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Compounds Sorted by Binding Targets per Compound

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Compounds Sorted Alphabetically
Compound Name (alphabetical)
Binding Targets
Enz. Inhib. Data
ITC Data
Alternate Compound Names
  • 3-phosphoinositide dependent protein kinase-1
  • 5'-AMP-activated protein kinase Complex 1
  • 5'-AMP-activated protein kinase catalytic subunit alpha-2
  • ALK tyrosine kinase receptor
  • AP2-associated protein kinase 1
  • Aurora kinase A/Targeting protein for Xklp2
  • Axin-1/Glycogen synthase kinase-3 beta
  • BMP-2-inducible protein kinase
  • BR serine/threonine-protein kinase 1
  • CAMK2A
  • CAMK2B
  • CDK19/Cyclin C
  • CDK7/Cyclin H/MNAT1
  • CaM kinase I gamma
  • CaM kinase II
  • CaM-kinase kinase alpha
  • CaM-kinase kinase beta
  • Calmodulin/Proto-oncogene tyrosine-protein kinase Src
  • Citron Rho-interacting kinase
  • Cyclin-C
  • Cyclin-Dependent Kinase 9 (CDK9)
  • Cytoplasmic tyrosine-protein kinase BMX
  • Death-associated protein kinase 1
  • Death-associated protein kinase 2
  • Death-associated protein kinase 3
  • Dual specificity mitogen-activated protein kinase kinase 1/Mitogen-activated protein kinase 1/RAF proto-oncogene serine/threonine-protein kinase
  • Dual specificity mitogen-activated protein kinase kinase 6
  • Dual specificity protein kinase CLK1/CLK4
  • Dual specificity protein kinase CLK2
  • Dual specificity tyrosine-phosphorylation-regulated kinase 1B
  • Dual-specificity tyrosine-phosphorylation regulated kinase 1A
  • Ephrin receptor
  • Ephrin type-A receptor 7
  • Epithelial discoidin domain-containing receptor 1
  • Fibroblast growth factor receptor 1
  • Fibroblast growth factor receptor 2
  • Fibroblast growth factor receptor 3
  • Fibroblast growth factor receptor 4
  • Focal adhesion kinase 1/vascular endothelial growth factor receptor 3
  • Glycogen synthase kinase-3
  • Hepatocyte growth factor receptor
  • High affinity nerve growth factor receptor
  • Homeodomain-interacting protein kinase 2 (HIPK2)
  • Homeodomain-interacting protein kinase 3
  • Homeodomain-interacting protein kinase 4
  • Inhibitor of nuclear factor kappa-B kinase subunit epsilon
  • Insulin receptor
  • Interleukin-1 receptor-associated kinase 1
  • Interleukin-1 receptor-associated kinase 4
  • LIM domain kinase 1
  • Leukocyte tyrosine kinase receptor
  • MAP kinase-interacting serine/threonine-protein kinase 1/2
  • MAP/microtubule affinity-regulating kinase 2
  • MAP/microtubule affinity-regulating kinase 3
  • Macrophage colony-stimulating factor 1 receptor (CSF1R)
  • Maternal embryonic leucine zipper kinase
  • Mitogen-activated protein kinase 10
  • Mitogen-activated protein kinase 12
  • Mitogen-activated protein kinase 15
  • Mitogen-activated protein kinase 8
  • Mitogen-activated protein kinase 9
  • Mitogen-activated protein kinase kinase kinase 11
  • Mitogen-activated protein kinase kinase kinase 14
  • Mitogen-activated protein kinase kinase kinase 2
  • Mitogen-activated protein kinase kinase kinase 5
  • Mitogen-activated protein kinase kinase kinase 7
  • Mitogen-activated protein kinase kinase kinase 9
  • Mitogen-activated protein kinase kinase kinase kinase 1
  • Mitogen-activated protein kinase kinase kinase kinase 2
  • Mitogen-activated protein kinase kinase kinase kinase 5
  • Myosin light chain kinase, smooth muscle
  • Myosin-IIIB
  • Myotonin-protein kinase
  • NT-3 growth factor receptor
  • NUAK family SNF1-like kinase 1
  • NUAK family SNF1-like kinase 2
  • Non-receptor tyrosine-protein kinase TNK1
  • Non-receptor tyrosine-protein kinase TYK2
  • PKC alpha and beta-2
  • PTK2B protein tyrosine kinase 2 beta (PTK2B)
  • Peripheral plasma membrane protein CASK
  • Phosphorylase kinase
  • Platelet-derived growth factor receptor beta
  • Protein kinase C iota type/zeta type
  • Protein kinase C theta type
  • Protein kinase C, PKC; classical/novel
  • Protein kinase N1
  • Protein kinase N2
  • Proto-oncogene tyrosine-protein kinase receptor Ret
  • Receptor protein-tyrosine kinase erbB-4
  • Rho-associated protein kinase 1
  • Rho-associated protein kinase 2
  • Rhodopsin kinase
  • Ribosomal protein S6 kinase
  • Ribosomal protein S6 kinase (P70S6K)
  • Ribosomal protein S6 kinase alpha 1
  • Ribosomal protein S6 kinase alpha 2
  • Ribosomal protein S6 kinase alpha 6
  • Ribosomal protein S6 kinase alpha-1/alpha-3
  • Serine/threonine-protein kinase 16
  • Serine/threonine-protein kinase 17A
  • Serine/threonine-protein kinase 2
  • Serine/threonine-protein kinase 24
  • Serine/threonine-protein kinase 25
  • Serine/threonine-protein kinase 32A
  • Serine/threonine-protein kinase 32B
  • Serine/threonine-protein kinase 32C
  • Serine/threonine-protein kinase 33
  • Serine/threonine-protein kinase 38-like
  • Serine/threonine-protein kinase 4 (STK4)
  • Serine/threonine-protein kinase AKT
  • Serine/threonine-protein kinase AKT2
  • Serine/threonine-protein kinase D2
  • Serine/threonine-protein kinase DCLK3
  • Serine/threonine-protein kinase LATS2
  • Serine/threonine-protein kinase MARK1
  • Serine/threonine-protein kinase MRCK-A
  • Serine/threonine-protein kinase MST2
  • Serine/threonine-protein kinase MST4
  • Serine/threonine-protein kinase PAK 4
  • Serine/threonine-protein kinase PAK6
  • Serine/threonine-protein kinase PAK7
  • Serine/threonine-protein kinase PLK4
  • Serine/threonine-protein kinase SIK1
  • Serine/threonine-protein kinase SIK2
  • Serine/threonine-protein kinase Sgk1
  • Serine/threonine-protein kinase Sgk2
  • Serine/threonine-protein kinase Sgk3
  • Serine/threonine-protein kinase TAO1
  • Serine/threonine-protein kinase TAO3
  • Serine/threonine-protein kinase TBK1
  • Serine/threonine-protein kinase ULK1
  • Serine/threonine-protein kinase ULK2
  • Serine/threonine-protein kinase ULK3
  • Serine/threonine-protein kinase pim-1
  • TGF-beta receptor type II
  • TNNI3K
  • TRAF2- and NCK-interacting kinase
  • Testis-specific serine/threonine-protein kinase 1
  • Testis-specific serine/threonine-protein kinase 3
  • Tyrosine kinase non-receptor protein 2
  • Tyrosine-protein kinase ABL2
  • Tyrosine-protein kinase BTK
  • Tyrosine-protein kinase Blk
  • Tyrosine-protein kinase CSK
  • Tyrosine-protein kinase FER
  • Tyrosine-protein kinase FES
  • Tyrosine-protein kinase FRK
  • Tyrosine-protein kinase Fgr
  • Tyrosine-protein kinase Fyn
  • Tyrosine-protein kinase HCK
  • Tyrosine-protein kinase ITK/TSK
  • Tyrosine-protein kinase JAK3
  • Tyrosine-protein kinase Lck
  • Tyrosine-protein kinase Lyn
  • Tyrosine-protein kinase Mer
  • Tyrosine-protein kinase SYK
  • Tyrosine-protein kinase TEC
  • Tyrosine-protein kinase Yes
  • Tyrosine-protein kinase receptor TYRO3
  • Tyrosine-protein kinase receptor UFO
  • Vascular endothelial growth factor receptor 2
  • Vascular endothelial growth factor receptor 2 and tyrosine-protein kinase TIE-2 (KDR and TIE2)
  • Voltage-gated potassium channel subunit Kv7.1/Misshapen-like kinase 1
  • [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial
  • cAMP-dependent protein kinase (PKA)
  • cGMP-dependent protein kinase 1 beta
  • cGMP-dependent protein kinase 2
179 Kd
  • CHEMBL4576489