
  • P2X7 rat
  • US10047092, 26
  • US10053463, 26
  • US9040534, 26
6 Ki 6 IC50
  • P2X purinoceptor 7
  • P2X purinoceptor 7 (P2X7)
  • P2X7 rat
  • US10047092, 32
  • US10053463, 32
  • US9040534, 32
4 Ki 8 IC50
  • P2X purinoceptor 7
  • P2X purinoceptor 7 (P2X7)
  • P2X7 rat
  • US10047092, 33
  • US10053463, 33
  • US9040534, 33
6 Ki 6 IC50
  • P2X purinoceptor 7
  • P2X purinoceptor 7 (P2X7)
  • P2X7 rat
  • US10047092, 34
  • US10053463, 34
  • US9040534, 34
6 Ki 6 IC50
  • P2X purinoceptor 7
  • P2X purinoceptor 7 (P2X7)
  • P2X7 rat
  • US10047092, 45
  • US10053463, 45
  • US9040534, 45
4 Ki 8 IC50
  • P2X purinoceptor 7
  • P2X purinoceptor 7 (P2X7)
  • P2X7 rat
  • US10047092, 52
  • US10053463, 52
  • US9040534, 52
6 Ki 6 IC50
  • P2X purinoceptor 7
  • P2X purinoceptor 7 (P2X7)
  • P2X7 rat
  • US10047092, 75
  • US10053463, 75
  • US9040534, 75
6 Ki 6 IC50
  • P2X purinoceptor 7
  • P2X purinoceptor 7 (P2X7)
  • P2X7 rat
  • US10047092, 76
  • US10053463, 76
  • US9040534, 76
4 Ki 8 IC50
  • P2X purinoceptor 7
  • P2X purinoceptor 7 (P2X7)
  • P2X7 rat
  • US10047092, 80
  • US10053463, 80
  • US9040534, 80
4 Ki 8 IC50
  • P2X purinoceptor 7
  • P2X purinoceptor 7 (P2X7)
  • P2X7 rat
  • US10047092, 85
  • US10053463, 85
  • US9040534, 85
4 Ki 8 IC50
  • P2X purinoceptor 7
  • P2X purinoceptor 7 (P2X7)
  • P2X7 rat
  • US10047092, 86
  • US10053463, 86
  • US9040534, 86
4 Ki 8 IC50
  • P2X purinoceptor 7
  • P2X purinoceptor 7 (P2X7)
  • P2X7 rat
  • US10047092, 88
  • US10053463, 88
  • US9040534, 88
6 Ki 6 IC50
  • P2X purinoceptor 7
  • P2X purinoceptor 7 (P2X7)
  • P2X7 rat
  • US10047092, 92
  • US10053463, 92
  • US9040534, 92
6 Ki 6 IC50
  • P2X purinoceptor 7
  • P2X purinoceptor 7 (P2X7)
  • P2X7 rat
  • US10047092, 94
  • US10053463, 94
  • US9040534, 94
12 IC50
  • Fibroblast growth factor receptor 1
  • Fibroblast growth factor receptor 2
  • Fibroblast growth factor receptor 3
  • Fibroblast growth factor receptor 4
  • US10124003, Ref. Ex. Compound 3
  • US10835536, Ex. Comp 2
  • US10894048, Ex Comp 2
  • US9108973, 2
12 IC50
  • Activin receptor type-1
  • Activin receptor-like kinase 3 (ALK-3)
  • Bone morphogenetic protein receptor type-1B (BMPR1B) aa 168-495
  • Serine/threonine-protein kinase receptor R3
  • Serine/threonine-protein kinase receptor R3 (ALK1)
  • US10017516, Compound 47
  • US9682983, 47
  • US9682983, 49
12 IC50
  • Activin receptor type-1
  • Activin receptor type-1B
  • Activin receptor type-1B/Activin receptor-like kinase 4 (ALK-4)
  • Activin receptor-like kinase 3 (ALK-3)
  • Bone morphogenetic protein receptor type-1B (BMPR1B) aa 168-495
  • Serine/threonine-protein kinase receptor R3
  • Serine/threonine-protein kinase receptor R3 (ALK1)
  • TGF-beta receptor type-1
  • US10017516, Compound 54
  • US9682983, 54
12 IC50
  • Activin receptor type-1
  • Activin receptor type-1B
  • Activin receptor type-1B/Activin receptor-like kinase 4 (ALK-4)
  • Activin receptor-like kinase 3 (ALK-3)
  • Bone morphogenetic protein receptor type-1B (BMPR1B) aa 168-495
  • Serine/threonine-protein kinase receptor R3
  • Serine/threonine-protein kinase receptor R3 (ALK1)
  • TGF-beta receptor type-1
  • US10017516, Compound 62
  • US9682983, 62
12 Ki
  • Coagulation factor VII
  • Coagulation factor X
  • Prothrombin
  • Trypsin-1
  • Tryptase
  • 2-(1H-1,3-benzodiazol-2-ylmethyl)-1H-1,3-benzodiazole-6-carboximidamide
  • 2-(1H-benzimidazol-2-ylmethyl)-1H-benzimidazole-6-carboximidamide
  • APD-1
  • CHEMBL46148
12 Ki
  • Orexin receptor type 1
  • Orexin receptor type 1 (OX1)
  • Orexin receptor type 2
  • US9062078, 1
  • US9475819, 1
  • US9637496, 1
  • US9695183, 1
12 Ki
  • Orexin receptor type 1
  • Orexin receptor type 1 (OX1)
  • Orexin receptor type 2
  • US9062078, 33
  • US9475819, 33
  • US9637496, 33
  • US9695183, 33
12 Ki
  • Orexin receptor type 1
  • Orexin receptor type 1 (OX1)
  • Orexin receptor type 2
  • US9062078, 35
  • US9475819, 35
  • US9637496, 35
  • US9695183, 35
12 Ki
  • Orexin receptor type 1
  • Orexin receptor type 1 (OX1)
  • Orexin receptor type 2
  • US9062078, 49
  • US9475819, 49
  • US9637496, 49
  • US9695183, 49
12 Ki
  • Orexin receptor type 1
  • Orexin receptor type 1 (OX1)
  • Orexin receptor type 2
  • US9062078, 58
  • US9475819, 58
  • US9637496, 58
  • US9695183, 58
12 Ki
  • Orexin receptor type 1
  • Orexin receptor type 1 (OX1)
  • Orexin receptor type 2
  • US9062078, 62
  • US9475819, 62
  • US9637496, 62
  • US9695183, 62
12 Ki
  • Orexin receptor type 1
  • Orexin receptor type 1 (OX1)
  • Orexin receptor type 2
  • US9062078, 63
  • US9475819, 63
  • US9637496, 63
  • US9695183, 63
12 Ki
  • Orexin receptor type 1
  • Orexin receptor type 1 (OX1)
  • Orexin receptor type 2
  • US9062078, 64
  • US9475819, 64
  • US9637496, 64
  • US9695183, 64
12 Ki
  • Orexin receptor type 1
  • Orexin receptor type 1 (OX1)
  • Orexin receptor type 2
  • US9062078, 66
  • US9475819, 66
  • US9637496, 66
  • US9695183, 66
12 Ki
  • Orexin receptor type 1
  • Orexin receptor type 1 (OX1)
  • Orexin receptor type 2
  • US9062078, 67
  • US9475819, 67
  • US9637496, 67
  • US9695183, 67
12 Ki
  • Orexin receptor type 1
  • Orexin receptor type 1 (OX1)
  • Orexin receptor type 2
  • US9062078, 68
  • US9475819, 68
  • US9637496, 68
  • US9695183, 68
12 Ki
  • Orexin receptor type 1
  • Orexin receptor type 1 (OX1)
  • Orexin receptor type 2
  • US9062078, 69
  • US9475819, 69
  • US9637496, 69
  • US9695183, 69
12 Ki
  • Orexin receptor type 1
  • Orexin receptor type 1 (OX1)
  • Orexin receptor type 2
  • US9062078, 70
  • US9475819, 70
  • US9637496, 70
  • US9695183, 70
12 Ki
  • Orexin receptor type 1
  • Orexin receptor type 1 (OX1)
  • Orexin receptor type 2
  • US9062078, 72
  • US9475819, 72
  • US9637496, 72
  • US9695183, 72
12 Ki
  • Orexin receptor type 1
  • Orexin receptor type 1 (OX1)
  • Orexin receptor type 2
  • US9062078, 75
  • US9475819, 75
  • US9637496, 75
  • US9695183, 75
12 Ki
  • Orexin receptor type 1
  • Orexin receptor type 1 (OX1)
  • Orexin receptor type 2
  • US9062078, 88
  • US9475819, 88
  • US9637496, 88
  • US9695183, 88
12 Ki
  • Orexin receptor type 1
  • Orexin receptor type 1 (OX1)
  • Orexin receptor type 2
  • US9062078, 89
  • US9475819, 89
  • US9637496, 89
  • US9695183, 89
12 Ki
  • Orexin receptor type 1
  • Orexin receptor type 1 (OX1)
  • Orexin receptor type 2
  • US9062078, 92
  • US9475819, 92
  • US9637496, 92
  • US9695183, 92
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