BDBM172643 US9090628, 303

SMILES CC(C)n1nc(C)nc1-c1cn2CCOc3cnc(cc3-c2n1)[C@H](C)N1CCN(CC1)C(C)(C)C

InChI Key InChIKey=DKDCWBXTCFPFMR-SFHVURJKSA-N

Data  1 KI  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 172643   

LigandPNGBDBM172643(US9090628, 303)
Affinity DataKi:  1.90nMAssay Description:Binding affinity to PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM172643(US9090628, 303)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of PI3Kdelta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM172643(US9090628, 303)
Affinity DataIC50:  28nMAssay Description:Inhibition of PI3Kdelta in human whole blood assessed as suppression of CD69 expressionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM172643(US9090628, 303)
Affinity DataIC50:  1.92nMpH: 7.5Assay Description:PI3K enzymatic activity was assayed by measuring the amount of product phosphatidylinositol 3,4,5-phosphate (PIP3) formed from substrate 4,5 phosphat...More data for this Ligand-Target Pair
In DepthDetails US Patent