Search by Compound Name


Compound Name:

Compounds Sorted by Binding Data per Compound

1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29
30 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55
56 57 58 59 60 61 62 63 64 65 66 67 68 69 70 71 72 73 74 75 76 77 78 79 80 81
82 83 84 85 86 87 88 89 90 91 92 93 94 95 96 97 98 99 100 101 102 103 104 105
106 107 108 109 110 111 112 113 114 115 116 117 118 119 120 121 122 123 124
125 127 128 129 130 132 133 134 135 136 137 138 139 140 141 143 144 145 146
147 148 149 150 151 153 154 155 156 159 160 161 163 164 165 168 170 171 173
174 176 178 179 183 184 186 188 189 190 191 192 193 196 198 199 200 203 204
205 206 207 208 209 210 216 220 224 226 227 229 232 237 238 241 243 248 252
253 259 261 270 274 276 277 285 291 303 304 313 318 323 325 328 333 335 337
339 341 353 360 361 365 389 393 398 401 413 433 442 444 445 446 447 448 451
453 454 455 457 458 460 463 465 467 473 477 478 482 484 499 504 505 506 517
521 525 543 549 551 554 591 606 663 691 708 796 804 821 825 833 842 847 854
855 861 873 879 883 887 913 914 925 926 938 947 1010 1027 1050 1052 1081 1082
1099 1115 1130 1133 1206 1262 1543 1639 1903 2029
Compounds Sorted Alphabetically
Compound Name (alphabetical)
Enz. Inhib. Data
ITC Data
Binding Targets
Alternate Compound Names
2 Ki 1 EC50
  • Cathepsin B
  • Cathepsin H
  • Kallikrein 7
  • 2-(4-Bromo-phenyl)-2,3-dihydro-1H-quinazolin-4-one
  • 2-(4-bromophenyl)-2,3-dihydro-1H-quinazolin-4-one
  • MLS001212491
  • SMR000515221
  • cid_3117357
3 IC50
  • Cytochrome P450 19A1
  • Thromboxane A2 Synthase (P450 TxA2)
  • 5-(1H-imidazol-1-ylmethyl)-5,6,7,8-tetrahydroquinoline
  • 5-[(Imidazol-1-yl)methyl]-5,6,7,8-tetrahydroquinoline
  • tetrahydroquinoline 45
3 IC50
  • Cytochrome P450 19A1
  • Thromboxane A2 Synthase (P450 TxA2)
  • 5-[2-(1H-imidazol-1-yl)ethyl]quinoline
  • 5-[2-(Imidazol-1-yl)ethyl]quinoline
  • CHEMBL54803
  • quinoline 33
3 IC50
  • Cytochrome P450 19A1
  • Thromboxane A2 Synthase (P450 TxA2)
  • 5-[3-(1H-imidazol-1-yl)propyl]-7,8-dihydroquinoline
  • 5-[3-(Imidazol-1-yl)propyl]-7,8-dihydroquinoline
  • CHEMBL53290
  • dihydroquinoline 50
3 IC50
  • Cytochrome P450 19A1
  • Thromboxane A2 Synthase (P450 TxA2)
  • 1-[(2Z)-2-(6,7-dihydro-1-benzofuran-4(5H)-ylidene)ethyl]-1H-imidazole
  • 1-{2-[(4Z)-4,5,6,7-tetrahydro-1-benzofuran-4-ylidene]ethyl}-1H-imidazole
  • CHEMBL56059
  • Tetrahydrobenzo[b]furan 34Z
3 IC50
  • Cytochrome P450 19A1
  • Thromboxane A2 Synthase (P450 TxA2)
  • 1-[(2E)-2-(6,7-dihydro-1-benzothien-4(5H)-ylidene)ethyl]-1H-imidazole
  • 1-{2-[(4E)-4,5,6,7-tetrahydro-1-benzothiophen-4-ylidene]ethyl}-1H-imidazole
  • CHEMBL57513
  • Tetrahydrobenzo[b]thiophene 35E
3 IC50
  • EBifunctional epoxide hydrolase 2
  • Epoxide hydrolase 1
  • Soluble epoxide hydrolase (sEH)
  • US8501783, 1163
  • US9296693, 2
3 IC50
  • Fibroblast growth factor receptor 4
  • US10189794, Compound I-208
  • US10618902, Compound I-208
  • US9695132, I-208
3 IC50
  • Cytochrome P450 19A1
  • Thromboxane A2 Synthase (P450 TxA2)
  • 1-[(2Z)-2-(6,7-dihydro-1-benzothien-4(5H)-ylidene)ethyl]-1H-imidazole
  • 1-{2-[(4Z)-4,5,6,7-tetrahydro-1-benzothiophen-4-ylidene]ethyl}-1H-imidazole
  • CHEMBL55558
  • tetrahydrobenzo[b]thiophene 35Z
3 IC50
  • Cytochrome P450 19A1
  • Thromboxane A2 Synthase (P450 TxA2)
  • 1-[2-(1-benzothiophen-4-yl)ethyl]-1H-imidazole
  • 1-[2-(Benzo[b]thiophen-4-yl)ethyl]-1H-imidazole
  • Benzo[b]thiophene 32
  • CHEMBL460382
3 Ki
  • Prostaglandin transporter (PGT)
  • TBXA2R
  • (5Z)-7-[(1R,4S,5R,6R)-6-[(1E,3S)-3-hydroxyoct-1-en-1-yl]-2,3-dioxabicyclo[2.2.1]heptan-5-yl]hept-5-enoic acid
  • (5Z,13E,15S)-9alpha, 11alpha-epidioxy-15-hydroxyprosta-5,13-dienoic acid
  • 9,11-epoxymethano PGH2
  • PGH2
  • Prostaglandin H2
2 Ki 1 IC50
  • Cytochrome P450 19A1
  • (2S,15S)-15-methyl-2-[(methylsulfanyl)methyl]tetracyclo[8.7.0.0^{2,7}.0^{11,15}]heptadec-6-ene-5,14-dione
  • CHEMBL101540
  • RU54115 Analog 57
3 IC50
  • Hepatocyte growth factor receptor
  • Phosphodiesterase 3
  • US8507676, 63
  • US9062045, Comparator No. 2
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 1.2
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 1.3
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 1.4
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 1.6
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 1.7
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 1.9
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 1.10
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 1.11
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 1.12
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 1.16
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 1.20
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 1.24
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 1.28
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 1.31
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 1.32
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 1.33
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 1.34
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 1.35
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 1.36
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 1.37
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 1.38
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 1.39
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 1.40
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 1.48
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 1.51
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 1.60
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 1.63
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 2.1
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 1.0
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 3.1
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 3.4
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 3.5
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 3.6
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 3.7
3 IC50
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Vascular endothelial growth factor receptor 2
  • US8507510, 3.8
3 IC50
  • Fibroblast growth factor receptor 4
  • US10189794, Compound I-118
  • US10774052, Compound I-118
  • US9695132, I-118
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 1
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 2
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 3
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 4
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 5
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 6
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 7
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 8
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 9
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 10
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 11
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 12
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 14
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 15
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 16
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 22
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 23
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 24
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 25
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 27
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 28
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 29
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 30
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 31
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 32
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 33
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 34
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 35
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 36
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 37
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 38
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 39
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 40
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 41
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 42
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 43
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 44
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 45
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 46
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 47
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 48
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 49
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 50
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 51
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 52
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 53
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 54
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 55
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 56
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 58
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 59
3 Ki
  • Amine oxidase (flavin-containing) A
  • Amine oxidase [flavin-containing] B
  • Lysine-specific histone demethylase 1A
  • US8524717, 60
3 IC50
  • Cathepsin D
  • HIV-1 Protease
  • CHEMBL168640
  • lysine sulfonamide analogue 13
  • lysine sulfonamide analogue 13RS
  • lysine sulfonamide analogue 13SS
  • lysine sulfonamide analogue 13c
  • methyl N-[(1S)-1-{[(5R)-5-[(4-aminobenzene)(2-methylpropyl)sulfonamido]-6-hydroxyhexyl]carbamoyl}-2,2-diphenylethyl]carbamate
  • methyl N-[(1S)-1-{[(5S)-5-[(4-aminobenzene)(2-methylpropyl)sulfonamido]-6-hydroxyhexyl]carbamoyl}-2,2-diphenylethyl]carbamate
2 Ki 1 EC50
  • Delta-type opioid receptor
  • Serine/threonine-protein kinase PAK 4
  • US8530494, 11
  • US8530652, 53
  • US8530652, 98
2 Ki 1 EC50
  • Serine/threonine-protein kinase PAK 4
  • US8530494, 29
  • US8530494, 7
  • US8530652, 57
3 IC50
  • Deoxyuridine 5'-triphosphate nucleotidohydrolase (dUTPase)
  • CHEMBL2057911
  • US8530490, 8
3 IC50
  • Deoxyuridine 5'-triphosphate nucleotidohydrolase (dUTPase)
  • CHEMBL2057600
  • US8530490, 26
3 IC50
  • SRSF protein kinase 1 (SRPK1)
  • Serine/threonine-protein kinase SRPK1
  • US10696661, Compound 74
  • US9695160, 42
  • US9796707, Compound 42
2 IC50 1 EC50
  • Deoxyuridine 5'-triphosphate nucleotidohydrolase (dUTPase)
  • CHEMBL2147986
  • US8530490, 105
3 IC50
  • Deoxyuridine 5'-triphosphate nucleotidohydrolase (dUTPase)
  • CHEMBL2057599
  • US8530490, 159
2 IC50 1 EC50
  • Deoxyuridine 5'-triphosphate nucleotidohydrolase (dUTPase)
  • CHEMBL2147972
  • US8530490, 176
2 IC50 1 EC50
  • Deoxyuridine 5'-triphosphate nucleotidohydrolase (dUTPase)
  • CHEMBL2147974
  • US8530490, 177
2 IC50 1 EC50
  • Deoxyuridine 5'-triphosphate nucleotidohydrolase (dUTPase)
  • CHEMBL2147975
  • US8530490, 178
1 Ki 2 Kd
  • Orexin receptor type 1
  • Orexin receptor type 2
  • US8530648, 10
3 Ki
  • Caspase-3
  • Caspase-7
  • Caspase-8
  • 2-(2,3-dihydro-1,4-benzodioxin-2-yl)-4-[3-(trifluoromethyl)phenyl]-1,3-thiazole
  • BI-9B12
  • Burnham Institute Compound 1
1 Ki 2 IC50
  • Caspase-3
  • Caspase-7
  • Caspase-8
  • BI-7E7
  • Burnham Institute Compound 2
  • ethyl 2-(2,3-dihydro-1,4-benzodioxin-2-yl)-1,3-thiazole-4-carboxylate
3 IC50
  • Caspase-3
  • Caspase-7
  • Caspase-8
  • 2-(2,3-dihydro-1,4-benzodioxin-2-yl)-N-(furan-2-ylmethyl)-1,3-thiazole-4-carboxamide
  • BI-9C8
  • Burnham Institute Compound 3
3 IC50
  • Caspase-3
  • Caspase-7
  • Caspase-8
  • BI-9C3
  • Burnham Institute Compound 4
  • phenyl 2-(2,3-dihydro-1,4-benzodioxin-2-yl)-1,3-thiazole-4-carboxylate
3 IC50
  • Caspase-3
  • Caspase-7
  • Caspase-8
  • BI-9B11
  • Burnham Institute Compound 5
  • [2-(2,3-dihydro-1,4-benzodioxin-2-yl)-1,3-thiazol-4-yl](thiophen-2-ylsulfanyl)methanone
3 IC50
  • Caspase-3
  • Caspase-7
  • Caspase-8
  • 2-(2,3-dihydro-1,4-benzodioxin-2-yl)-1,3-thiazole-4-carboxylic acid
  • BI-9C1
  • Burnham Institute Compound 6
3 IC50
  • Caspase-3
  • Caspase-7
  • Caspase-8
  • 2-(2,3-dihydro-1,4-benzodioxin-2-yl)-N,N-dimethyl-1,3-thiazole-4-carboxamide
  • BI-9C7
  • Burnham Institute Compound 7
1 Ki 2 Kd
  • Orexin receptor type 1
  • Orexin receptor type 2
  • US8530648, 148
3 IC50
  • Caspase-3
  • Caspase-7
  • Caspase-8
  • 4-chlorophenyl 2-(2,3-dihydro-1,4-benzodioxin-2-yl)-1,3-thiazole-4-carboxylate
  • BI-9C4
  • Burnham Institute Compound 8
3 IC50
  • Caspase-3
  • Caspase-7
  • Caspase-8
  • BI-9C5
  • Burnham Institute Compound 9
  • ethyl 2-(2,3-dihydro-1,4-benzodioxin-2-yl)-4-methyl-1,3-thiazole-5-carboxylate
3 IC50
  • Caspase-3
  • Caspase-7
  • Caspase-8
  • 4-{[2-(2,3-dihydro-1,4-benzodioxin-2-yl)-1,3-thiazol-4-yl]carbonyl}morpholine
  • BI-9C2
  • Burnham Institute Compound 10
3 IC50
  • Caspase-3
  • Caspase-7
  • Caspase-8
  • 2-(2,3-dihydro-1,4-benzodioxin-2-yl)-4-methyl-1,3-thiazole-5-carboxylic acid
  • BI-9C6
  • Burnham Institute Compound 11
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