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Compounds Sorted by Binding Data per Compound

1 2 3 4 5 6 7 8 9 10 11 12 13 14 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29
30 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 49 50 51 52 53 54 55
56 57 58 59 60 61 62 63 64 65 66 67 68 69 70 71 72 73 74 75 76 77 78 79 80 81
82 83 84 85 86 87 88 89 90 91 92 93 94 95 96 97 98 99 100 101 102 103 104 105
106 107 108 109 110 111 112 113 114 115 116 117 118 119 120 121 122 123 124
125 127 128 129 130 132 133 134 135 136 137 138 139 140 141 143 144 145 146
147 148 149 150 151 153 154 155 156 159 160 161 163 164 165 168 170 171 173
174 176 178 179 183 184 186 188 189 190 191 192 193 196 198 199 200 203 204
205 206 207 208 209 210 216 220 224 226 227 229 232 237 238 241 243 248 252
253 259 261 270 274 276 277 285 291 303 304 313 318 323 325 328 333 335 337
339 341 353 360 361 365 389 393 398 401 413 433 442 444 445 446 447 448 451
453 454 455 457 458 460 463 465 467 473 477 478 482 484 499 504 505 506 517
521 525 543 549 551 554 591 606 663 691 708 796 804 821 825 833 842 847 854
855 861 873 879 883 887 913 914 925 926 938 947 1010 1027 1050 1052 1081 1082
1099 1115 1130 1133 1206 1262 1543 1639 1903 2029
Compounds Sorted Alphabetically
Compound Name (alphabetical)
Enz. Inhib. Data
ITC Data
Binding Targets
Alternate Compound Names
69 Ki 3 IC50 2 Kd 1 EC50
  • 5-HT5B
  • 5-hydroxytryptamine receptor 1B
  • 5-hydroxytryptamine receptor 1D
  • 5-hydroxytryptamine receptor 2A
  • 5-hydroxytryptamine receptor 2B
  • 5-hydroxytryptamine receptor 2C
  • 5-hydroxytryptamine receptor 3A
  • 5-hydroxytryptamine receptor 4 (5-HT4)
  • 5-hydroxytryptamine receptor 5A
  • 5-hydroxytryptamine receptor 7
  • HTR3A
  • HTR4
  • HTR5A
  • Neuronal acetylcholine receptor
  • Serotonin (5-HT) receptor
  • Serotonin 3 receptor (5HT3)
  • Serotonin 3a (5-HT3a)/3b (5-HT3b) receptor
  • Serotonin receptor 2a and 2c (5HT2A and 5HT2C)
  • (zacopride)4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3-yl)-5-chloro-2-methoxy-benzamide
  • 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3-yl)-5-chloro-2-methoxy-benzamide
  • 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3-yl)-5-chloro-2-methoxy-benzamide (Zacopride)
  • 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3-yl)-5-chloro-2-methoxy-benzamide(zacopride)
  • CHEMBL18041
  • HTR5A4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3-yl)-5-chloro-2-methoxy-benzamide
  • ZACOPRIDE
  • ZACOPRIDE,R
  • ZACOPRIDE,RS
  • ZACOPRIDE,S
75 IC50
  • 5-hydroxytryptamine receptor 1A
  • 5-hydroxytryptamine receptor 1B
  • 5-hydroxytryptamine receptor 2A
  • 5-hydroxytryptamine receptor 2C
  • 5-hydroxytryptamine receptor 3A
  • 5-hydroxytryptamine receptor 5A
  • 5-hydroxytryptamine receptor 6
  • 5-hydroxytryptamine receptor 7
  • Adenosine receptor A1
  • Adenosine receptor A2a
  • Adenosine receptor A3
  • Adrenergic alpha1B
  • Alpha-2A adrenergic receptor
  • Alpha-2B adrenergic receptor
  • C-C chemokine receptor type 1
  • C-X-C chemokine receptor type 2
  • Cannabinoid receptor 1
  • Cannabinoid receptor 2
  • Cholecystokinin receptor
  • D(1A) dopamine receptor
  • D(1B) dopamine receptor
  • D(2) dopamine receptor
  • D(3) dopamine receptor
  • Delta-type opioid receptor
  • Endothelin-1 receptor
  • Histamine H1 receptor
  • Histamine H2 Receptor
  • KCNQ (Kv7) potassium channel
  • Kappa-type opioid receptor
  • Mu-type opioid receptor
  • Muscarinic acetylcholine receptor M1
  • Muscarinic acetylcholine receptor M2
  • Muscarinic acetylcholine receptor M3
  • Muscarinic acetylcholine receptor M4
  • Muscarinic acetylcholine receptor M5
  • Nociceptin receptor
  • P2X purinoceptor 2
  • P2X purinoceptor 3
  • Potassium voltage-gated channel subfamily H member 2
  • Purinergic receptor P2Y2
  • Sigma non-opioid intracellular receptor 1
  • Sodium channel protein type 10 subunit alpha
  • Sodium channel protein type 2 alpha subunit
  • Sodium channel protein type 5 subunit alpha
  • Sodium channel protein type 9 subunit alpha
  • Sodium channel protein type X alpha subunit
  • Transient receptor potential cation channel subfamily V member 1
  • Translocator protein
  • Voltage-gated calcium channel subunit alpha Cav2.2
  • Voltage-gated sodium channel subunit alpha Nav1.3 (Nav1.3)
  • Voltage-gated sodium channel subunit alpha Nav1.8
  • 5-(4-chlorophenyl)-N-(3,5-dimethoxyphenyl)furan-2-carboxamide
  • A-803467
  • CHEMBL250699
75 IC50
  • 72 kDa type IV collagenase
  • Angiotensin-converting enzyme
  • Beta-secretase 1
  • Calpain1/2
  • Caspase-1
  • Caspase-10
  • Caspase-14
  • Caspase-2
  • Caspase-3
  • Caspase-4
  • Caspase-5
  • Caspase-6
  • Caspase-7
  • Caspase-8
  • Caspase-9
  • Cathepsin B
  • Cathepsin D
  • Cathepsin E
  • Cathepsin K
  • Cathepsin L2
  • Cathepsin S
  • Cathepsin Z
  • Chymase
  • Coagulation factor X
  • Coagulation factor XI
  • Collagenase 3
  • Dipeptidyl peptidase 4
  • Dipeptidyl peptidase 9
  • Dipeptidyl peptidase I
  • Dipeptidyl peptidase VIII
  • Disintegrin and metalloproteinase domain-containing protein 10 (ADAM10)
  • Disintegrin and metalloproteinase domain-containing protein 17
  • Disintegrin and metalloproteinase domain-containing protein 9 (ADAM9)
  • Elastase
  • Interstitial collagenase
  • Kallikrein 4
  • Kallikrein 5
  • Kallikrein 8
  • Matrix metalloproteinase 10
  • Matrix metalloproteinase 11
  • Matrix metalloproteinase-12 (MMP12)
  • Matrix metalloproteinase-14 (MMP14)
  • Matrix metalloproteinase-7 (MMP7)
  • Matrix metalloproteinase-9
  • Neutrophil collagenase
  • Papain
  • Plasma kallikrein
  • Plasminogen
  • Pro-cathepsin H
  • Prothrombin
  • Renin
  • Stromelysin-1
  • Trypsin
  • Tryptase
  • Urokinase-type plasminogen activator
  • Vitamin K-dependent protein C
  • CHEMBL567893
  • Grassystatin A
75 IC50
  • 3-phosphoinositide dependent protein kinase-1
  • Aurora kinase A/Targeting protein for Xklp2
  • Aurora kinase B
  • Axin-1/Glycogen synthase kinase-3 beta
  • BDNF/NT-3 growth factors receptor
  • CaM kinase IV
  • Casein kinase I isoform delta
  • Cyclin-Dependent Kinase 5 (CDK5)
  • Cyclin-dependent kinase 1
  • Cyclin-dependent kinase 2
  • Death-associated protein kinase 3
  • Dual-specificity tyrosine-phosphorylation regulated kinase 1A
  • Ephrin type-A receptor 2
  • Epidermal growth factor receptor
  • Fibroblast growth factor receptor 1
  • Fibroblast growth factor receptor 3
  • Glycogen synthase kinase-3
  • Hepatocyte growth factor receptor
  • High affinity immunoglobulin gamma Fc receptor I
  • High affinity nerve growth factor receptor
  • Inhibitor of nuclear factor kappa-B kinase subunit alpha
  • Insulin receptor-related protein
  • Interleukin-1 receptor-associated kinase 4
  • LIM domain kinase 1
  • MAP kinase-activated protein kinase 2
  • MAP kinase-activated protein kinase 3
  • Macrophage colony-stimulating factor 1 receptor (CSF1R)
  • Mast/stem cell growth factor receptor Kit
  • Mitogen-activated protein kinase 1
  • Mitogen-activated protein kinase 12
  • Mitogen-activated protein kinase 13 (MAPK13)
  • Mitogen-activated protein kinase 9
  • Mitogen-activated protein kinase kinase kinase 8
  • Non-receptor tyrosine-protein kinase TYK2
  • PAK 1/CDC42
  • Protein kinase C delta type
  • Protein kinase C, eta
  • Protein kinase C, gamma
  • Proto-oncogene tyrosine-protein kinase Src
  • RAC-alpha serine/threonine-protein kinase
  • Receptor protein-tyrosine kinase erbB-4
  • Receptor tyrosine-protein kinase erbB-2
  • Rho-associated protein kinase 1
  • Rho-associated protein kinase 2
  • Ribosomal protein S6 kinase (P70S6K)
  • Ribosomal protein S6 kinase alpha-3
  • Serine/threonine-protein kinase AKT
  • Serine/threonine-protein kinase AKT2
  • Serine/threonine-protein kinase CHK2
  • Serine/threonine-protein kinase Chk1/2
  • Serine/threonine-protein kinase D2
  • Serine/threonine-protein kinase MST2
  • Serine/threonine-protein kinase Nek2
  • Serine/threonine-protein kinase PAK 4
  • Serine/threonine-protein kinase PLK1
  • Serine/threonine-protein kinase PLK3
  • Serine/threonine-protein kinase PLK4
  • Serine/threonine-protein kinase Sgk1
  • Serine/threonine-protein kinase c-TAK1
  • Serine/threonine-protein kinase pim-1
  • Serine/threonine-protein kinase pim-2
  • Tyrosine-protein kinase ABL1
  • Tyrosine-protein kinase Blk
  • Tyrosine-protein kinase Fyn
  • Tyrosine-protein kinase ITK/TSK
  • Tyrosine-protein kinase JAK2
  • Tyrosine-protein kinase JAK3
  • Tyrosine-protein kinase Lck
  • Tyrosine-protein kinase Lyn
  • Tyrosine-protein kinase SYK
  • Tyrosine-protein kinase receptor FLT3
  • Vascular endothelial growth factor receptor 1
  • Vascular endothelial growth factor receptor 2
  • Vascular endothelial growth factor receptor 3
  • 5-(2-aminoethyl)-7-(7-(benzo[b]thiophen-2-yl)-1H-indazol-5-yl)-5H-pyrrolo[3,2-d]pyrimidin-2-amine
  • CHEMBL590109