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31 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Therapeutic Potential of 5-HT6 Receptor Agonists.EBI
Universit£
Discovery and SAR of org 24598-a selective glycine uptake inhibitor.EBI
Organon Research And Development Group
(R)-(+)-2-[[[3-(Morpholinomethyl)-2H-chromen-8-yl]oxy]methyl] morpholine methanesulfonate: a new selective rat 5-hydroxytryptamine1B receptor antagonist.EBI
Astra Arcus
Buspirone analogues. 2. Structure-activity relationships of aromatic imide derivatives.EBI
TBA
Discovery of 7-arylsulfonyl-1,2,3,4, 4a,9a-hexahydro-benzo[4,5]furo[2,3-c]pyridines: identification of a potent and selective 5-HT6 receptor antagonist showing activity in rat social recognition test.EBI
Cephalon
Novel brain penetrant benzofuropiperidine 5-HT6 receptor antagonists.EBI
Cephalon
8-Sulfonyl-substituted tetrahydro-1H-pyrido[4,3-b]indoles as 5-HT6 receptor antagonists.EBI
Chemical Diversity Research Institute
Novel sigma receptor ligands: synthesis and biological profile.EBI
University Of Catania
Synthesis and structure--activity relationship in a class of indolebutylpiperazines as dual 5-HT(1A) receptor agonists and serotonin reuptake inhibitors.EBI
Merck
Novel 2-aminotetralin and 3-aminochroman derivatives as selective serotonin 5-HT7 receptor agonists and antagonists.EBI
Uppsala University
N1-Azinylsulfonyl-1H-indoles: 5-HT6 Receptor Antagonists with Procognitive and Antidepressant-Like Properties.EBI
Jagiellonian University Medical College
3-[3-(Piperidin-1-yl)propyl]indoles as highly selective h5-HT(1D) receptor agonists.EBI
Merck Sharp & Dohme Research Laboratories
N-Substituted (2,3-dihydro-1,4-benzodioxin-2-yl)methylamine derivatives as D(2) antagonists/5-HT(1A) partial agonists with potential as atypical antipsychotic agents.EBI
Knoll Pharmaceuticals
Synthesis of azepino[4,5-b]indol-4-ones via MCR/free radical cyclization and in vitro-in silico studies as 5-Ht?R ligands.EBI
Universidad De Guanajuato
Development of high-affinity 5-HT3 receptor antagonists. Structure-affinity relationships of novel 1,7-annelated indole derivatives.EBI
Solvay Duphar
Synthesis and evaluation of a novel series of N,N-dimethylisotryptamines.EBI
TBA
Bicyclic heteroarylpiperazines as selective brain penetrant 5-HT6 receptor antagonists.EBI
Glaxosmithkline
The A128T resistance mutation reveals aberrant protein multimerization as the primary mechanism of action of allosteric HIV-1 integrase inhibitors.BDB
The Ohio State University
Benzimidazole derivatives as new a-glucosidase inhibitors and in silico studies.BDB
Universiti Teknologi Mara (Uitm)
Small Molecule Inhibitors of 8-Oxoguanine DNA Glycosylase-1 (OGG1).BDB
Oregon Health & Science University