Compile Data Set for Download or QSAR
maximum 50k data
Found 50 of affinity data for UniProtKB/TrEMBL: Q5S006
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50582730(CHEMBL5087055)
Affinity DataIC50:  11nMAssay Description:Inhibition of LRRK2-WT in C57BL/6 mouse brain at 10 to 150 mg/kg and measured after 1 hrs by western blottingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50582730(CHEMBL5087055)
Affinity DataIC50:  16nMAssay Description:Inhibition of LRRK2-WT-pSER935 in C57BL/6 mouse brain at 10 to 150 mg/kg and measured after 1 hrs by western blottingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50582731(CHEMBL5092087)
Affinity DataIC50:  22nMAssay Description:Inhibition of LRRK2-WT in C57BL/6 mouse brain at 10 to 150 mg/kg and measured after 1 hrs by western blottingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50582731(CHEMBL5092087)
Affinity DataIC50:  23nMAssay Description:Inhibition of LRRK2-WT-pSER935 in C57BL/6 mouse brain at 10 to 150 mg/kg and measured after 1 hrs by western blottingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597147(CHEMBL5183984)
Affinity DataEC50:  1.22E+4nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597148(CHEMBL5196289)
Affinity DataEC50:  2.10E+3nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597149(CHEMBL5185136)
Affinity DataEC50:  3.20E+3nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597150(CHEMBL5184765)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597151(CHEMBL5207757)
Affinity DataEC50:  5.70E+4nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597152(CHEMBL5191932)
Affinity DataEC50:  1.50E+4nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597153(CHEMBL5197009)
Affinity DataEC50:  800nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597154(CHEMBL5202841)
Affinity DataEC50:  1.50E+3nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597155(CHEMBL5199105)
Affinity DataEC50:  6.40E+3nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597156(CHEMBL5173076)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597157(CHEMBL5204372)
Affinity DataEC50:  1.08E+3nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597158(CHEMBL5185437)
Affinity DataEC50:  1.38E+3nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597159(CHEMBL5208171)
Affinity DataEC50:  1.67E+4nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597160(CHEMBL5177578)
Affinity DataEC50:  290nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597161(CHEMBL5173029)
Affinity DataEC50:  340nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597162(CHEMBL5200500)
Affinity DataEC50:  750nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597182(CHEMBL5181966)
Affinity DataEC50:  5.40E+3nMAssay Description:Inhibition of mouse full-length wild type LRRK2 transfected in HEK293 cells using LRRKtide as substrate incubated for 1 hr in presence of ATP by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597164(CHEMBL5179102)
Affinity DataEC50:  760nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597165(CHEMBL5190962)
Affinity DataEC50:  920nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597166(CHEMBL5198878)
Affinity DataEC50:  600nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597167(CHEMBL5207466)
Affinity DataEC50:  1.34E+4nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597168(CHEMBL5185379)
Affinity DataEC50:  2.17E+4nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597169(CHEMBL5198788)
Affinity DataEC50:  4.90E+3nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597170(CHEMBL5195211)
Affinity DataEC50:  1.43E+4nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597171(CHEMBL5170238)
Affinity DataEC50:  260nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597172(CHEMBL5187306)
Affinity DataEC50:  600nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597173(CHEMBL5202898)
Affinity DataEC50:  4.78E+3nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597174(CHEMBL5170423)
Affinity DataEC50:  1.96E+4nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597175(CHEMBL5199239)
Affinity DataEC50:  1.28E+3nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597176(CHEMBL5170225)
Affinity DataEC50:  690nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597177(CHEMBL5172291)
Affinity DataEC50:  390nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597178(CHEMBL5174380)
Affinity DataEC50:  390nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597179(CHEMBL5198203)
Affinity DataEC50:  1.71E+3nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597180(CHEMBL5194234)
Affinity DataEC50:  1.44E+3nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597181(CHEMBL5207639)
Affinity DataEC50:  3.12E+3nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597182(CHEMBL5181966)
Affinity DataEC50:  280nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597148(CHEMBL5196289)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of mouse full-length wild type LRRK2 transfected in HEK293 cells using LRRKtide as substrate incubated for 1 hr in presence of ATP by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597154(CHEMBL5202841)
Affinity DataEC50:  7.60E+4nMAssay Description:Inhibition of mouse full-length wild type LRRK2 transfected in HEK293 cells using LRRKtide as substrate incubated for 1 hr in presence of ATP by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597160(CHEMBL5177578)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of mouse full-length wild type LRRK2 transfected in HEK293 cells using LRRKtide as substrate incubated for 1 hr in presence of ATP by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597171(CHEMBL5170238)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of mouse full-length wild type LRRK2 transfected in HEK293 cells using LRRKtide as substrate incubated for 1 hr in presence of ATP by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597178(CHEMBL5174380)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of mouse full-length wild type LRRK2 transfected in HEK293 cells using LRRKtide as substrate incubated for 1 hr in presence of ATP by TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597146(CHEMBL5188336)
Affinity DataEC50:  1.22E+4nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597145(CHEMBL5198175)
Affinity DataEC50:  8.00E+4nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597144(CHEMBL5205363)
Affinity DataEC50:  5.10E+3nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM257207(US9493440, 51)
Affinity DataEC50:  30nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Mus musculus)
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50597163(CHEMBL5190480)
Affinity DataEC50:  2.31E+3nMAssay Description:Inhibition of mouse full-length LRRK2 G2019S mutant transfected in HEK293 cells using LRRKtide as substrate in presence of ATP by incubated for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed