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35 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
16250647 71 2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine and analogues as A2A adenosine receptor antagonists. Design, synthesis, and pharmacological characterization.EBI Universit£ degli Studi di Urbino Carlo Bo
12036354 23 Novel class of potent 4-arylalkyl substituted 3-isoxazolol GABA(A) antagonists: synthesis, pharmacology, and molecular modeling.EBI The Royal Danish School of Pharmacy
7650683 12 Partial GABAA receptor agonists. Synthesis and in vitro pharmacology of a series of nonannulated analogs of 4,5,6,7-tetrahydroisoxazolo[5,4-c]pyridin-3-ol.EBI Royal Danish School of Pharmacy
1652022 18 3-Thienyl- and 3-furylaminobutyric acids. Synthesis and binding GABAB receptor studies.EBI Laboratoire de Pharmacie Chimique, Facult� de Pharmacie, Lille, France.
1849996 7 Synthesis and biochemical evaluation of baclofen analogues locked in the baclofen solid-state conformation.EBI Centre de Neurochimie du CNRS
2153214 4 GABA agonists and uptake inhibitors. Synthesis, absolute stereochemistry, and enantioselectivity of (R)-(-)- and (S)-(+)-homo-beta-proline.EBI Royal Danish School of Pharmacy
3031294 10 Synthesis and pharmacological evaluation of gamma-aminobutyric acid analogues. New ligand for GABAB sites.EBI TBA
10560731 2 Aminomethyl-2,6-difluorophenols as a novel class of increased lipophilicity GABA(C) receptor antagonists.EBI The University of Sydney
 2 The first selective antagonist for a GABAC receptorEBI TBA
 7 A study of 3-amino-N-hydroxypropanesulfonamide derivatives as potential GABAB agonists and their fragmentation to 3-aminopropanesulfinic acidEBI TBA
 11 Biological activity of 3-aminopropyl (methyl) phosphinic acid, a potent and selective GABAB agonist with CNS activityEBI TBA
10354414 5 Synthesis and pharmacology of the baclofen homologues 5-amino-4-(4-chlorophenyl)pentanoic acid and the R- and S-enantiomers of 5-amino-3-(4-chlorophenyl)pentanoic acid.EBI The Royal Danish School of Pharmacy
7650685 49 Phosphinic acid analogues of GABA. 2. Selective, orally active GABAB antagonists.EBI Ciba-Geigy AG
7650684 39 Phosphinic acid analogues of GABA. 1. New potent and selective GABAB agonists.EBI Ciba-Geigy AG
2995665 3 Synthesis and activity of 5-(aminomethylene)-1,3-cyclohexanediones: enolic analogues of gamma-aminobutyric acid.EBI TBA
26833890 18 Synthesis, Biological Evaluation, and Molecular Docking of 8-imino-2-oxo-2H,8H-pyrano[2,3-f]chromene Analogs: New Dual AChE Inhibitors as Potential Drugs for the Treatment of Alzheimer's Disease.BDB Yogi Vemana University