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Compounds Sorted by Binding Data per Compound

1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29
30 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55
56 57 58 59 60 61 62 63 64 65 66 67 68 69 70 71 72 73 74 75 76 77 78 79 80 81
82 83 84 85 86 87 88 89 90 91 92 93 94 95 96 97 98 99 100 101 102 103 104 105
106 107 108 109 110 111 112 113 114 115 116 117 118 119 120 121 122 123 124
125 127 128 129 130 132 133 134 135 136 137 138 139 140 141 143 144 145 146
147 148 149 150 151 153 154 155 156 159 160 161 163 164 165 168 170 171 173
174 176 178 179 183 184 186 188 189 190 191 192 193 196 198 199 200 203 204
205 206 207 208 209 210 216 220 224 226 227 229 232 237 238 241 243 248 252
253 259 261 270 274 276 277 285 291 303 304 313 318 323 325 328 333 335 337
339 341 353 360 361 365 389 393 398 401 413 433 442 444 445 446 447 448 451
453 454 455 457 458 460 463 465 467 473 477 478 482 484 499 504 505 506 517
521 525 543 549 551 554 591 606 663 691 708 796 804 821 825 833 842 847 854
855 861 873 879 883 887 913 914 925 926 938 947 1010 1027 1050 1052 1081 1082
1099 1115 1130 1133 1206 1262 1543 1639 1903 2029
Compounds Sorted Alphabetically
Compound Name (alphabetical)
Enz. Inhib. Data
ITC Data
Binding Targets
Alternate Compound Names
8 Ki 131 IC50 1 Kd
  • Axin-1/Glycogen synthase kinase-3 beta
  • BRD4 bromodomain 1
  • BRD4 bromodomain 2
  • Bromodomain-containing protein 2
  • Bromodomain-containing protein 3
  • Bromodomain-containing protein 4
  • Bromodomain-containing protein 4 Bromo 1 domain(BRD4 BD1)
  • Bromodomain-containing protein 4 Bromo 2 domain(BRD4 BD2)
  • DNA-dependent protein kinase
  • Homo sapiens phosphodiesterase 2A (PDE2A)
  • PI3-kinase class I
  • PI3-kinase p110-alpha subunit
  • Peptidyl-prolyl cis-trans isomerase FKBP1B/Serine/threonine-protein kinase mTOR
  • Phosphatidylinositol 3-kinase regulatory subunit beta
  • Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
  • Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform (PI3K alpha)
  • Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform
  • Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
  • Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
  • Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit alpha
  • Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta
  • Phosphodiesterase 3
  • Phosphoinositide 3-Kinase (PI3K), delta
  • Phosphoinositide 3-Kinase (PI3K), gamma
  • Polo-Like Kinase 3
  • Polo-Like Kinase 4
  • Serine-protein kinase ATM
  • Serine/threonine-protein kinase ATR
  • Serine/threonine-protein kinase PLK1
  • Serine/threonine-protein kinase PLK2
  • Serine/threonine-protein kinase PLK3
  • Serine/threonine-protein kinase mTOR
  • Serine/threonine-protein kinase pim-1
  • Serine/threonine-protein kinase pim-3
  • mTOR/FKBP12A/FKBP12B
  • p110α/p85α
  • p110β/p85α
  • 2-(4-Morpholinyl)-8-phenyl-4H-1-benzopyran-4-one
  • 2-(morpholin-4-yl)-8-phenyl-4H-chromen-4-one
  • CHEMBL98350
  • LY294002
  • US10308662, Compound LY294002
  • US9505780, LY294002
18 Ki 10 IC50 43 Kd 69 EC50
  • Cellular retinoic acid-binding protein I
  • Cellular retinoic acid-binding protein II
  • NR2B Channel Blocker
  • Nuclear receptor ROR-gamma (RORC)
  • Oxysterols receptor LXR-alpha
  • Oxysterols receptor LXR-beta
  • Retinoic Acid Receptor, alpha
  • Retinoic Acid Receptor, beta
  • Retinoic Acid Receptor, gamma
  • Retinoic acid receptor RXR-alpha
  • Retinoic acid receptor RXR-alpha/Retinoic acid receptor beta
  • Retinoic acid receptor RXR-alpha/gamma
  • Retinoic acid receptor alpha
  • Retinoic acid receptor alpha/Retinoid X receptor alpha
  • Retinoic acid receptor beta
  • Retinoic acid receptor gamma
  • Retinoid X receptor alpha
  • Retinoid X receptor beta
  • Retinoid X receptor gamma
  • Retinoid X receptor gamma/retinoic acid receptor alpha
  • Retinoid receptor
  • 9-cis retinoic acid
  • 9C-RA
  • CHEMBL705
  • Panretin
  • alitretinoin
140 IC50
  • 5'-AMP-activated protein kinase subunit beta-1
  • 6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 3 (PFKFB3)
  • ALK tyrosine kinase receptor
  • Apoptosis Signal-regulating Kinase 1 (ASK1)
  • Aurora kinase A/Targeting protein for Xklp2
  • Axin-1/Glycogen synthase kinase-3 beta
  • BR serine/threonine-protein kinase 1
  • CaM kinase I alpha
  • CaM kinase IV
  • Casein kinase I isoform delta
  • Cell division cycle 7-related protein kinase
  • Cyclin-Dependent Kinase 5 (CDK5)
  • DNA-dependent protein kinase
  • Death-associated protein kinase 2
  • Death-associated protein kinase 3
  • Discoidin domain-containing receptor 2
  • Dual specificity mitogen-activated protein kinase kinase 1
  • Dual specificity mitogen-activated protein kinase kinase 4
  • Dual specificity mitogen-activated protein kinase kinase 6
  • Dual specificity mitogen-activated protein kinase kinase 7 (MAP2K7)
  • Dual specificity protein kinase CLK2
  • Dual-specificity tyrosine-phosphorylation regulated kinase 2
  • EPHB1
  • Ephrin type-A receptor 2
  • Epidermal growth factor receptor
  • Fibroblast growth factor receptor 1
  • Fibroblast growth factor receptor 2
  • Fibroblast growth factor receptor 3
  • Fibroblast growth factor receptor 4
  • Focal adhesion kinase 1
  • G protein-coupled receptor kinase 5
  • Glycogen synthase kinase-3
  • Heat shock protein HSP 90-beta
  • Hepatocyte growth factor receptor
  • Homeodomain-interacting protein kinase 2 (HIPK2)
  • Inhibitor of nuclear factor kappa-B kinase subunit alpha
  • Inhibitor of nuclear factor kappa-B kinase subunit beta
  • Insulin-like growth factor I receptor
  • Interleukin-1 receptor-associated kinase 1
  • LIM domain kinase 1
  • MAP kinase-activated protein kinase 2
  • MAP kinase-activated protein kinase 3
  • MAP kinase-activated protein kinase 5
  • MAP kinase-interacting serine/threonine-protein kinase 2
  • Mast/stem cell growth factor receptor Kit
  • Misshapen-like kinase 1
  • Mitogen-activated protein kinase 1
  • Mitogen-activated protein kinase 10
  • Mitogen-activated protein kinase 8
  • Mitogen-activated protein kinase kinase kinase 9 (MLK1)
  • Mitogen-activated protein kinase kinase kinase kinase 2
  • Muscle, skeletal receptor tyrosine protein kinase
  • Nuclear receptor subfamily 2 group C member 2
  • PAS domain-containing serine/threonine-protein kinase
  • PKC alpha and beta-2
  • PTK2B protein tyrosine kinase 2 beta (PTK2B)
  • Phosphatidylinositol 3-kinase catalytic subunit type 3
  • Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
  • Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform
  • Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
  • Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
  • Platelet-derived growth factor receptor beta
  • Protein kinase C (PKC)
  • Protein kinase C alpha type
  • Protein kinase C delta type
  • Protein kinase C iota (PKCι)
  • Protein kinase C theta type
  • Protein kinase C, epsilon
  • Protein kinase C, eta
  • Protein kinase C, gamma
  • Protein kinase N2
  • Proto-oncogene tyrosine-protein kinase ROS
  • Proto-oncogene tyrosine-protein kinase Src
  • Proto-oncogene tyrosine-protein kinase receptor Ret
  • RAC-alpha serine/threonine-protein kinase
  • RAF proto-oncogene serine/threonine-protein kinase
  • Receptor tyrosine-protein kinase erbB-2
  • Rho-associated protein kinase 1
  • Rho-associated protein kinase 2
  • Ribosomal protein S6 kinase (P70S6K)
  • Ribosomal protein S6 kinase alpha 1
  • Ribosomal protein S6 kinase alpha 2
  • Ribosomal protein S6 kinase alpha 5
  • Ribosomal protein S6 kinase alpha 6
  • Ribosomal protein S6 kinase alpha-3
  • Serine/threonine protein kinase NLK
  • Serine/threonine-protein kinase 10
  • Serine/threonine-protein kinase 11
  • Serine/threonine-protein kinase 33
  • Serine/threonine-protein kinase 4 (STK4)
  • Serine/threonine-protein kinase AKT
  • Serine/threonine-protein kinase AKT2
  • Serine/threonine-protein kinase CHK2
  • Serine/threonine-protein kinase Chk1/2
  • Serine/threonine-protein kinase D1
  • Serine/threonine-protein kinase D2
  • Serine/threonine-protein kinase MARK1
  • Serine/threonine-protein kinase NEK7
  • Serine/threonine-protein kinase Nek2
  • Serine/threonine-protein kinase PAK6
  • Serine/threonine-protein kinase PLK1
  • Serine/threonine-protein kinase PLK3
  • Serine/threonine-protein kinase RIPK2
  • Serine/threonine-protein kinase SRPK3
  • Serine/threonine-protein kinase Sgk1
  • Serine/threonine-protein kinase Sgk2
  • Serine/threonine-protein kinase Sgk3
  • Serine/threonine-protein kinase TAO1
  • Serine/threonine-protein kinase TBK1
  • Serine/threonine-protein kinase ULK2
  • Serine/threonine-protein kinase VRK2
  • Serine/threonine-protein kinase WNK2
  • Serine/threonine-protein kinase haspin
  • Serine/threonine-protein kinase pim-1
  • Testis-specific serine/threonine-protein kinase 1
  • Tyrosine kinase non-receptor protein 2
  • Tyrosine-protein kinase ABL1
  • Tyrosine-protein kinase ABL2
  • Tyrosine-protein kinase BRK
  • Tyrosine-protein kinase Blk
  • Tyrosine-protein kinase CSK
  • Tyrosine-protein kinase Fes/Fps
  • Tyrosine-protein kinase HCK
  • Tyrosine-protein kinase ITK/TSK
  • Tyrosine-protein kinase JAK2
  • Tyrosine-protein kinase Lyn
  • Tyrosine-protein kinase Mer
  • Tyrosine-protein kinase Yes
  • Tyrosine-protein kinase ZAP-70
  • Tyrosine-protein kinase receptor FLT3
  • Tyrosine-protein kinase receptor TYRO3
  • Tyrosine-protein kinase receptor UFO
  • Vascular endothelial growth factor receptor 1
  • Vascular endothelial growth factor receptor 2
  • [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial
  • cGMP-dependent protein kinase
  • p21-Activated kinase 3 (PAK3)
  • CHEMBL2333365