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Targets Binding with 7 Compounds
Target Name
Affinity Link(s)
Article(s)
UniProt
Files
14-3-3 protein sigma
IC50:
6
Kd:
1
3
5
2D
3D
TSV
4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase 9
Ki:
7
IC50:
7
1
3
2D
3D
TSV
Aldo-keto reductase family 1 member B10 [K125R,V301L]
IC50:
7
1
7
2D
3D
TSV
Alkanal monooxygenase alpha chain
EC50:
21
3
5
2D
3D
TSV
Alpha-crystallin B chain
EC50:
8
1
9
2D
3D
TSV
Alpha-glucosidase
IC50:
7
3
4
2D
3D
TSV
Aminoacyl tRNA synthase complex-interacting multifunctional protein 2
IC50:
10
Kd:
3
2
6
2D
3D
TSV
Angiotensin-converting enzyme/Ribosomal RNA small subunit methyltransferase NEP1
Ki:
14
2
11
2D
3D
TSV
Beta-2-microglobulin
IC50:
7
1
8
2D
3D
TSV
Beta-secretase 1 [22-454]
Ki:
7
1
11
2D
3D
TSV
Bromodomain-containing protein 2 [74-94]
Kd:
7
1
13
2D
3D
TSV
C-C motif chemokine 3
IC50:
7
1
1
2D
3D
TSV
C-C motif chemokine 4
IC50:
7
1
6
2D
3D
TSV
Calcium/calmodulin-dependent protein kinase type 1B
IC50:
7
Kd:
1
7
7
2D
3D
TSV
Calcium/calmodulin-dependent protein kinase type IV [15-340]
Ki:
7
1
3
2D
3D
TSV
Casein kinase I isoform alpha/delta/epsilon/gamma-1/gamma-2
IC50:
7
5
23
2D
3D
TSV
cGMP-gated cation channel alpha-1
Kd:
14
1
1
2D
3D
TSV
Choline/ethanolamine kinase
IC50:
2
Kd:
5
4
4
2D
3D
TSV
Complement C5
IC50:
3
Kd:
4
2
4
2D
3D
TSV
Complex of Baculoviral IAP repeat-containing protein 7 [1-159,S150G] and E3 ubiquitin-protein ligase XIAP [336-348]
Ki:
7
1
9
2D
3D
TSV
Complex of Sliding-clamp-loader large subunit [R175K] and Sliding-clamp-loader small subunit
Ki:
7
1
2
2D
3D
TSV
Complex of Sliding-clamp-loader large subunit [R175L] and Sliding-clamp-loader small subunit
Ki:
7
1
2
2D
3D
TSV
Cyclic GMP-AMP synthase
IC50:
12
Kd:
8
2
8
2D
3D
TSV
Cyclin homolog/dependent kinase 6
IC50:
7
1
3
2D
3D
TSV
Cysteine proteinase B
Ki:
5
IC50:
3
2
1
2D
3D
TSV
Cytochrome P450 130
Kd:
15
2
5
2D
3D
TSV
Cytochrome P450 2B4
Ki:
5
ITC:
2
2
3
2D
3D
TSV
Cytohesin-3
IC50:
3
Kd:
5
3
4
2D
3D
TSV
D(2) dopamine receptor/Metabotropic glutamate receptor 5
IC50:
3
EC50:
5
1
5
2D
3D
TSV
Dedicator of cytokinesis protein 2
IC50:
8
1
4
2D
3D
TSV
Delta-type/Mu-type opioid receptor
EC50:
14
2
33
2D
3D
TSV
Dickkopf-related protein 1
IC50:
1
EC50:
6
2
5
2D
3D
TSV
Dimer of Gag-Pol polyprotein [482-580,I502K,I528M,T553A,V564F]
Ki:
7
1
5
2D
3D
TSV
Dimer of Gag-Pol polyprotein [482-580,I502K,I528M,T553A]
Ki:
7
1
4
2D
3D
TSV
Dimer of Gag-Pol polyprotein [490-588,L523I,E525D,M526I,I544V,L553H,H559K,L579M]
Ki:
7
1
8
2D
3D
TSV
Dimer of Gag-Pol polyprotein [490-588,L523I,E525D,M526I,I544V,L553H,H559K,V572F,L579M]
Ki:
7
1
9
2D
3D
TSV
Dimer of Gag-Pol polyprotein [501-599,V583F]
Ki:
7
1
2
2D
3D
TSV
Dioxygenase
Ki:
1
IC50:
7
1
1
2D
3D
TSV
DNA topoisomerase 2
IC50:
7
3
7
2D
3D
TSV
Dual specificity protein phosphatase 4
IC50:
7
1
6
2D
3D
TSV
Endoglucanase-5
Ki:
7
1
1
2D
3D
TSV
Fumarate reductase
IC50:
7
1
1
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-3 [29-492]/beta-3 [26-473]/gamma-2 [40-467]
Ki:
7
1
15
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-6 [20-453]/beta-3 [26-473]/gamma-2 [40-467]
Ki:
7
1
16
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-6/beta-3
IC50:
7
EC50:
2
1
3
2D
3D
TSV
Gamma-aminobutyric acid receptor subunit alpha-6/beta-3/delta
IC50:
10
1
4
2D
3D
TSV
Geranylgeranyl transferase type-2 subunit alpha
IC50:
7
1
1
2D
3D
TSV
Glucoamylase, intracellular sporulation-specific
Ki:
4
IC50:
3
1
4
2D
3D
TSV
Glycoprotein G
EC50:
7
1
4
2D
3D
TSV
Granulocyte-macrophage colony-stimulating factor
IC50:
7
1
5
2D
3D
TSV
GTP-binding nuclear protein GSP1/CNR1
Ki:
7
1
3
2D
3D
TSV
Heat shock protein HSP 90-alpha [1-236]
Kd:
7
1
8
2D
3D
TSV
High affinity immunoglobulin epsilon receptor subunit alpha
IC50:
7
1
1
2D
3D
TSV
Histone H1.0
Ki:
7
1
6
2D
3D
TSV
Histone-binding protein RBBP4/Polycomb protein EED/Polycomb protein SUZ12/Zinc finger protein AEBP2
IC50:
8
1
21
2D
3D
TSV
Histone-lysine N-methyltransferase KMT5C
IC50:
7
3
4
2D
3D
TSV
Homoisocitrate dehydrogenase, mitochondrial
Ki:
7
2
3
2D
3D
TSV
HTH-type quorum-sensing regulator RhlR
IC50:
8
3
3
2D
3D
TSV
inhibitionask1 alphascreen
IC50:
7
1
0
2D
3D
TSV
Integrin alpha-3
IC50:
7
Kd:
1
1
7
2D
3D
TSV
Interleukin-10
EC50:
7
1
1
2D
3D
TSV
Interstitial collagenase [100-268]
IC50:
8
1
3
2D
3D
TSV
Isoform 2 of Vascular endothelial growth factor receptor 3 (Short) 98-1298]
IC50:
7
1
7
2D
3D
TSV
Isoform 3 of Ribosomal protein S6 kinase alpha-2 (3)
Ki:
7
1
8
2D
3D
TSV
Macrophage colony-stimulating factor 1 receptor [538-678,753-922]
IC50:
14
1
8
2D
3D
TSV
Mannosyl-oligosaccharide alpha-1,2-mannosidase IA
Ki:
1
IC50:
7
1
7
2D
3D
TSV
Mast cell carboxypeptidase A
Ki:
6
Kd:
2
5
5
2D
3D
TSV
Mast/stem cell growth factor receptor Kit [N822K]
Kd:
7
1
9
2D
3D
TSV
Mast/stem cell growth factor receptor Kit [V559D]
Kd:
7
1
9
2D
3D
TSV
Mediator of DNA damage checkpoint protein 1
IC50:
7
1
16
2D
3D
TSV
Methyl-accepting chemotaxis protein NahY
Kd:
7
ITC:
7
1
1
2D
3D
TSV
N-acetyltransferase domain-containing protein
Kd:
7
ITC:
7
1
1
2D
3D
TSV
Na+/H+ exchanger regulatory factor-1 PDZ domain (PDZ2)
Ki:
1
Kd:
6
ITC:
5
1
5
2D
3D
TSV
Neurotensin receptor type 1 [45-272,291-390,C386A,C388A]
Kd:
12
1
7
2D
3D
TSV
Non-receptor tyrosine-protein kinase TYK2/Tyrosine-protein kinase JAK1/Tyrosine-protein kinase JAK2
IC50:
9
3
9
2D
3D
TSV
Penicillin-binding protein, transpeptidase domain protein
IC50:
12
2
1
2D
3D
TSV
Penicillopepsin-1
Ki:
9
1
1
2D
3D
TSV
Phosducin-like protein 3
Kd:
7
1
4
2D
3D
TSV
Phosphatidylserine lipase ABHD16A
IC50:
12
2
8
2D
3D
TSV
Phospholipase C-γ1 SH2 domain (PLCC)
ITC:
7
1
6
2D
3D
TSV
Potassium voltage-gated channel subfamily B member 1
IC50:
7
EC50:
1
3
4
2D
3D
TSV
Potassium voltage-gated channel subfamily B member 2
IC50:
7
2
4
2D
3D
TSV
Potassium voltage-gated channel subfamily D member 2
IC50:
8
1
4
2D
3D
TSV
Potassium voltage-gated channel subfamily KQT member 3/5
EC50:
7
1
17
2D
3D
TSV
Potassium voltage-gated channel subfamily KQT member 5
EC50:
8
3
14
2D
3D
TSV
Presenilin-2
IC50:
8
1
5
2D
3D
TSV
Putative lanosterol 14-alpha-demethylase
Kd:
7
2
4
2D
3D
TSV
Pyridoxal kinase
Ki:
5
IC50:
2
4
4
2D
3D
TSV
RCG37580
EC50:
8
1
3
2D
3D
TSV
Receptor-type tyrosine-protein phosphatase zeta
IC50:
7
1
6
2D
3D
TSV
Retinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit gamma
IC50:
7
1
1
2D
3D
TSV
Rho-associated protein kinase 2 [1-543,T431N]
IC50:
7
1
6
2D
3D
TSV
Ribonucleoside-diphosphate reductase subunit alpha
Kd:
7
1
6
2D
3D
TSV
Serine hydrolase RBBP9
IC50:
8
1
5
2D
3D
TSV
Serine/threonine-protein kinase WNK3
IC50:
7
7
7
2D
3D
TSV
Sodium channel protein type 1 subunit alpha [1489-1708]
IC50:
6
Kd:
1
2
5
2D
3D
TSV
Sodium channel protein type 1 subunit alpha/subunit beta-1
IC50:
14
1
10
2D
3D
TSV
Solute carrier family 22 member 7
Ki:
1
IC50:
14
3
9
2D
3D
TSV
Sphingomyelin phosphodiesterase [1-45,48-631]
IC50:
7
2
9
2D
3D
TSV
Suppressor of tumorigenicity 14 protein [596-855]
Ki:
7
1
6
2D
3D
TSV
Testis-specific serine/threonine-protein kinase 3
IC50:
6
Kd:
2
7
3
2D
3D
TSV
Transforming growth factor beta-1 proprotein
IC50:
7
1
4
2D
3D
TSV
Tyrosine-protein kinase ABL1 [201-500,E255K]
Kd:
7
1
9
2D
3D
TSV
Tyrosine-protein kinase ABL1 [201-500,F359V]
Kd:
7
1
9
2D
3D
TSV
Tyrosine-protein kinase ABL1 [201-500,H396P]
Kd:
7
1
9
2D
3D
TSV
Tyrosine-protein kinase ABL1 [201-500,M351T]
Kd:
7
1
9
2D
3D
TSV
Tyrosine-protein kinase ABL1 [201-500,Q252H]
Kd:
7
1
9
2D
3D
TSV
Tyrosine-protein kinase ABL1 [201-500,T315I]
Kd:
7
1
9
2D
3D
TSV
Tyrosine-protein kinase ABL1 [201-500,T315N]
Kd:
7
1
9
2D
3D
TSV
Tyrosine-protein kinase ABL1 [201-500,Y253F]
Kd:
7
1
9
2D
3D
TSV
Tyrosine-protein kinase ABL1 [201-500]
Kd:
7
1
8
2D
3D
TSV
U4/U6 small nuclear ribonucleoprotein Prp4
Kd:
7
1
7
2D
3D
TSV
UDP-glucuronosyltransferase 1A10
Ki:
7
5
5
2D
3D
TSV
V-type proton ATPase subunit S1
IC50:
12
2
5
2D
3D
TSV
Vitamin D-binding protein
IC50:
7
Kd:
1
2
2
2D
3D
TSV