BDBM101739 US9695160, 33::US9796707, Compound 33

SMILES FC(F)(F)c1ccc(N2CCN(Cc3ccccn3)CC2)c(NC(=O)c2cnc(o2)-c2ccccc2)c1

InChI Key InChIKey=CLWSDTWEUVBGNB-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 101739   

TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM101739(US9695160, 33 | US9796707, Compound 33)
Affinity DataIC50:  4.03E+3nMAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSRSF protein kinase 1(Homo sapiens (Human))
The University Of Nottingham

US Patent
LigandPNGBDBM101739(US9695160, 33 | US9796707, Compound 33)
Affinity DataIC50:  4.03E+3nMT: 2°CAssay Description:Candidate compounds were screened by the Kinase-Glo assay (Promega; Koresawa and Okabe, 2004), the results of which are shown in Table 1 and Table 2....More data for this Ligand-Target Pair
In DepthDetails US Patent