Target Name
Affinity Link(s)
Article(s)
UniProt
Files
(S)-6-hydroxynicotine oxidase [K287M]
Kd: 1
1
2D 3D TSV 
(S)-6-hydroxynicotine oxidase [N166A]
Kd: 1
1
2D 3D TSV 
(S)-6-hydroxynicotine oxidase [Y311F]
Kd: 1
1
2D 3D TSV 
1-phosphatidylinositol 4,5-bisphosphate phosphodiesterase delta-4
Ki: 1
1
2D 3D TSV 
14-3-3 protein beta/alpha
Kd: 1
1
2D 3D TSV 
14-3-3 protein eta
Kd: 1
1
2D 3D TSV 
14-3-3 protein theta
Kd: 1
1
2D 3D TSV 
2',5'-phosphodiesterase 12
IC50: 2
1
2D 3D TSV 
2-C-methyl-D-erythritol 2,4-cyclodiphosphate synthase, chloroplastic
IC50: 1
1
2D 3D TSV 
2-C-methyl-D-erythritol 4-phosphate cytidylyltransferase
Ki: 1
1
2D 3D TSV 
26S proteasome regulatory subunit 6B
IC50: 1
1
2D 3D TSV 
3-hydroxyanthranilate 3,4-dioxygenase
IC50: 2
1
2D 3D TSV 
3-isopropylmalate dehydrogenase
Ki: 1
1
2D 3D TSV 
3-oxoacyl-[acyl-carrier-protein] synthase 1 [C171Q]
Ki: 1
1
2D 3D TSV 
5'-AMP-activated protein kinase catalytic subunit alpha-1/catalytic subunit alpha-2/subunit beta-1/subunit beta-2/subunit gamma-1/subunit gamma-2/subunit gamma-3
EC50: 1
1
2D 3D TSV 
5'-AMP-activated protein kinase catalytic subunit alpha-1/subunit beta-1/subunit gamma-2
EC50: 1
1
2D 3D TSV 
5'-AMP-activated protein kinase catalytic subunit alpha-1/subunit beta-1/subunit gamma-3
EC50: 1
1
2D 3D TSV 
5'-AMP-activated protein kinase catalytic subunit alpha-1/subunit beta-2/subunit gamma-3
EC50: 1
1
2D 3D TSV 
5'-AMP-activated protein kinase catalytic subunit alpha-2/subunit beta-1/subunit gamma-2
EC50: 1
1
2D 3D TSV 
5'-AMP-activated protein kinase catalytic subunit alpha-2/subunit beta-2/subunit gamma-2
EC50: 1
1
2D 3D TSV 
5'-AMP-activated protein kinase subunit gamma-2
EC50: 1
1
2D 3D TSV 
5-hydroxytryptamine receptor 3A/3C
IC50: 1
1
2D 3D TSV 
5-hydroxytryptamine receptor 3A/3E
IC50: 1
1
2D 3D TSV 
6-phosphogluconolactonase
Kd: 1
1
2D 3D TSV 
7-methylguanosine phosphate-specific 5'-nucleotidase
IC50: 2
1
2D 3D TSV 
Ab N1G9
ITC: 4
1
0
2D 3D TSV 
Acetyl-CoA acetyltransferase, mitochondrial
IC50: 1
1
2D 3D TSV 
Acid-sensing ion channel 1/2
IC50: 1
1
2D 3D TSV 
Actin-related protein 2
IC50: 1
1
2D 3D TSV 
Activation-induced cytidine deaminase
Ki: 1
1
2D 3D TSV 
Acyl-protein thioesterase 1/2
IC50: 1
1
2D 3D TSV 
Acylamino-acid-releasing enzyme
Ki: 1 IC50: 1
1
2D 3D TSV 
Adenosine 3'-phospho 5'-phosphosulfate transporter 1
Ki: 1
1
2D 3D TSV 
Adenylate kinase 4, mitochondrial
Ki: 1
1
2D 3D TSV 
Adiponectin receptor protein 1
Kd: 1
1
2D 3D TSV 
Adiponectin receptor protein 2
Kd: 1
1
2D 3D TSV 
ADP-ribose glycohydrolase MACROD1
Kd: 1
1
2D 3D TSV 
ADP-ribose glycohydrolase MACROD2
Kd: 1
1
2D 3D TSV 
ADP-ribose pyrophosphatase, mitochondrial
IC50: 1
1
2D 3D TSV 
ADP-ribosylation factor 1
Kd: 1
1
2D 3D TSV 
ADP-sugar pyrophosphatase
IC50: 1
1
2D 3D TSV 
AFG3-like protein 2
Kd: 1
1
2D 3D TSV 
Aldo-keto reductase family 1 member B1 [L301M]
IC50: 1
1
2D 3D TSV 
Aldo-keto reductase family 1 member C1 [H222S]
Ki: 1
1
2D 3D TSV 
Aldo-keto reductase family 1 member C1 [L306A]
Ki: 1
1
2D 3D TSV 
Aldo-keto reductase family 1 member C1 [L308A]
Ki: 1
1
2D 3D TSV 
Aldo-keto reductase family 1 member C1 [L54V]
Ki: 1
1
2D 3D TSV 
Alkaline ceramidase 2
IC50: 1
1
2D 3D TSV 
Alpha-1,2-mannosidase/Alpha-1,2-mannosidase family protein/Alpha-1,2-mannosidase, putative/Glycoside hydrolase family 92/Putative alpha-1,2-mannosidase
Ki: 1
1
2D 3D TSV 
Alpha-1,4-glucan:maltose-1-phosphate maltosyltransferase
IC50: 1
1
2D 3D TSV 
Alpha-2A adrenergic/Mu-type opioid receptor
EC50: 1
1
2D 3D TSV 
Alpha-amylase type A isozyme
Ki: 1
1
2D 3D TSV 
Alpha-crystallin A chain
EC50: 1
1
2D 3D TSV 
Alpha-galactosidase C
IC50: 1
1
2D 3D TSV 
Alpha-ketoglutarate-dependent dioxygenase FTO [31-505]
IC50: 1
1
2D 3D TSV 
Amine oxidase [flavin-containing]
Ki: 1
1
2D 3D TSV 
AMP deaminase
IC50: 1
1
2D 3D TSV 
Angiotensinogen
Ki: 1
1
2D 3D TSV 
Antithrombin-III/Coagulation factor X
IC50: 1
1
2D 3D TSV 
AP-1 complex subunit beta-1
Kd: 1
1
2D 3D TSV 
AP-3 complex subunit sigma-2
Ki: 1
1
2D 3D TSV 
apocytochrome b562
ITC: 2
1
2D 3D TSV 
Arachidonate 5-lipoxygenase
IC50: 1
1
2D 3D TSV 
Arginine vasopressin-induced protein 1
Ki: 1
1
2D 3D TSV 
Aspartate ammonia-lyase
Ki: 1
1
2D 3D TSV 
Ataxin-3
IC50: 1
1
2D 3D TSV 
Ataxin-3-like protein
IC50: 1
1
2D 3D TSV 
ATP receptor
Ki: 2
1
2D 3D TSV 
ATP synthase epsilon chain/gamma chain/subunit a/subunit alpha/subunit b/subunit b-delta/subunit beta/subunit c
IC50: 1
1
2D 3D TSV 
ATP-dependent 6-phosphofructokinase, liver type
EC50: 1
1
2D 3D TSV 
ATP-dependent 6-phosphofructokinase, muscle type
EC50: 1
1
2D 3D TSV 
ATP-dependent Clp protease ATP-binding subunit clpX-like, mitochondrial
IC50: 1
1
2D 3D TSV 
Atrial natriuretic peptide receptor 1/2/3
IC50: 1
1
2D 3D TSV 
Atypical chemokine receptor 2
IC50: 1 EC50: 1
1
2D 3D TSV 
Aureobasidin-resistance protein
IC50: 1
1
2D 3D TSV 
Aurora kinase A/Targeting protein for Xklp2
IC50: 1
1
2D 3D TSV 
Aurora kinase B
IC50: 3
3
2D 3D TSV 
Aurora kinase B [2-344]/Inner centromere protein [826-918]
IC50: 1
1
2D 3D TSV 
Avidin
Kd: 1
1
2D 3D TSV 
B-cell CLL/lymphoma 9 protein/Catenin beta-1
Ki: 1
1
2D 3D TSV 
Baculoviral IAP repeat-containing protein 3/Mucosa-associated lymphoid tissue lymphoma translocation protein 1
IC50: 1
1
2D 3D TSV 
Bcl-2 homologous antagonist/killer/Induced myeloid leukemia cell differentiation protein Mcl-1
IC50: 1
1
2D 3D TSV 
BCR/ABL p210 fusion protein
EC50: 1
1
2D 3D TSV 
Beta-chimaerin
Ki: 1
1
2D 3D TSV 
Beta-lactamase OXA-2
IC50: 1
1
2D 3D TSV 
Bifunctional coenzyme A synthase
IC50: 1
1
2D 3D TSV 
Bifunctional cytochrome P450/NADPH--P450 reductase
Kd: 1
1
2D 3D TSV 
Bifunctional methylenetetrahydrofolate dehydrogenase/cyclohydrolase 2, mitochondrial
IC50: 1
1
2D 3D TSV 
BioDB n*138 SEQ ID NO: 2
IC50: 1
1
0
2D 3D TSV 
Bis(5'-nucleosyl)-tetraphosphatase [asymmetrical]
IC50: 1
1
2D 3D TSV 
BRISC and BRCA1-A complex member 1/BRISC and BRCA1-A complex member 2/BRISC complex subunit Abraxas 2/Lys-63-specific deubiquitinase BRCC36
IC50: 1
1
2D 3D TSV 
Bromodomain testis-specific protein [27-133]
IC50: 1
1
2D 3D TSV 
Bromodomain-containing protein 2 [349-450]
IC50: 1
1
2D 3D TSV 
Bromodomain-containing protein 2 [74-180]
IC50: 1
1
2D 3D TSV 
Bromodomain-containing protein 3 [311-412]
IC50: 1
1
2D 3D TSV 
Bromodomain-containing protein 3 [34-140]
IC50: 1
1
2D 3D TSV 
Bromodomain-containing protein 4 [44-166,N140A]
Kd: 2
1
2D 3D TSV 
Bromodomain-containing protein 4 [44-166,Y97F]
Kd: 2
1
2D 3D TSV 
BTB/POZ domain-containing protein KCTD11
Kd: 1
1
2D 3D TSV 
C-terminal processing protease of the D1 protein
Ki: 1
1
2D 3D TSV 
C-terminal-binding protein 1 [A52D]
Kd: 1
1
2D 3D TSV 
C-terminal-binding protein 1 [E295A]
Kd: 1
1
2D 3D TSV 
C-terminal-binding protein 1 [H315A]
Kd: 1
1
2D 3D TSV 
C-terminal-binding protein 1 [R266Q]
Kd: 1
1
2D 3D TSV 
C-terminal-binding protein 1 [V66R]
Kd: 1
1
2D 3D TSV 
C-terminal-binding protein 1 [W318F]
Kd: 1
1
2D 3D TSV 
C-type lectin domain family 4 member C
IC50: 1
1
2D 3D TSV 
C-type lectin domain family 4 member K
IC50: 1
1
2D 3D TSV 
Cadherin-2
IC50: 1
1
2D 3D TSV 
Calcitonin gene-related peptide type 1 receptor/Receptor activity-modifying protein 2
Ki: 1
1
2D 3D TSV 
Calcitonin gene-related peptide type 1 receptor/Receptor activity-modifying protein 3
Ki: 1
1
2D 3D TSV 
Calcium release-activated calcium channel protein 1/Short transient receptor potential channel 1/Short transient receptor potential channel 3/Stromal interaction molecule 1
IC50: 1
1
2D 3D TSV 
Calcium/calmodulin-dependent protein kinase kinase 2 [ P274E]
IC50: 1
1
2D 3D TSV 
Calcium/calmodulin-dependent protein kinase type II subunit alpha/beta
EC50: 1
1
2D 3D TSV 
Calcium/calmodulin-dependent protein kinase type II subunit delta/gamma
EC50: 1
1
2D 3D TSV 
Calcium/calmodulin-dependent protein kinase with a kinase domain and 2 calmodulin-like EF hands
IC50: 1
1
2D 3D TSV 
Calcium/calmodulin-dependent protein kinase with a kinase domain and 4 calmodulin like EF hands
IC50: 1
1
2D 3D TSV 
Calnexin
IC50: 1
1
2D 3D TSV 
cAMP-activated global transcriptional regulator CRP
ITC: 12
1
0
2D 3D TSV 
cAMP-dependent protein kinase catalytic subunit alpha [L49I,T183A]
IC50: 1
1
2D 3D TSV 
cAMP-dependent protein kinase type I-alpha regulatory subunit [K242A]
Kd: 1
1
2D 3D TSV 
cAMP-dependent protein kinase type I-alpha regulatory subunit [K244A]
Kd: 1
1
2D 3D TSV 
cAMP-dependent protein kinase type I-alpha regulatory subunit [R241A]
Kd: 1
1
2D 3D TSV 
cAMP-dependent protein kinase type I-alpha regulatory subunit [R243A]
Kd: 1
1
2D 3D TSV 
cAMP-specific 3',5'-cyclic phosphodiesterase 4A [559-660]
IC50: 1
1
2D 3D TSV 
Carbamate kinase
IC50: 1
1
2D 3D TSV 
Carbonate dehydratase
Ki: 4
1
2D 3D TSV 
Carbonic anhydrase 1 + BH
Ki: 2
1
2D 3D TSV 
Carbonic anhydrase 13 + BH
Ki: 2
1
2D 3D TSV 
Carbonic anhydrase 2/3/4/6
Ki: 1
1
2D 3D TSV 
Carbonic anhydrase 3 + BH
Ki: 2
1
2D 3D TSV 
Carbonic anhydrase 7 + BH
Ki: 2
1
2D 3D TSV 
Cardiac ryanodine receptor 2
Ki: 1
1
2D 3D TSV 
Casein kinase II subunit alpha/alpha 3/alpha'/beta
IC50: 1
1
2D 3D TSV 
Caseinolytic protein C1 (ClpC1 NTD E89A)
Kd: 1 ITC: 1
1
2D 3D TSV 
Caseinolytic protein C1 (ClpC1 NTD E89Q)
Kd: 1 ITC: 1
1
2D 3D TSV 
Caseinolytic protein C1 (ClpC1 NTD F2A)
Kd: 1 ITC: 1
1
2D 3D TSV 
Caseinolytic protein C1 (ClpC1 NTD F2Y)
Kd: 1 ITC: 1
1
2D 3D TSV 
Caseinolytic protein C1 (ClpC1 NTD F80A)
Kd: 1 ITC: 1
1
2D 3D TSV 
Caseinolytic protein C1 (ClpC1 NTD F80Y)
Kd: 1 ITC: 1
1
2D 3D TSV 
Caseinolytic protein C1 (ClpC1 NTD)
Kd: 1 ITC: 1
1
2D 3D TSV 
Caseinolytic protein C1 (ClpC1 NTD-D1)
Kd: 1 ITC: 1
1
2D 3D TSV 
Caspase-1/Caspase-10/Caspase-14/Caspase-2/Caspase-3/Caspase-4/Caspase-5/Caspase-6/Caspase-7/Caspase-8/Caspase-9/Inactive caspase-12
EC50: 1
1
2D 3D TSV 
Caspase-3|IST-1 Complex
ITC: 1
1
2D 3D TSV 
Catenin beta-1/Transcription factor 4
IC50: 1
1
2D 3D TSV 
Catenin beta-1/Transcription factor 7-like 2
IC50: 1
1
2D 3D TSV 
Cathepsin B-like protease
Ki: 1
1
2D 3D TSV 
Caveolin-1
Kd: 1
1
2D 3D TSV 
CCR2 protein
IC50: 1
1
2D 3D TSV 
CD40 ligand
IC50: 1
1
2D 3D TSV 
CDK-activating kinase assembly factor MAT1
IC50: 1
1
2D 3D TSV 
Cell division control protein 28, putative
IC50: 1
1
2D 3D TSV 
Cell division cycle 7-related protein kinase/G2/mitotic-specific cyclin-B1
IC50: 1
1
2D 3D TSV 
Cgd2_1060 protein
IC50: 1
1
2D 3D TSV 
Cgd5_820 protein
IC50: 1
1
2D 3D TSV 
Chaperonin GroEL/Co-chaperonin GroES
IC50: 1
1
2D 3D TSV 
Chemokine (C-C motif) receptor 1
IC50: 1
1
2D 3D TSV 
Chemokine receptor
IC50: 1
1
2D 3D TSV 
Chemotaxis protein CheA
IC50: 1
1
2D 3D TSV 
Chitin synthase 1/2/3
IC50: 1
1
2D 3D TSV 
Chitin synthase 2
IC50: 1
1
2D 3D TSV 
Chromaffin granule amine transporter
Ki: 1
1
2D 3D TSV 
Chromobox protein homolog 3
Kd: 1
1
2D 3D TSV 
Chymotrypsin-C/Chymotrypsin-like protease CTRL-1/Chymotrypsinogen B/Chymotrypsinogen B2
IC50: 1
1
2D 3D TSV 
Coagulation factor XII [20-615]
IC50: 1
1
2D 3D TSV 
Coiled-coil domain-containing protein 6/Proto-oncogene tyrosine-protein kinase receptor Ret
IC50: 1
1
2D 3D TSV 
Complement C2
IC50: 4
1
2D 3D TSV 
Complement factor H
IC50: 1
1
2D 3D TSV 
Corticoliberin
Ki: 1
1
2D 3D TSV 
Cryptochrome-2/Period circadian protein homolog 2
EC50: 1
1
2D 3D TSV 
Cyclin-A2 [171-432]/Cyclin-dependent kinase 2 [F82H]
IC50: 1
1
2D 3D TSV 
Cyclin-A2 [171-432]/Cyclin-dependent kinase 2 [L83V,H84D]
IC50: 1
1
2D 3D TSV 
Cyclin-dependent kinase 1/G2/mitotic-specific cyclin-B1/G2/mitotic-specific cyclin-B2/G2/mitotic-specific cyclin-B3/cAMP-dependent protein kinase
IC50: 1
1
2D 3D TSV 
Cyclin-dependent kinase 10
Kd: 1
1
2D 3D TSV 
Cyclin-dependent kinase 2-associated protein 2
IC50: 1
1
2D 3D TSV 
Cyclin-dependent kinase 20
Kd: 1
1
2D 3D TSV 
Cyclin-dependent kinase 4/G1/S-specific cyclin-D2
IC50: 1
1
2D 3D TSV 
Cyclin-dependent kinase-like 1
IC50: 1
1
2D 3D TSV 
Cyclin-dependent kinase-like 4
IC50: 1
1
2D 3D TSV 
Cyclin-dependent protein kinase PHO85/PHO85 cyclin PHO80/Phosphate system positive regulatory protein PHO81
Ki: 1 IC50: 1
1
2D 3D TSV 
Cyclin-H/Cyclin-dependent kinase 9
IC50: 1
1
2D 3D TSV 
Cyclin-O/Cyclin-dependent kinase 2
IC50: 1
1
2D 3D TSV 
Cyclin-T2/Cyclin-dependent kinase 9
IC50: 1
1
2D 3D TSV 
Cyclin-Y/Cyclin-dependent kinase 14
IC50: 1
1
2D 3D TSV 
Cyclin-Y/Cyclin-dependent kinase 17
IC50: 2
2
2D 3D TSV 
Cyclin-Y/Cyclin-dependent kinase 18
IC50: 1
1
2D 3D TSV 
Cyclin-Y/Cyclin-dependent kinase 2
IC50: 1
1
2D 3D TSV 
Cys-loop ligand-gated ion channel
IC50: 1
1
2D 3D TSV 
Cytochrome P450 2B11
Ki: 2
1
2D 3D TSV 
Cytochrome P450 3A2
Ki: 1
1
2D 3D TSV 
Cytochrome P450 3A6
Ki: 1
1
2D 3D TSV 
Cytochrome P450 3A7
Ki: 1
1
2D 3D TSV 
Cytochrome P450 3A7 [T409R]
IC50: 1
1
2D 3D TSV 
Cytochrome P450 4X1
IC50: 1
1
2D 3D TSV 
Cytochrome P450 71B1
IC50: 1
1
2D 3D TSV 
Cytosol aminopeptidase [435-519]
Ki: 1
1
2D 3D TSV 
Deoxyguanosine kinase, mitochondrial
IC50: 1
1
2D 3D TSV 
DEP domain-containing mTOR-interacting protein
Kd: 1
1
2D 3D TSV 
Deubiquitinase OTUD6B
IC50: 1
1
2D 3D TSV 
Deubiquitinating protein VCPIP1
IC50: 1
1
2D 3D TSV 
Diacylglycerol kinase alpha/zeta
IC50: 1
1
2D 3D TSV 
Diacylglycerol kinase beta
IC50: 1
1
2D 3D TSV 
Diacylglycerol kinase gamma
IC50: 1
1
2D 3D TSV 
Diacylglycerol O-acyltransferase 1 [148-636]
IC50: 1
1
2D 3D TSV 
Dihydrofolate synthase/folylpolyglutamate synthase
Ki: 1
1
2D 3D TSV 
Dihydrolipoyl dehydrogenase, mitochondrial
IC50: 1
1
2D 3D TSV 
Dimer of Gag-Pol polyprotein [489-587,I536L]
Ki: 1
1
2D 3D TSV 
Dimer of Gag-Pol polyprotein [489-587,I539L]
Ki: 1
1
2D 3D TSV 
Dimer of Gag-Pol polyprotein [489-587,I573V]
Ki: 1
1
2D 3D TSV 
Dimer of Gag-Pol polyprotein [489-587,L512I]
Ki: 1
1
2D 3D TSV 
Dimer of Gag-Pol polyprotein [489-587,L512V]
Ki: 1
1
2D 3D TSV 
Dimer of Gag-Pol polyprotein [489-587,L565M]
Ki: 1
1
2D 3D TSV 
Dimer of Gag-Pol polyprotein [489-587,V521I]
Ki: 1
1
2D 3D TSV 
Dimer of Gag-Pol polyprotein [489-587,V571I]
Ki: 1
1
2D 3D TSV 
Dimer of Gag-Pol polyprotein [501-599,A572V,V583T,I585V]
Ki: 1
1
2D 3D TSV 
Dimer of Prostaglandin G/H synthase 2
Kd: 1
1
2D 3D TSV 
Dimer of Prostaglandin G/H synthase 2 [R120A]
Kd: 1
1
2D 3D TSV 
Dimer of Prostaglandin G/H synthase 2 [R120Q]
Kd: 1
1
2D 3D TSV 
Dimer of Prostaglandin G/H synthase 2 [S530A]
Kd: 1
1
2D 3D TSV 
Dimer of Prostaglandin G/H synthase 2 [Y385F]
Kd: 1
1
2D 3D TSV 
Dimer of Retinoic acid receptor RXR-alpha
Kd: 2
1
2D 3D TSV 
Dimer of Type-1 angiotensin II receptor
Ki: 1
1
2D 3D TSV 
Dipeptidyl carboxypeptidase
IC50: 1
1
2D 3D TSV 
Dipeptidyl peptidase 9 [D301A]
Ki: 1
1
2D 3D TSV 
Dipeptidyl peptidase 9 [E286A,E297A]
Ki: 1
1
2D 3D TSV 
Dipeptidyl peptidase 9 [E286A]
Ki: 1
1
2D 3D TSV 
Dipeptidyl peptidase 9 [H289A]
Ki: 1
1
2D 3D TSV 
Dipeptidyl peptidase 9 [I288A]
Ki: 1
1
2D 3D TSV 
Dipeptidyl peptidase 9 [K299A]
Ki: 1
1
2D 3D TSV 
Dipeptidyl peptidase 9 [L295A]
Ki: 1
1
2D 3D TSV 
Dipeptidyl peptidase 9 [R298A]
Ki: 1
1
2D 3D TSV 
Dipeptidyl peptidase 9 [S292A]
Ki: 1
1
2D 3D TSV 
Dipeptidyl peptidase 9 [V285A]
Ki: 1
1
2D 3D TSV 
Dipeptidyl peptidase 9 [V290A]
Ki: 1
1
2D 3D TSV 
Dipeptidyl peptidase 9 [Y277A]
Ki: 1
1
2D 3D TSV 
Dipeptidyl peptidase 9 [Y303D]
Ki: 1
1
2D 3D TSV 
Dipeptidyl peptidase 9 [Y305A]
Ki: 1
1
2D 3D TSV 
Dipeptidyl peptidase 9 [Y305D]
Ki: 1
1
2D 3D TSV 
DNA (cytosine-5)-methyltransferase 1 [351-1600]
IC50: 1
1
2D 3D TSV 
DNA (cytosine-5)-methyltransferase 3-like/3A
IC50: 1
1
2D 3D TSV 
DNA (cytosine-5)-methyltransferase 3-like/3B
IC50: 1
1
2D 3D TSV 
DNA (cytosine-5)-methyltransferase 3A [590-912]
IC50: 1
1
2D 3D TSV 
DNA damage-binding protein 1
IC50: 1
1
2D 3D TSV 
DNA excision repair protein ERCC-1/repair endonuclease XPF
Kd: 1
1
2D 3D TSV 
DNA ligase 4
IC50: 1
1
2D 3D TSV 
DNA primase TraC
IC50: 1
1
2D 3D TSV 
DNA repair and recombination protein RAD54-like
EC50: 1
1
2D 3D TSV 
DNA topoisomerase type IB small subunit
Kd: 1
1
2D 3D TSV 
DNA-binding protein Ikaros/Protein cereblon
EC50: 1
1
2D 3D TSV 
DNA-dependent protein kinase catalytic subunit/Ephrin type-B receptor 4
IC50: 1
1
2D 3D TSV 
DNA-dependent protein kinase catalytic subunit/Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform
IC50: 2
1
2D 3D TSV 
DNA-dependent protein kinase catalytic subunit/Platelet-derived growth factor receptor beta [525-1106]
IC50: 1
1
2D 3D TSV 
DNA-dependent protein kinase catalytic subunit/Proto-oncogene tyrosine-protein kinase Src
IC50: 2
1
2D 3D TSV 
DNA-dependent protein kinase catalytic subunit/Receptor protein-tyrosine kinase
IC50: 1
1
2D 3D TSV 
DNA-dependent protein kinase catalytic subunit/Tyrosine-protein kinase ABL1
IC50: 1
1
2D 3D TSV 
DNA-dependent protein kinase catalytic subunit/Tyrosine-protein kinase HCK
IC50: 1
1
2D 3D TSV 
DNA-dependent protein kinase catalytic subunit/Vascular endothelial growth factor receptor 2
IC50: 1
1
2D 3D TSV 
DNA-directed RNA polymerase subunit alpha/beta/beta'/omega
IC50: 1
1
2D 3D TSV 
dTDP-4-dehydrorhamnose 3,5-epimerase/reductase
IC50: 1
1
2D 3D TSV 
Dual specificity protein kinase CLK1/CLK2
IC50: 1
1
2D 3D TSV 
Dual specificity protein phosphatase 14
IC50: 1
1
2D 3D TSV 
Dual specificity protein phosphatase 2
IC50: 1
1
2D 3D TSV 
Dual specificity tyrosine-phosphorylation-regulated kinase 2 [393-601]
IC50: 1
1
2D 3D TSV 
E3 ubiquitin-protein ligase RNF31/RanBP-type and C3HC4-type zinc finger-containing protein 1/Sharpin
IC50: 1
1
2D 3D TSV 
E3 ubiquitin-protein ligase XIAP [124-240,C202A,C213G]
IC50: 1
1
2D 3D TSV 
Ecdysone receptor/Gene regulation protein
Ki: 1
1
2D 3D TSV 
Ecdysone receptor/Nuclear receptor RXR-l
Ki: 1
1
2D 3D TSV 
Ecdysone receptor/Protein ultraspiracle
EC50: 1
1
2D 3D TSV 
Ecdysone receptor/Protein ultraspiracle homolog
Ki: 1
1
2D 3D TSV 
Ecdysone receptor/Ultraspiracle isoform-A
EC50: 1
1
2D 3D TSV 
Ecdysone receptor/USP
Ki: 1
1
2D 3D TSV 
Ectonucleotide pyrophosphatase/phosphodiesterase 2
IC50: 1
1
2D 3D TSV 
Elongin-B/Elongin-C/von Hippel-Lindau disease tumor suppressor
IC50: 1
1
2D 3D TSV 
Endochitinase B1 [D246A]
Kd: 1
1
2D 3D TSV 
Endochitinase B1 [E177A]
Kd: 1
1
2D 3D TSV 
Endopolygalacturonase
Kd: 1
1
2D 3D TSV 
Ephrin type-A receptor 3 ligand binding domain (EphA3-LBD)
Kd: 1 ITC: 1
1
2D 3D TSV 
Ephrin type-A receptor 4 ligand binding domain (D61G/E62G-EphA4-LBD)
Kd: 1 ITC: 1
1
2D 3D TSV 
Ephrin type-A receptor 4 ligand binding domain (I159A-EphA4-LBD)
Kd: 1 ITC: 1
1
2D 3D TSV 
Ephrin type-A receptor 4 ligand binding domain (I59A-EphA4-LBD)
Kd: 1 ITC: 1
1
2D 3D TSV 
Ephrin type-A receptor 4 ligand binding domain (I59G-EphA4-LBD)
Kd: 1 ITC: 1
1
2D 3D TSV 
Ephrin type-A receptor 4 ligand binding domain (I67A-EphA4-LBD)
Kd: 1 ITC: 1
1
2D 3D TSV 
Ephrin type-A receptor 4 ligand binding domain (M164A-EphA4-LBD)
Kd: 1 ITC: 1
1
2D 3D TSV 
Ephrin type-A receptor 4 ligand binding domain (M60A-EphA4-LBD)
Kd: 1 ITC: 1
1
2D 3D TSV 
Ephrin type-B receptor 4/Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
IC50: 1
1
2D 3D TSV 
Ephrin type-B receptor 4/Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
IC50: 1
1
2D 3D TSV 
Ephrin type-B receptor 4/Serine/threonine-protein kinase mTOR
IC50: 1
1
2D 3D TSV 
Epidermal growth factor receptor [1-746,748-748,750-1210,A750P]
Kd: 1
1
2D 3D TSV 
Epidermal growth factor receptor [1-746,748-750,752-1210]
Kd: 1
1
2D 3D TSV 
Epidermal growth factor receptor [1-746,748-751,753-1210,P753S]
Kd: 1
1
2D 3D TSV 
Epsin-1
IC50: 2
2
2D 3D TSV 
Estrogen-Related Receptor, alpha Mutant (C325S)
ITC: 1
1
0
2D 3D TSV 
ETS translocation variant 1
Kd: 1
1
2D 3D TSV 
Eukaryotic peptide chain release factor GTP-binding subunit
IC50: 1 EC50: 1
1
2D 3D TSV 
EWS-Fli1 protein
Kd: 1
1
2D 3D TSV 
Exo-1,4-beta-xylosidase xlnD
Ki: 1
1
2D 3D TSV 
Extracellular serine/threonine protein kinase FAM20C
IC50: 1
1
2D 3D TSV 
FAD-Binding Domain
ITC: 1
1
2D 3D TSV 
Fanconi anemia group F protein
Kd: 1
1
2D 3D TSV 
Ferrochelatase, mitochondrial
EC50: 1
1
2D 3D TSV 
Fibroblast growth factor receptor 2 [406-821]
IC50: 1
1
2D 3D TSV 
FimH
Kd: 1
1
2D 3D TSV 
FMN_red domain-containing protein
Ki: 1
1
2D 3D TSV 
FMRFamide-like neuropeptides 14
Ki: 1
1
2D 3D TSV 
Forkhead box protein O3
Kd: 1
1
2D 3D TSV 
Friend leukemia integration 1 transcription factor/RNA-binding protein EWS
IC50: 1
1
2D 3D TSV 
Frizzled-8
Kd: 1
1
2D 3D TSV 
FYVE, RhoGEF and PH domain-containing protein 1
Ki: 1
1
2D 3D TSV 
G protein-activated inward rectifier potassium channel 1/2
IC50: 1
1
2D 3D TSV 
G protein-activated inward rectifier potassium channel 1/4
EC50: 1
1
2D 3D TSV 
G-protein coupled receptor 135
EC50: 1
1
2D 3D TSV 
G-protein coupled receptor 37-like 1
IC50: 1
1
2D 3D TSV 
G-protein coupled receptor 81
EC50: 1
1
2D 3D TSV 
G1/S-specific cyclin-D2
IC50: 2
2
2D 3D TSV 
G1/S-specific cyclin-D3
IC50: 1
1
2D 3D TSV 
Gag-Pol polyprotein [K103N]
IC50: 2
1
2D 3D TSV 
Galactofuranosyltransferase GlfT2
IC50: 1
1
2D 3D TSV 
Gamma-aminobutyric acid receptor subunit alpha-1 [28-456]/beta-2 [26-512]/gamma-2 [40-467,F116C]
Other: 1
1
2D 3D TSV 
Gamma-aminobutyric acid receptor subunit alpha-1 [D97C]/beta-2 [26-512]/gamma-2 [40-467]
Other: 1
1
2D 3D TSV 
Gamma-aminobutyric acid receptor subunit alpha-1 [Y209C]/beta-2 [26-512]/gamma-2 [40-467]
Other: 1
1
2D 3D TSV 
Gamma-aminobutyric acid receptor subunit alpha-1/beta-1
Ki: 1
1
2D 3D TSV 
Gamma-aminobutyric acid receptor subunit alpha-1/gamma-2
IC50: 1
1
2D 3D TSV 
Gamma-aminobutyric acid receptor subunit alpha-4/beta-2/delta
EC50: 1
1
2D 3D TSV 
Gamma-aminobutyric acid receptor subunit alpha-4/beta-3
IC50: 1 EC50: 1
1
2D 3D TSV 
Gamma-aminobutyric acid receptor subunit gamma-2
EC50: 1
1
2D 3D TSV 
GDH/6PGL endoplasmic bifunctional protein
IC50: 1
1
2D 3D TSV 
Genome polyprotein [1027-1207,A156T]
IC50: 1
1
2D 3D TSV 
Genome polyprotein [2420-3010,C2735L]
Kd: 1 Koff: 1 Kon: 1
1
2D 3D TSV 
Genome polyprotein [2420-3010,L2811I]
Kd: 1 Koff: 1 Kon: 1
1
2D 3D TSV 
Genome polyprotein [2420-3010,M2833T]
Kd: 1 Koff: 1 Kon: 1
1
2D 3D TSV 
Genome polyprotein [2420-3010,M2842T]
Kd: 1 Koff: 1 Kon: 1
1
2D 3D TSV 
Genome polyprotein [2420-3010,P2914L]
Kd: 2 Koff: 2 Kon: 2
1
2D 3D TSV 
Genome polyprotein [2420-3010,S2701T]
Kd: 1 Koff: 1 Kon: 1
1
2D 3D TSV 
Genome polyprotein [2420-3010,V2913A]
Kd: 1 Koff: 1 Kon: 1
1
2D 3D TSV 
Geranylgeranyl pyrophosphate synthase BTS1 [Y107A,F108A]
IC50: 1
1
2D 3D TSV 
Geranylgeranyl transferase type-2 subunit alpha/beta
IC50: 1
1
2D 3D TSV 
Glucagon receptor [1-477]
IC50: 1
1
2D 3D TSV 
Glucoamylase
Ki: 1 IC50: 1
1
2D 3D TSV 
Glucoamylase 1
Ki: 1 IC50: 1
1
2D 3D TSV 
Glucose-1-phosphate cytidylyltransferase
Ki: 1
1
2D 3D TSV 
Glucose-6-phosphate isomerase
Ki: 1
1
2D 3D TSV 
Glutamate decarboxylase 2
Ki: 1
1
2D 3D TSV 
Glutamate receptor ionotropic, NMDA 1 [F484A,T518L]/3A
Ki: 1 IC50: 1
1
2D 3D TSV 
Glutamate receptor ionotropic, NMDA 1 [F484A,T518L]/3B
Ki: 1 IC50: 1
1
2D 3D TSV 
Glutamate receptor-interacting protein 1
Ki: 1
1
2D 3D TSV 
Glutamate--cysteine ligase
Ki: 1
1
2D 3D TSV 
Glutaredoxin-1
Ki: 1
1
2D 3D TSV 
Glutathione S-transferase theta-1
Ki: 1
1
2D 3D TSV 
Glutathione transferase
IC50: 1
1
2D 3D TSV 
Glycine receptor subunit alpha-2/beta
IC50: 1
1
2D 3D TSV 
Glycogen [starch] synthase, liver
EC50: 2
1
2D 3D TSV 
Glycoprotein IIb/Integrin beta
IC50: 1
1
2D 3D TSV 
Glyoxylate Regulatory Protein (C-AllR)
ITC: 1
1
2D 3D TSV 
GRB10-interacting GYF protein 2
Kd: 1
1
2D 3D TSV 
Growth factor receptor-bound protein 10
Kd: 1
1
2D 3D TSV 
Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2/G(I)/G(S)/G(T) subunit beta-1
IC50: 1
1
2D 3D TSV 
Guanine nucleotide-binding protein G(q) subunit alpha/subunit alpha-11
IC50: 1
1
2D 3D TSV 
Heme oxygenase HutZ [D132E]
Kd: 2
1
2D 3D TSV 
Heme oxygenase HutZ [D132L]
Kd: 1
1
2D 3D TSV 
Heme oxygenase HutZ [D132N]
Kd: 2
1
2D 3D TSV 
Heme-binding protein HutZ
Kd: 2
1
2D 3D TSV 
Hepatocyte growth factor
Kd: 1
1
2D 3D TSV 
Hepatocyte growth factor receptor [1078-1345,D1228H,L1272V]
Ki: 1
1
2D 3D TSV 
Hepatocyte growth factor receptor [1078-1345,H1094R,L1272V]
Ki: 1
1
2D 3D TSV 
Hepatocyte growth factor receptor [1078-1345,M1250T,L1272V]
Ki: 1
1
2D 3D TSV 
Hepatocyte growth factor receptor [1078-1345,V1092I,L1272V]
Ki: 1
1
2D 3D TSV 
Hepatocyte growth factor receptor [1078-1345,Y1230H,L1272V]
Ki: 1
1
2D 3D TSV 
Hepatocyte growth factor receptor/Nucleoprotein TPR
IC50: 1
1
2D 3D TSV 
Heterogeneous nuclear ribonucleoprotein A1
Kd: 1
1
2D 3D TSV 
High affinity cAMP-specific and IBMX-insensitive 3',5'-cyclic phosphodiesterase 8A/8B
IC50: 1
1
2D 3D TSV 
Histidine decarboxylase
Ki: 1
1
2D 3D TSV 
Histidine--tRNA ligase, cytoplasmic
IC50: 1
1
2D 3D TSV 
Histidine-binding periplasmic protein [1-238]
Kd: 1 ITC: 1
1
2D 3D TSV 
Histone deacetylase 1/3/4/6/7
IC50: 1
1
2D 3D TSV 
Histone deacetylase 6 [440-798,S531A]
Kd: 1
1
2D 3D TSV 
Histone deacetylase 6 [60-420,H82F,F202Y]
Kd: 1
1
2D 3D TSV 
Histone deacetylase 6 [84-835,H255V]
Kd: 1
1
2D 3D TSV 
Histone deacetylase 6 [84-835,H651V]
Kd: 1
1
2D 3D TSV 
Histone deacetylase 8 [R223M]
IC50: 1
1
2D 3D TSV 
Histone demethylase UTY [818-1347,P1214I]
Kd: 1
1
2D 3D TSV 
Histone demethylase UTY [818-1347,S1138G]
Kd: 1
1
2D 3D TSV 
Histone demethylase UTY [818-1347]
Kd: 1
1
2D 3D TSV 
Histone H4
Kd: 1
1
2D 3D TSV 
Histone-lysine N-methyltransferase 2C
IC50: 1
1
2D 3D TSV 
Histone-lysine N-methyltransferase ASH1L
IC50: 2
1
2D 3D TSV 
Histone-lysine N-methyltransferase E(z)
IC50: 2
2
2D 3D TSV 
Histone-lysine N-methyltransferase EZH2/Polycomb protein EED [40-441]/Polycomb protein SUZ12 [559-739]
Kd: 1
1
2D 3D TSV 
Histone-lysine N-methyltransferase PR-Set7
IC50: 2
2
2D 3D TSV 
Histone-lysine N-methyltransferase Su(var)3-9
IC50: 3
3
2D 3D TSV 
Histone-lysine N-methyltransferase, H3 lysine-9 specific dim-5
IC50: 1
1
2D 3D TSV 
hRXRα-LBD⋅9cRA
ITC: 3
1
2D 3D TSV 
hRXRα-LBD⋅9cUAB30
ITC: 3
1
2D 3D TSV 
hRXRα-LBD⋅Targretin
ITC: 3
1
2D 3D TSV 
Hyaluronate lyase
IC50: 1
1
2D 3D TSV 
Hyaluronidase-1/Hyaluronidase-2
IC50: 1
1
2D 3D TSV 
Hydrolase, alpha/beta hydrolase fold family
IC50: 1
1
2D 3D TSV 
Hydroxyacid oxidase 1
IC50: 1
1
2D 3D TSV 
Inactive tyrosine-protein kinase PEAK1
IC50: 2
2
2D 3D TSV 
Inner capsid protein sigma-2
Ki: 1
1
2D 3D TSV 
Inosine triphosphate pyrophosphatase
IC50: 1
1
2D 3D TSV 
Inositol hexakisphosphate kinase 3
Ki: 1 IC50: 1
1
2D 3D TSV 
Inositol-trisphosphate 3-kinase C
Ki: 1
1
2D 3D TSV 
Insulin receptor substrate 1
Ki: 1
1
2D 3D TSV 
Integrin alpha-1/beta-1
IC50: 1
1
2D 3D TSV 
Integrin alpha-10/beta-1
IC50: 1
1
2D 3D TSV 
Integrin alpha-5/beta-6/beta-8
IC50: 1
1
2D 3D TSV 
Integrin beta-1
IC50: 1
1
2D 3D TSV 
Integrin beta-3/subunit alpha 2b
EC50: 1
1
2D 3D TSV 
Interferon alpha/beta receptor 1
Kd: 1
1
2D 3D TSV 
Interleukin-1 alpha
Ki: 1
1
2D 3D TSV 
Interleukin-1 receptor-associated kinase 1 [184-712]
IC50: 1
1
2D 3D TSV 
Interleukin-1 receptor-associated kinase-like 2
Kd: 1
1
2D 3D TSV 
Interleukin-18
Ki: 1
1
2D 3D TSV 
Interleukin-23 receptor
IC50: 2 Kd: 2
1
2D 3D TSV 
Intermediate conductance calcium-activated potassium channel protein 4/Potassium voltage-gated channel subfamily E member 1/Potassium voltage-gated channel subfamily KQT member 1
IC50: 1
1
2D 3D TSV 
Isoform 1 of Calcitonin receptor (1)/Receptor activity-modifying protein 1
Ki: 1
1
2D 3D TSV 
Isoform 1 of Calcitonin receptor (1)/Receptor activity-modifying protein 3
Ki: 1
1
2D 3D TSV 
Isoform 2 of Proto-oncogene tyrosine-protein kinase receptor Ret
Kd: 1
1
2D 3D TSV 
Isoform 4 of Dual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A (PDE11A1)
IC50: 2
1
2D 3D TSV 
Isoform 5 of Histone deacetylase 7 (5) 18-991]
IC50: 1
1
2D 3D TSV 
Isoform 5-HT4(E) of 5-hydroxytryptamine receptor 4 (H5-HT4(g))
Ki: 1 IC50: 1
1
2D 3D TSV 
Isoform 6 of Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A (PDE1A1)
IC50: 1
1
2D 3D TSV 
Isoform A1-A of Heterogeneous nuclear ribonucleoprotein A1 (A1-A)
Kd: 1
1
2D 3D TSV 
Isoform A1-A of Heterogeneous nuclear ribonucleoprotein A1 (A1-A) 68-320]
Kd: 1
1
2D 3D TSV 
Isoform Cytoplasmic of Fumarate hydratase, mitochondrial (Cytoplasmic)
Ki: 1
1
2D 3D TSV 
Isopentenyl-diphosphate Delta-isomerase 1
IC50: 1
1
2D 3D TSV 
IspB protein
IC50: 2
1
2D 3D TSV 
Jacalin
Kd: 1
1
2D 3D TSV 
Jak1 protein
IC50: 1
1
2D 3D TSV 
Josephin-1
IC50: 1
1
2D 3D TSV 
Josephin-2
IC50: 1
1
2D 3D TSV 
Juvenile hormone esterase, isoform A/B
IC50: 1
1
2D 3D TSV 
Kappa-type opioid receptor [1-7]
Ki: 1
1
2D 3D TSV 
Kinase suppressor of Ras 1
IC50: 2
2
2D 3D TSV 
Kinesin heavy chain isoform 5C
IC50: 1
1
2D 3D TSV 
Kinesin-like protein KIF11 [A356T]
Ki: 2
1
2D 3D TSV 
Kinesin-like protein KIF14
IC50: 1
1
2D 3D TSV 
Kinesin-like protein KIF1B
IC50: 1
1
2D 3D TSV 
Kinesin-like protein KIF2C
IC50: 1
1
2D 3D TSV 
Kinesin-like protein KIF3A
IC50: 1
1
2D 3D TSV 
La-related protein 7
Ki: 1
1
2D 3D TSV 
Leucyl-tRNA synthetase (LeuRS)
Kd: 1 ITC: 1
1
2D 3D TSV 
Leucyl-tRNA synthetase K510A mutant (K510A)
Kd: 1 ITC: 1
1
2D 3D TSV 
Leucyl-tRNA synthetase K510E mutant (K510E)
Kd: 1 ITC: 1
1
2D 3D TSV 
Long-chain-fatty-acid--AMP ligase FadD32
Ki: 1
1
2D 3D TSV 
Low affinity immunoglobulin gamma Fc region receptor II-a
IC50: 1
1
2D 3D TSV 
Low affinity immunoglobulin gamma Fc region receptor III-B
IC50: 1
1
2D 3D TSV 
Luteinizing hormone/choriogondaotropin receptor
IC50: 1
1
2D 3D TSV 
Lymphotoxin-alpha
Kd: 1
1
2D 3D TSV 
Lymphotoxin-beta
IC50: 1
1
2D 3D TSV 
Lysine-specific histone demethylase 1A/REST corepressor 1 [4-485]
Ki: 1
1
2D 3D TSV 
Lysine-specific histone demethylase 1A/REST corepressor 3
IC50: 1
1
2D 3D TSV 
Lysophosphatidic acid receptor 1/3
Ki: 1
1
2D 3D TSV 
Lysosomal acid/Non-lysosomal glucosylceramidase
IC50: 1
1
2D 3D TSV 
Lysosomal alpha-glucosidase/Maltase-glucoamylase/Probable maltase-glucoamylase 2/Sucrase-isomaltase, intestinal
IC50: 1
1
2D 3D TSV 
Lysozyme C
IC50: 1 ITC: 21
4
2D 3D TSV 
Lysyl oxidase homolog 1
IC50: 1
1
2D 3D TSV 
M-phase inducer phosphatase 1/Protein-glutamine gamma-glutamyltransferase 2
IC50: 1
1
2D 3D TSV 
Major pollen allergen Bet v 1-A
Kd: 1
1
2D 3D TSV 
Mannoprotein ligand-binding domain 2 (Mp1p-LBD2 I332A)
ITC: 1
1
0
2D 3D TSV 
Mannoprotein ligand-binding domain 2 (Mp1p-LBD2 V309D)
ITC: 1
1
0
2D 3D TSV 
Mannoprotein ligand-binding domain 2 (Mp1p-LBD2)
ITC: 2
1
0
2D 3D TSV 
Matrix metallopeptidase 12 [174-211]
IC50: 1
1
2D 3D TSV 
Mediator of RNA polymerase II transcription subunit 23
Kd: 1
1
2D 3D TSV 
Meso-diaminopimelate D-dehydrogenase
IC50: 2
1
2D 3D TSV 
Mitochondrial complex I (NADH dehydrogenase)
IC50: 1
1
2D 3D TSV 
Mitochondrial sodium/calcium exchanger protein
IC50: 1
1
2D 3D TSV 
Mitochondrial succinate dehydrogenase subunit C/Succinate dehydrogenase [ubiquinone] iron-sulfur subunit, mitochondrial
IC50: 1
1
2D 3D TSV 
Mitogen-activated protein kinase 1 [L114A]
Kd: 1
1
2D 3D TSV 
Mitogen-activated protein kinase 1 [L198A,L232A]
Kd: 1
1
2D 3D TSV 
Mitogen-activated protein kinase 1 [L198A,L235A]
Kd: 1
1
2D 3D TSV 
Mitogen-activated protein kinase 1 [L232A]
Kd: 1
1
2D 3D TSV 
Mitogen-activated protein kinase 1 [L235A]
Kd: 1
1
2D 3D TSV 
Mitogen-activated protein kinase 1 [L265A]
Kd: 1
1
2D 3D TSV 
Mitogen-activated protein kinase 1 [R275A]
Kd: 1
1
2D 3D TSV 
Mitogen-activated protein kinase 1 [Y191A]
Kd: 1
1
2D 3D TSV 
Mitogen-activated protein kinase 11/14
IC50: 1
1
2D 3D TSV 
Mitogen-activated protein kinase 8 [1-363]
IC50: 1
1
2D 3D TSV 
Mitogen-Activated Protein Kinase 9 (JNK2) Mutant (C162S)
ITC: 1
1
0
2D 3D TSV 
Mitogen-Activated Protein Kinase 9 (JNK2) Mutant (R127A)
ITC: 1
1
0
2D 3D TSV 
Mitogen-activated protein kinase kinase kinase 8 [30-404]
IC50: 1
1
2D 3D TSV 
Mobilization protein A
EC50: 1
1
2D 3D TSV 
Multidrug resistance protein 1
Ki: 1
1
2D 3D TSV 
Myoferlin
Kd: 1
1
2D 3D TSV 
Myosin heavy chain, non-muscle
IC50: 1
1
2D 3D TSV 
Myosin IC heavy chain
IC50: 1
1
2D 3D TSV 
Myosin-10
IC50: 1
1
2D 3D TSV 
Myosin-14
IC50: 1
1
2D 3D TSV 
Myosin-2 heavy chain, non muscle
IC50: 1
1
2D 3D TSV 
Myosin-7
IC50: 1
1
2D 3D TSV 
Myosin-9
IC50: 1
1
2D 3D TSV 
Myosin-J heavy chain
IC50: 1
1
2D 3D TSV 
N-alpha-acetyltransferase 40
IC50: 1
1
2D 3D TSV 
N-lysine methyltransferase SETD6
IC50: 1
1
2D 3D TSV 
Na(+)/H(+) antiporter NhaA
IC50: 2
1
2D 3D TSV 
Nanos homolog 2
Ki: 1
1
2D 3D TSV 
NEDD8
IC50: 1
1
2D 3D TSV 
NEDD8-activating enzyme E1 catalytic/regulatory subunit
EC50: 1
1
2D 3D TSV 
NEDD8-conjugating enzyme Ubc12
Kd: 1
1
2D 3D TSV 
Neurogenic locus notch homolog protein 2
IC50: 1
1
2D 3D TSV 
Neurogenic locus notch homolog protein 4
IC50: 1
1
2D 3D TSV 
Neuronal acetylcholine receptor subunit alpha-7/beta-2
IC50: 1
1
2D 3D TSV 
Neurotensin receptor 1
Ki: 1
1
2D 3D TSV 
NF-kappa-B essential modulator
EC50: 1
1
2D 3D TSV 
Nitric-oxide synthase (NADPH)
IC50: 1
1
2D 3D TSV 
NmrA-like family domain-containing protein 1
Kd: 1
1
2D 3D TSV 
Non-receptor tyrosine-protein kinase TYK2 [870-1187]
IC50: 1
1
2D 3D TSV 
Non-structural protein 1
IC50: 2
1
2D 3D TSV 
Nonmuscle myosin heavy chain
IC50: 1
1
2D 3D TSV 
Nucleotide triphosphate diphosphatase NUDT15
IC50: 1
1
2D 3D TSV 
O15496/P04054/P14555/P39877/Q5R387/Q9BX93/Q9BZM1/Q9BZM2/Q9NZ20/Q9NZK7/Q9UNK4
IC50: 1
1
2D 3D TSV 
Olfactory receptor 145
Ki: 1
1
2D 3D TSV 
OTU domain-containing protein 1
IC50: 1
1
2D 3D TSV 
OTU domain-containing protein 3
IC50: 1
1
2D 3D TSV 
OTU domain-containing protein 6A
IC50: 1
1
2D 3D TSV 
Outer Membrane Phospholipase A
ITC: 2
1
2D 3D TSV 
Outer-membrane lipoprotein carrier protein
Kd: 1
1
2D 3D TSV 
Oxygen-insensitive NAD(P)H nitroreductase
IC50: 1
1
2D 3D TSV 
p2X7 purinoceptor
IC50: 1
1
2D 3D TSV 
Paired box protein Pax-2 [1-81]
Kd: 2
1
2D 3D TSV 
Pantothenate kinase 2, mitochondrial
IC50: 1
1
2D 3D TSV 
Peptidoglycan-N-acetylglucosamine deacetylase BC_1960
Ki: 1 IC50: 1
1
2D 3D TSV 
Peptidoglycan-N-acetylglucosamine deacetylase BC_1974
Ki: 1 IC50: 1
1
2D 3D TSV 
Peptidyl-prolyl cis-trans isomerase FKBP14
Ki: 1
1
2D 3D TSV 
Peptidyl-prolyl cis-trans isomerase FKBP2
Ki: 1
1
2D 3D TSV 
Peroxiredoxin-like 2A
IC50: 1
1
2D 3D TSV 
PHD finger protein 13
IC50: 1
1
2D 3D TSV 
Phosphate regulon sensor protein PhoR
IC50: 1
1
2D 3D TSV 
Phosphate system positive regulatory protein PHO81
IC50: 4
1
2D 3D TSV 
Phosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit alpha isoform [E545K]
IC50: 1
1
2D 3D TSV 
Phosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit alpha isoform [H1047R]
IC50: 1
1
2D 3D TSV 
Phosphatidylinositol 3-kinase regulatory subunit alpha/4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
IC50: 1
1
2D 3D TSV 
Phosphatidylinositol 3-kinase regulatory subunit beta/4,5-bisphosphate 3-kinase catalytic subunit delta isoform
IC50: 1
1
2D 3D TSV 
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform/Platelet-derived growth factor receptor beta [525-1106]
IC50: 1
1
2D 3D TSV 
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform/Proto-oncogene tyrosine-protein kinase Src
IC50: 2
1
2D 3D TSV 
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform/Receptor protein-tyrosine kinase
IC50: 1
1
2D 3D TSV 
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform/Tyrosine-protein kinase ABL1
IC50: 1
1
2D 3D TSV 
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform/Tyrosine-protein kinase HCK
IC50: 1
1
2D 3D TSV 
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform/Vascular endothelial growth factor receptor 2
IC50: 1
1
2D 3D TSV 
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha/beta isoform
IC50: 2
1
2D 3D TSV 
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform/Serine/threonine-protein kinase mTOR
IC50: 2
1
2D 3D TSV 
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform/Platelet-derived growth factor receptor beta [525-1106]
IC50: 1
1
2D 3D TSV 
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform/Proto-oncogene tyrosine-protein kinase Src
IC50: 2
1
2D 3D TSV 
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform/Receptor protein-tyrosine kinase
IC50: 1
1
2D 3D TSV 
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform/Tyrosine-protein kinase ABL1
IC50: 1
1
2D 3D TSV 
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform/Tyrosine-protein kinase HCK
IC50: 1
1
2D 3D TSV 
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform/Vascular endothelial growth factor receptor 2
IC50: 1
1
2D 3D TSV 
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta/gamma isoform
IC50: 2
1
2D 3D TSV 
Phosphatidylinositol 4-phosphate 5-kinase type-1 beta
IC50: 1
1
2D 3D TSV 
Phosphatidylinositol-4,5-bisphosphate 3-kinase
IC50: 1
1
2D 3D TSV 
Phosphodiesterase 3a
Ki: 1
1
2D 3D TSV 
Phosphoglycerate kinase 1/2
Kd: 1
1
2D 3D TSV 
Phospholipase A2 group XV
IC50: 1
1
2D 3D TSV 
Phosphoprotein
IC50: 1
1
2D 3D TSV 
Phosphotransferase pUL97
Ki: 1
1
2D 3D TSV 
Plasmepsin III
IC50: 1
1
2D 3D TSV 
Platelet-derived growth factor receptor alpha [551-1089,V561D]
IC50: 1
1
2D 3D TSV 
Platelet-derived growth factor receptor beta [525-1106] /Serine/threonine-protein kinase mTOR
IC50: 1
1
2D 3D TSV 
PLD alpha C2
ITC: 1
1
2D 3D TSV 
PLD beta C2
ITC: 2
1
2D 3D TSV 
Poly [ADP-ribose] polymerase tankyrase-1 [1030-1317]
IC50: 1
1
2D 3D TSV 
Poly [ADP-ribose] polymerase tankyrase-2 [873-1161]
IC50: 1
1
2D 3D TSV 
Polymerase acidic protein/Polymerase basic protein 2/RNA-directed RNA polymerase catalytic subunit
EC50: 1
1
2D 3D TSV 
Polypeptide N-acetylgalactosaminyltransferase 1
IC50: 1
1
2D 3D TSV 
Polypeptide N-acetylgalactosaminyltransferase 10
IC50: 1
1
2D 3D TSV 
Polypeptide N-acetylgalactosaminyltransferase 13
IC50: 1
1
2D 3D TSV 
Polypeptide N-acetylgalactosaminyltransferase 14
IC50: 1
1
2D 3D TSV 
Polypeptide N-acetylgalactosaminyltransferase 3
IC50: 1
1
2D 3D TSV 
Polypeptide N-acetylgalactosaminyltransferase 6
IC50: 1
1
2D 3D TSV 
Potassium channel subfamily K member 17
IC50: 1
1
2D 3D TSV 
Potassium channel subfamily K member 5
IC50: 1
1
2D 3D TSV 
Potassium channel subfamily T member 2
IC50: 1
1
2D 3D TSV 
Potassium voltage-gated channel subfamily A member 1/2
IC50: 3
1
2D 3D TSV 
Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 3
IC50: 1
1
2D 3D TSV 
Probable glutamate--tRNA ligase, mitochondrial
Ki: 1
1
2D 3D TSV 
Probable JmjC domain-containing histone demethylation protein 2C
IC50: 1
1
2D 3D TSV 
Probable linoleate 9S-lipoxygenase 5
IC50: 1
1
2D 3D TSV 
Probable salicylate monooxygenase
Kd: 1
1
2D 3D TSV 
Probable salicylate monooxygenase [H213A]
Kd: 1
1
2D 3D TSV 
Probable salicylate monooxygenase [Y105F]
Kd: 1
1
2D 3D TSV 
Proenkephalin-B
Kd: 1
1
2D 3D TSV 
Programmed cell death 1 ligand 2
EC50: 2
2
2D 3D TSV 
Prohibitin-2
EC50: 1
1
2D 3D TSV 
Prokineticin-2
IC50: 1 EC50: 1
1
2D 3D TSV 
Proline iminopeptidase
Ki: 1
1
2D 3D TSV 
Prosaposin
Kd: 2
1
2D 3D TSV 
Prostaglandin G/H synthase 2 [R120A,Y385F]
Kd: 1
1
2D 3D TSV 
Prostaglandin G/H synthase 2 [S530A]
Kd: 1
1
2D 3D TSV 
Prostaglandin G/H synthase 2 [Y385F]
Kd: 1
1
2D 3D TSV 
Proteasome assembly chaperone 1/2
IC50: 1
1
2D 3D TSV 
Protein farnesyltransferase subunit beta
Kd: 1
1
2D 3D TSV 
Protein FosB/Transcription factor JunD
IC50: 1
1
2D 3D TSV 
Protein kinase C-binding protein 1
IC50: 1
1
2D 3D TSV 
Protein kinase C-like 1
IC50: 1
1
2D 3D TSV 
Protein max
IC50: 1
1
2D 3D TSV 
Protein mono-ADP-ribosyltransferase PARP10 [809-1017,L926Y]
IC50: 1
1
2D 3D TSV 
Protein mono-ADP-ribosyltransferase PARP10 [809-1017,R931A]
IC50: 1
1
2D 3D TSV 
Protein mono-ADP-ribosyltransferase PARP10 [809-1017,S927A]
IC50: 1
1
2D 3D TSV 
Protein mono-ADP-ribosyltransferase PARP10 [809-1017]
IC50: 1
1
2D 3D TSV 
Protein mono-ADP-ribosyltransferase PARP12 [489-701]
IC50: 1
1
2D 3D TSV 
Protein mono-ADP-ribosyltransferase PARP14 [1535-1801,Y1660L]
IC50: 1
1
2D 3D TSV 
Protein mono-ADP-ribosyltransferase PARP14 [1535-1801]
IC50: 1
1
2D 3D TSV 
Protein mono-ADP-ribosyltransferase PARP15 [460-656,Y598L]
IC50: 1
1
2D 3D TSV 
Protein mono-ADP-ribosyltransferase PARP15 [460-656]
IC50: 1
1
2D 3D TSV 
Protein mono-ADP-ribosyltransferase PARP16 [1-280]
IC50: 1
1
2D 3D TSV 
Protein mono-ADP-ribosyltransferase PARP4 [250-565]
IC50: 1
1
2D 3D TSV 
Protein odd-skipped-related 1
IC50: 2
2
2D 3D TSV 
Protein orai-2/Stromal interaction molecule 1
IC50: 1
1
2D 3D TSV 
Protein orai-3/Stromal interaction molecule 1
IC50: 1
1
2D 3D TSV 
Protein phosphatase 1 regulatory subunit 15A
IC50: 1
1
2D 3D TSV 
Protein phosphatase 1 regulatory subunit 15B
IC50: 1
1
2D 3D TSV 
Protein Red
IC50: 1
1
2D 3D TSV 
Protein-glutamine gamma-glutamyltransferase 2/Receptor protein-tyrosine kinase
IC50: 1
1
2D 3D TSV 
Protein-glutamine gamma-glutamyltransferase 2/Receptor-type tyrosine-protein phosphatase eta
IC50: 1
1
2D 3D TSV 
Protein-glutamine gamma-glutamyltransferase 2/Tyrosine-protein kinase JAK3
IC50: 1
1
2D 3D TSV 
Protein-serine/threonine kinase/[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1/2/4, mitochondrial
IC50: 1
1
2D 3D TSV 
Proteinase K
IC50: 1
1
2D 3D TSV 
Proto-oncogene tyrosine-protein kinase Src/Serine/threonine-protein kinase mTOR
IC50: 2
1
2D 3D TSV 
Proto-oncogene vav
Kd: 1
1
2D 3D TSV 
Protoporphyrinogen oxidase, mitochondrial
Ki: 1
1
2D 3D TSV 
Putative choline uptake ABC transporter permease protein
Ki: 1
1
2D 3D TSV 
Putative FAD-containing monooxygenase MymA
IC50: 1
1
2D 3D TSV 
Putative peripheral benzodiazepine receptor-related protein
IC50: 1
1
2D 3D TSV 
Pyridoxine-5'-phosphate oxidase
Ki: 1
1
2D 3D TSV 
Pyruvate-flavodoxin oxidoreductase
Ki: 1
1
2D 3D TSV 
RAF proto-oncogene serine/threonine-protein kinase [305-648]
IC50: 1
1
2D 3D TSV 
Rapamycin-insensitive companion of mTOR/Serine/threonine-protein kinase mTOR/Target of rapamycin complex 2 subunit MAPKAP1/Target of rapamycin complex subunit LST8
IC50: 1
1
2D 3D TSV 
Ras-related protein Rab-6A
Kd: 1
1
2D 3D TSV 
Ras-related protein Rab-7L1
Ki: 1
1
2D 3D TSV 
Receptor protein-tyrosine kinase/Serine/threonine-protein kinase mTOR
IC50: 1
1
2D 3D TSV 
Receptor-interacting serine/threonine kinase 1
Ki: 1
1
2D 3D TSV 
Receptor-type tyrosine-protein kinase FLT3 [563-993,D835Y]
IC50: 1
1
2D 3D TSV 
Receptor-type tyrosine-protein kinase FLT3 [K663Q]
Kd: 1
1
2D 3D TSV 
Receptor-type tyrosine-protein kinase FLT3 [R834Q]
Kd: 1
1
2D 3D TSV 
Receptor-type tyrosine-protein phosphatase R
IC50: 1
1
2D 3D TSV 
Regulatory-associated protein of mTOR/Serine/threonine-protein kinase mTOR/Target of rapamycin complex subunit LST8
IC50: 1
1
2D 3D TSV 
Relaxin-3 receptor 1/2
EC50: 1
1
2D 3D TSV 
Reticulon-4
IC50: 1
1
2D 3D TSV 
Rho guanine nucleotide exchange factor 1
IC50: 1
1
2D 3D TSV 
Rho-associated protein kinase 2 [6-553]
IC50: 1
1
2D 3D TSV 
Rho-related GTP-binding protein RhoC/Transforming protein RhoA
IC50: 1
1
2D 3D TSV 
Ribonucleoside-diphosphate reductase large subunit/subunit M2/subunit M2 B
IC50: 1
1
2D 3D TSV 
Ribosomal oxygenase 1
IC50: 1
1
2D 3D TSV 
Ribosomal oxygenase 2
IC50: 1
1
2D 3D TSV 
Ribosomal protein S6 kinase alpha-1 [E551G,S637N,G697A]
IC50: 1
1
2D 3D TSV 
RISC-loading complex subunit TARBP2
Kd: 1
1
2D 3D TSV 
RNA 5'-monophosphate methyltransferase
IC50: 1
1
2D 3D TSV 
RNA guanine-N7 methyltransferase activating subunit
IC50: 1
1
2D 3D TSV 
RNA(23-mer)
ITC: 9
1
0
2D 3D TSV 
Ryanodine receptor 2
EC50: 1
1
2D 3D TSV 
Ryanodine receptor 3
IC50: 1
1
2D 3D TSV 
S-methylmethionine--homocysteine S-methyltransferase BHMT2
Ki: 1 IC50: 1
1
2D 3D TSV 
Salicylate synthase
Ki: 1
1
2D 3D TSV 
Serine/threonine-protein kinase 31
Ki: 1
1
2D 3D TSV 
Serine/threonine-protein kinase B-raf [410-766,V600E]
IC50: 1
1
2D 3D TSV 
Serine/threonine-protein kinase haspin [465-798]
IC50: 1 Kd: 1 ITC: 1
1
2D 3D TSV 
Serine/threonine-protein kinase mTOR/Tyrosine-protein kinase ABL1
IC50: 1
1
2D 3D TSV 
Serine/threonine-protein kinase mTOR/Tyrosine-protein kinase HCK
IC50: 1
1
2D 3D TSV 
Serine/threonine-protein kinase mTOR/Vascular endothelial growth factor receptor 2
IC50: 1
1
2D 3D TSV 
Serine/threonine-protein kinase Nek10
Kd: 1
1
2D 3D TSV 
Serine/threonine-protein kinase Nek8
IC50: 2
2
2D 3D TSV 
Serine/threonine-protein kinase WNK1 [1-434]
IC50: 1
1
2D 3D TSV 
Serine/threonine-protein kinase WNK1 [1-444]
IC50: 1
1
2D 3D TSV 
Serine/threonine-protein kinase WNK1 [166-489]
IC50: 1
1
2D 3D TSV 
Serine/threonine-protein kinase WNK2 [166-489]
IC50: 1
1
2D 3D TSV 
Serine/threonine-protein kinase WNK3 [1-434]
IC50: 1
1
2D 3D TSV 
Serine/threonine-protein kinase WNK4 [1-444]
IC50: 1
1
2D 3D TSV 
Serine/threonine-protein kinase-transforming protein raf [E280V]
Kd: 1
1
2D 3D TSV 
Serine/threonine-protein kinase-transforming protein raf [F278H]
Kd: 1
1
2D 3D TSV 
Serine/threonine-protein kinase/endoribonuclease IRE2
IC50: 2
2
2D 3D TSV 
Serine/threonine-protein phosphatase 2A 55 kDa regulatory subunit B alpha isoform
IC50: 1
1
2D 3D TSV 
SHC-transforming protein 2
IC50: 1
1
2D 3D TSV 
Short transient receptor potential channel 1/5
IC50: 1
1
2D 3D TSV 
Short transient receptor potential channel 3/6
IC50: 1
1
2D 3D TSV 
Signal peptidase IB
IC50: 1
1
2D 3D TSV 
Signal transducer and activator of transcription 2
Kd: 1
1
2D 3D TSV 
Signal transducer and transcription activator 6
IC50: 1
1
2D 3D TSV 
Similar to RIKEN cDNA 2010106G01 (Predicted)
IC50: 1
1
2D 3D TSV 
Sodium channel protein type 1/10/11/2/3/4/5/7/8/9 subunit alpha
IC50: 1
1
2D 3D TSV 
Sodium channel protein type 1/2/3/4/5/8/9/10/11 subunit alpha
Kd: 1
1
2D 3D TSV 
Sodium channel protein type 4 subunit alpha/subunit beta-1/subunit beta-2
IC50: 1
1
2D 3D TSV 
Sodium channel protein type 9 subunit alpha/subunit beta-1/subunit beta-2
IC50: 1
1
2D 3D TSV 
Sodium channel subunit beta-3
Ki: 1
1
2D 3D TSV 
Sodium-dependent phosphate transport protein 1
Ki: 1
1
2D 3D TSV 
Sodium/hydrogen exchanger 1/2/3
IC50: 1
1
2D 3D TSV 
Sodium/hydrogen exchanger isoform 3
IC50: 1
1
2D 3D TSV 
Sodium/potassium-transporting ATPase subunit alpha-4/beta-3
IC50: 1
1
2D 3D TSV 
Soluble maltase-glucoamylase
IC50: 1
1
2D 3D TSV 
Solute carrier family 2, facilitated glucose transporter member 14
IC50: 1
1
2D 3D TSV 
Solute carrier family 2, facilitated glucose transporter member 5
Ki: 2
1
2D 3D TSV 
Solute carrier family 22 member 16
Ki: 1
1
2D 3D TSV 
Solute carrier family 5 (neutral amino acid transporters, system A), member 4b
IC50: 1
1
2D 3D TSV 
Solute carrier organic anion transporter family member 1B2
Ki: 1
1
2D 3D TSV 
Somatostatin receptor subtype 3
IC50: 1
1
2D 3D TSV 
Speckle-type POZ protein
Kd: 1
1
2D 3D TSV 
Sporulation initiation phosphotransferase F/kinase A
IC50: 1
1
2D 3D TSV 
SRC kinase signaling inhibitor 1
IC50: 1
1
2D 3D TSV 
SRSF protein kinase 1
Ki: 1
1
2D 3D TSV 
Streptavadin(N23A)
ITC: 2
1
0
2D 3D TSV 
Streptavadin(N23E)
ITC: 2
1
0
2D 3D TSV 
Streptavadin(S27A)
ITC: 2
1
0
2D 3D TSV 
Streptavadin(W108F)
ITC: 1
1
0
2D 3D TSV 
Streptavadin(W120F)
ITC: 1
1
0
2D 3D TSV 
Streptavadin(W79F)
ITC: 1
1
0
2D 3D TSV 
Streptavadin(Y43A)
ITC: 2
1
0
2D 3D TSV 
Streptavidin (Y43F)
ITC: 2
1
0
2D 3D TSV 
Streptavidin [37-163,Y46S,Y107S,R108K,E125D,R127K,E140N]
Kd: 1
1
2D 3D TSV 
Streptopain
Ki: 1 IC50: 1
1
2D 3D TSV 
Succinate dehydrogenase [ubiquinone] cytochrome b small/cytochrome b560 subunit, mitochondrial
IC50: 1
1
2D 3D TSV 
Sulfate anion transporter 1
Ki: 1
1
2D 3D TSV 
Sulfhydryl oxidase 1
IC50: 1
1
2D 3D TSV 
Synaptic vesicle membrane protein VAT-1 homolog
IC50: 2
1
2D 3D TSV 
Synaptic vesicular amine transporter [V41F]
Kd: 1
1
2D 3D TSV 
Syndecan-2/Syntenin-1
IC50: 1
1
2D 3D TSV 
Targeting protein for Xklp2
Ki: 1
1
2D 3D TSV 
Taste receptor type 2 member 1
EC50: 1
1
2D 3D TSV 
Taste receptor type 2 member 16
IC50: 1 EC50: 1
1
2D 3D TSV 
Taste receptor type 2 member 4
EC50: 1
1
2D 3D TSV 
Taste receptor type 2 member 41
EC50: 1
1
2D 3D TSV 
Taste receptor type 2 member 60
EC50: 1
1
2D 3D TSV 
Taste receptor type 2 member 9
EC50: 1
1
2D 3D TSV 
TATA box-binding protein-associated factor RNA polymerase I subunit A
IC50: 1
1
2D 3D TSV 
Testis-specific serine/threonine-protein kinase 4
IC50: 1
1
2D 3D TSV 
TGF-beta-activated kinase 1 and MAP3K7-binding protein 1
IC50: 1
1
2D 3D TSV 
Thiamine transporter 1
Ki: 2
1
2D 3D TSV 
Thiol:disulfide interchange protein [27-205]/AFDQIDNAPEE
Kd: 1 ITC: 1
2
2D 3D TSV 
Thioredoxin, mitochondrial
Ki: 1
1
2D 3D TSV 
Thymidine Kinase (TK.dT)
ITC: 4
1
2D 3D TSV 
Trans-sialidase [3-643,D247A]
Kd: 1
1
2D 3D TSV 
Transcription factor Dp-2
IC50: 2
1
2D 3D TSV 
Transcription factor ETV6
IC50: 1
1
2D 3D TSV 
Transcription initiation factor TFIID subunit 11
Kd: 1
1
2D 3D TSV 
Transducer protein Htr4
Ki: 1
1
2D 3D TSV 
Transient receptor potential cation channel subfamily M member 1
IC50: 1
1
2D 3D TSV 
Transient receptor potential cation channel subfamily V member 5
IC50: 1
1
2D 3D TSV 
Transient receptor potential protein 5
IC50: 1
1
2D 3D TSV 
Translation factor GUF1, mitochondrial
IC50: 1
1
2D 3D TSV 
TREK-2 two-pore-domain K+ channel
EC50: 1
1
2D 3D TSV 
Tribbles homolog 2
IC50: 1
1
2D 3D TSV 
tRNA-dihydrouridine(20) synthase [NAD(P)+]-like
IC50: 1
1
2D 3D TSV 
Tryptophan synthase alpha/beta chain
Ki: 1
1
2D 3D TSV 
Tubulin alpha chain-like 3/1A chain/1B chain/1C chain/3C chain/3E chain/4A chain/8 chain
IC50: 1
1
2D 3D TSV 
Tubulin alpha-8 chain
IC50: 1
1
2D 3D TSV 
Tubulin polyglutamylase TTLL7
IC50: 1
1
2D 3D TSV 
Tumor necrosis factor ligand superfamily member 6
IC50: 1
1
2D 3D TSV 
Type III pantothenate kinase
Ki: 1
1
2D 3D TSV 
Tyramine receptor
IC50: 1
1
2D 3D TSV 
Tyrosine-protein kinase ABL1 [1-999,E255V]
Kd: 1
1
2D 3D TSV 
Tyrosine-protein kinase ABL1 [1-999,Y253H]
Kd: 1
1
2D 3D TSV 
Tyrosine-protein kinase JAK2 [866-1054]
IC50: 1
1
2D 3D TSV 
Tyrosine-protein kinase JAK3 [1-973]
IC50: 1
1
2D 3D TSV 
Tyrosine-protein kinase transforming protein Fps
Ki: 1
1
2D 3D TSV 
Tyrosine-protein phosphatase non-receptor type 1 [G117E]
IC50: 1
1
2D 3D TSV 
Tyrosine-protein phosphatase non-receptor type 1 [M114V]
IC50: 1
1
2D 3D TSV 
Tyrosine-protein phosphatase non-receptor type 1 [V113I]
IC50: 1
1
2D 3D TSV 
Tyrosine-protein phosphatase non-receptor type 1 [V113L,M114V]
IC50: 1
1
2D 3D TSV 
Tyrosine-protein phosphatase non-receptor type 21
IC50: 1
1
2D 3D TSV 
Tyrosyl-DNA phosphodiesterase 2 [Q278R,I281T,K282R,P318T,Y321C]
IC50: 1
1
2D 3D TSV 
Ubiquitin carboxyl-terminal hydrolase 10
IC50: 1
1
2D 3D TSV 
Ubiquitin carboxyl-terminal hydrolase 11
IC50: 1
1
2D 3D TSV 
Ubiquitin carboxyl-terminal hydrolase 13
IC50: 1
1
2D 3D TSV 
Ubiquitin carboxyl-terminal hydrolase 16
IC50: 1
1
2D 3D TSV 
Ubiquitin carboxyl-terminal hydrolase 27
IC50: 1
1
2D 3D TSV 
Ubiquitin carboxyl-terminal hydrolase 35
IC50: 1
1
2D 3D TSV 
Ubiquitin carboxyl-terminal hydrolase 36
IC50: 1
1
2D 3D TSV 
Ubiquitin carboxyl-terminal hydrolase 45
IC50: 1
1
2D 3D TSV 
Ubiquitin carboxyl-terminal hydrolase 6
IC50: 1
1
2D 3D TSV 
Ubiquitin carboxyl-terminal hydrolase CYLD
IC50: 1
1
2D 3D TSV 
Ubiquitin thioesterase OTU1
IC50: 1
1
2D 3D TSV 
Ubiquitin thioesterase OTUB2
IC50: 1
1
2D 3D TSV 
Ubiquitin-conjugating enzyme E2 B
IC50: 1
1
2D 3D TSV 
Ubiquitin-conjugating enzyme E2 T
Kd: 1
1
2D 3D TSV 
Ubiquitin-like modifier-activating enzyme 1 [957-994]
IC50: 3
1
2D 3D TSV 
Ubiquitin-like modifier-activating enzyme 7
IC50: 1
1
2D 3D TSV 
UDP-glucuronosyltransferase 1A3
Ki: 2
1
2D 3D TSV 
UDP-N-acetylmuramate--L-alanine ligase [A299V,V378L,T444A]
IC50: 1
1
2D 3D TSV 
Ultraspiracle protein
IC50: 1
1
2D 3D TSV 
Unconventional myosin-Ib
IC50: 1
1
2D 3D TSV 
Unconventional myosin-X
IC50: 1
1
2D 3D TSV 
Unconventional myosin-XV
IC50: 1
1
2D 3D TSV 
Uracil phosphoribosyltransferase
Ki: 1
1
2D 3D TSV 
Urease subunit alpha [1-30]/beta/gamma
IC50: 1
1
2D 3D TSV 
Urease subunit alpha/beta
IC50: 1
1
2D 3D TSV 
Uridine diphosphate glucose pyrophosphatase NUDT14
IC50: 1
1
2D 3D TSV 
Uridine-cytidine kinase 1
Ki: 1
1
2D 3D TSV 
V-type proton ATPase subunit B, brain isoform
IC50: 1
1
2D 3D TSV 
V-type proton ATPase subunit C
IC50: 1
1
2D 3D TSV 
Vacuolar protein sorting-associated protein 35
IC50: 1
1
2D 3D TSV 
Vacuolar protein sorting-associated protein 4B
IC50: 2
1
2D 3D TSV 
Vascular endothelial growth factor receptor 2 [807-1356]
IC50: 1
1
2D 3D TSV 
Vesicle amine transport protein 1 homolog (T. californica)-like
Ki: 1
1
2D 3D TSV 
Vesicle-fusing ATPase
IC50: 1
1
2D 3D TSV 
Vitamin K epoxide reductase complex subunit 1-like protein 1
Ki: 2
1
2D 3D TSV 
Voltage-dependent anion-selective channel protein 2
Kd: 1
1
2D 3D TSV 
Voltage-dependent L-type calcium channel subunit alpha-1C/L-type calcium channel subunit beta-2/calcium channel subunit alpha-2/delta-1
IC50: 1
1
2D 3D TSV 
Voltage-dependent L-type calcium channel subunit beta-3/N-type calcium channel subunit alpha-1B
IC50: 1
1
2D 3D TSV 
Voltage-dependent R-type calcium channel subunit alpha-1E
IC50: 1
1
2D 3D TSV 
Voltage-dependent T-type calcium channel subunit alpha-1G/alpha-1H/alpha-1I
IC50: 1
1
2D 3D TSV 
Voltage-gated sodium channel Nav1.5 cardiac isoform
IC50: 1
1
2D 3D TSV 
Xanthine dehydrogenase
Ki: 1
1
2D 3D TSV 
Zinc finger protein GLI1/GLI2
IC50: 1
1
2D 3D TSV 
Zinc finger protein GLIS2
IC50: 1
1
2D 3D TSV 
[3-methyl-2-oxobutanoate dehydrogenase [lipoamide]] kinase, mitochondrial
IC50: 1
1
2D 3D TSV