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IC50
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EC50
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-TΔS°
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Compounds Sorted by Binding Targets per Compound
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512
Compounds Sorted Alphabetically
Compound Name
(alphabetical)
Binding Targets
Enz. Inhib. Data
ITC Data
Alternate Compound Names
Ki
IC50
Kd
EC50
K
off
K
on
Other
BDBM50536675
3-phosphoinositide dependent protein kinase-1
5'-AMP-activated protein kinase Complex 1
Activin receptor type-1B
Aurora kinase A/B
Axin-1/Glycogen synthase kinase-3 beta
BRAF/CRAF
CaM kinase IV
Calmodulin/Proto-oncogene tyrosine-protein kinase Src
Casein kinase I isoform alpha
Casein kinase II subunit alpha
Cyclin-Dependent Kinase 5 (CDK5)
Cyclin-Dependent Kinase 9 (CDK9)
Cyclin-dependent kinase 2
Cyclin-dependent kinase 7
Cytoplasmic tyrosine-protein kinase BMX
Death-associated protein kinase 1
Dual specificity mitogen-activated protein kinase kinase 1/Mitogen-activated protein kinase 1/RAF proto-oncogene serine/threonine-protein kinase
Dual specificity mitogen-activated protein kinase kinase 6
Dual specificity protein kinase CLK2
Dual-specificity tyrosine-phosphorylation regulated kinase 1A
Ephrin receptor
Ephrin type-A receptor 3 (EPHA3)
Ephrin type-B receptor 2
Epidermal growth factor receptor
Fibroblast growth factor receptor 2
G protein-coupled receptor kinase 4
G protein-coupled receptor kinase 6
G-protein coupled receptor kinase 2
Glycogen synthase kinase-3
Hepatocyte growth factor receptor
High affinity nerve growth factor receptor
Inhibitor of NF-kappa-B kinase alpha/beta
Inhibitor of nuclear factor kappa-B kinase subunit epsilon
Insulin receptor
Insulin-like growth factor I receptor
Interleukin-1 receptor-associated kinase 1
Interleukin-1 receptor-associated kinase 4
Leucine-rich repeat serine/threonine-protein kinase 2
MAP kinase-activated protein kinase 2
MAP kinase-activated protein kinase 5
MAP/microtubule affinity-regulating kinase 4
Macrophage colony stimulating factor receptor
Mast/stem cell growth factor receptor Kit
Mitogen-activated protein kinase 14
Mitogen-activated protein kinase 8
Mitogen-activated protein kinase 9
NT-3 growth factor receptor
NUAK family SNF1-like kinase 1
Non-receptor tyrosine-protein kinase TYK2
PAK 1/CDC42
PAS domain-containing serine/threonine-protein kinase
Phosphoinositide 3-Kinase (PI3K), delta
Protein kinase C iota type/zeta type
Protein kinase C theta type
Protein kinase N1
RAC-alpha serine/threonine-protein kinase
RAF proto-oncogene serine/threonine-protein kinase
Receptor tyrosine-protein kinase erbB-2
Rho-associated protein kinase 1
Rho-associated protein kinase 2
Ribosomal protein S6 kinase (P70S6K)
Ribosomal protein S6 kinase alpha-1/alpha-3
Serine/threonine-protein kinase AKT
Serine/threonine-protein kinase AKT2
Serine/threonine-protein kinase Chk1/2
Serine/threonine-protein kinase MRCK-A
Serine/threonine-protein kinase MST4
Serine/threonine-protein kinase NEK2
Serine/threonine-protein kinase NEK6
Serine/threonine-protein kinase Nek4
Serine/threonine-protein kinase PLK1
Serine/threonine-protein kinase SRPK1
Serine/threonine-protein kinase Sgk1
Serine/threonine-protein kinase TAO2
Serine/threonine-protein kinase TBK1
Serine/threonine-protein kinase c-TAK1
Serine/threonine-protein kinase pim-1
Sphingosine kinase 1
Testis-specific serine/threonine-protein kinase 1
Tyrosine-protein kinase ABL1
Tyrosine-protein kinase BRK
Tyrosine-protein kinase BTK
Tyrosine-protein kinase HCK
Tyrosine-protein kinase ITK/TSK
Tyrosine-protein kinase JAK1
Tyrosine-protein kinase JAK2
Tyrosine-protein kinase JAK3
Tyrosine-protein kinase Lck
Tyrosine-protein kinase SYK
Tyrosine-protein kinase ZAP-70
Tyrosine-protein kinase receptor FLT3
Vascular endothelial growth factor receptor 2
Vascular endothelial growth factor receptor 2 and tyrosine-protein kinase TIE-2 (KDR and TIE2)
Voltage-gated potassium channel subunit Kv7.1/Misshapen-like kinase 1
cAMP-dependent protein kinase (PKA)
p38 delta/gamma
0
100
0
0
0
0
0
0
CHEMBL4569508
BDBM50536678
3-phosphoinositide dependent protein kinase-1
5'-AMP-activated protein kinase Complex 1
Activin receptor type-1B
Aurora kinase A/B
Axin-1/Glycogen synthase kinase-3 beta
BRAF/CRAF
CaM kinase IV
Calmodulin/Proto-oncogene tyrosine-protein kinase Src
Casein kinase I isoform alpha
Casein kinase II subunit alpha
Cyclin-Dependent Kinase 5 (CDK5)
Cyclin-Dependent Kinase 9 (CDK9)
Cyclin-dependent kinase 2
Cyclin-dependent kinase 7
Cytoplasmic tyrosine-protein kinase BMX
Death-associated protein kinase 1
Dual specificity mitogen-activated protein kinase kinase 1/Mitogen-activated protein kinase 1/RAF proto-oncogene serine/threonine-protein kinase
Dual specificity mitogen-activated protein kinase kinase 6
Dual specificity protein kinase CLK2
Dual-specificity tyrosine-phosphorylation regulated kinase 1A
Ephrin receptor
Ephrin type-A receptor 3 (EPHA3)
Ephrin type-B receptor 2
Epidermal growth factor receptor
Fibroblast growth factor receptor 2
G protein-coupled receptor kinase 4
G protein-coupled receptor kinase 6
G-protein coupled receptor kinase 2
Glycogen synthase kinase-3
Hepatocyte growth factor receptor
High affinity nerve growth factor receptor
Inhibitor of NF-kappa-B kinase alpha/beta
Inhibitor of nuclear factor kappa-B kinase subunit epsilon
Insulin receptor
Insulin-like growth factor I receptor
Interleukin-1 receptor-associated kinase 1
Interleukin-1 receptor-associated kinase 4
Leucine-rich repeat serine/threonine-protein kinase 2
MAP kinase-activated protein kinase 2
MAP kinase-activated protein kinase 5
MAP/microtubule affinity-regulating kinase 4
Macrophage colony stimulating factor receptor
Mast/stem cell growth factor receptor Kit
Mitogen-activated protein kinase 14
Mitogen-activated protein kinase 8
Mitogen-activated protein kinase 9
NT-3 growth factor receptor
NUAK family SNF1-like kinase 1
Non-receptor tyrosine-protein kinase TYK2
PAK 1/CDC42
PAS domain-containing serine/threonine-protein kinase
Phosphoinositide 3-Kinase (PI3K), delta
Protein kinase C iota type/zeta type
Protein kinase C theta type
Protein kinase N1
RAC-alpha serine/threonine-protein kinase
RAF proto-oncogene serine/threonine-protein kinase
Receptor tyrosine-protein kinase erbB-2
Rho-associated protein kinase 1
Rho-associated protein kinase 2
Ribosomal protein S6 kinase (P70S6K)
Ribosomal protein S6 kinase alpha-1/alpha-3
Serine/threonine-protein kinase AKT
Serine/threonine-protein kinase AKT2
Serine/threonine-protein kinase Chk1/2
Serine/threonine-protein kinase MRCK-A
Serine/threonine-protein kinase MST4
Serine/threonine-protein kinase NEK2
Serine/threonine-protein kinase NEK6
Serine/threonine-protein kinase Nek4
Serine/threonine-protein kinase PLK1
Serine/threonine-protein kinase SRPK1
Serine/threonine-protein kinase Sgk1
Serine/threonine-protein kinase TAO2
Serine/threonine-protein kinase TBK1
Serine/threonine-protein kinase c-TAK1
Serine/threonine-protein kinase pim-1
Sphingosine kinase 1
Testis-specific serine/threonine-protein kinase 1
Tyrosine-protein kinase ABL1
Tyrosine-protein kinase BRK
Tyrosine-protein kinase BTK
Tyrosine-protein kinase HCK
Tyrosine-protein kinase ITK/TSK
Tyrosine-protein kinase JAK1
Tyrosine-protein kinase JAK2
Tyrosine-protein kinase JAK3
Tyrosine-protein kinase Lck
Tyrosine-protein kinase SYK
Tyrosine-protein kinase ZAP-70
Tyrosine-protein kinase receptor FLT3
Vascular endothelial growth factor receptor 2
Vascular endothelial growth factor receptor 2 and tyrosine-protein kinase TIE-2 (KDR and TIE2)
Voltage-gated potassium channel subunit Kv7.1/Misshapen-like kinase 1
cAMP-dependent protein kinase (PKA)
p38 delta/gamma
0
100
0
0
0
0
0
0
CHEMBL4550702
BDBM50536681
3-phosphoinositide dependent protein kinase-1
5'-AMP-activated protein kinase Complex 1
Activin receptor type-1B
Aurora kinase A/B
Axin-1/Glycogen synthase kinase-3 beta
BRAF/CRAF
CaM kinase IV
Calmodulin/Proto-oncogene tyrosine-protein kinase Src
Casein kinase I isoform alpha
Casein kinase II subunit alpha
Cyclin-Dependent Kinase 5 (CDK5)
Cyclin-Dependent Kinase 9 (CDK9)
Cyclin-dependent kinase 2
Cyclin-dependent kinase 7
Cytoplasmic tyrosine-protein kinase BMX
Death-associated protein kinase 1
Dual specificity mitogen-activated protein kinase kinase 1/Mitogen-activated protein kinase 1/RAF proto-oncogene serine/threonine-protein kinase
Dual specificity mitogen-activated protein kinase kinase 6
Dual specificity protein kinase CLK2
Dual-specificity tyrosine-phosphorylation regulated kinase 1A
Ephrin receptor
Ephrin type-A receptor 3 (EPHA3)
Ephrin type-B receptor 2
Epidermal growth factor receptor
Fibroblast growth factor receptor 2
G protein-coupled receptor kinase 4
G protein-coupled receptor kinase 6
G-protein coupled receptor kinase 2
Glycogen synthase kinase-3
Hepatocyte growth factor receptor
High affinity nerve growth factor receptor
Inhibitor of NF-kappa-B kinase alpha/beta
Inhibitor of nuclear factor kappa-B kinase subunit epsilon
Insulin receptor
Insulin-like growth factor I receptor
Interleukin-1 receptor-associated kinase 1
Interleukin-1 receptor-associated kinase 4
Leucine-rich repeat serine/threonine-protein kinase 2
MAP kinase-activated protein kinase 2
MAP kinase-activated protein kinase 5
MAP/microtubule affinity-regulating kinase 4
Macrophage colony stimulating factor receptor
Mast/stem cell growth factor receptor Kit
Mitogen-activated protein kinase 14
Mitogen-activated protein kinase 8
Mitogen-activated protein kinase 9
NT-3 growth factor receptor
NUAK family SNF1-like kinase 1
Non-receptor tyrosine-protein kinase TYK2
PAK 1/CDC42
PAS domain-containing serine/threonine-protein kinase
Phosphoinositide 3-Kinase (PI3K), delta
Protein kinase C iota type/zeta type
Protein kinase C theta type
Protein kinase N1
RAC-alpha serine/threonine-protein kinase
RAF proto-oncogene serine/threonine-protein kinase
Receptor tyrosine-protein kinase erbB-2
Rho-associated protein kinase 1
Rho-associated protein kinase 2
Ribosomal protein S6 kinase (P70S6K)
Ribosomal protein S6 kinase alpha-1/alpha-3
Serine/threonine-protein kinase AKT
Serine/threonine-protein kinase AKT2
Serine/threonine-protein kinase Chk1/2
Serine/threonine-protein kinase MRCK-A
Serine/threonine-protein kinase MST4
Serine/threonine-protein kinase NEK2
Serine/threonine-protein kinase NEK6
Serine/threonine-protein kinase Nek4
Serine/threonine-protein kinase PLK1
Serine/threonine-protein kinase SRPK1
Serine/threonine-protein kinase Sgk1
Serine/threonine-protein kinase TAO2
Serine/threonine-protein kinase TBK1
Serine/threonine-protein kinase c-TAK1
Serine/threonine-protein kinase pim-1
Sphingosine kinase 1
Testis-specific serine/threonine-protein kinase 1
Tyrosine-protein kinase ABL1
Tyrosine-protein kinase BRK
Tyrosine-protein kinase BTK
Tyrosine-protein kinase HCK
Tyrosine-protein kinase ITK/TSK
Tyrosine-protein kinase JAK1
Tyrosine-protein kinase JAK2
Tyrosine-protein kinase JAK3
Tyrosine-protein kinase Lck
Tyrosine-protein kinase SYK
Tyrosine-protein kinase ZAP-70
Tyrosine-protein kinase receptor FLT3
Vascular endothelial growth factor receptor 2
Vascular endothelial growth factor receptor 2 and tyrosine-protein kinase TIE-2 (KDR and TIE2)
Voltage-gated potassium channel subunit Kv7.1/Misshapen-like kinase 1
cAMP-dependent protein kinase (PKA)
p38 delta/gamma
0
100
0
0
0
0
0
0
CHEMBL4552628