BDBM17281 7-({2-[(1-ethanimidoylpiperidin-4-yl)oxy]-9H-carbazol-9-yl}methyl)naphthalene-2-carboximidamide::CHEMBL369251::Naphthylamidine template, II::ZK-806450
SMILES CC(=N)N1CCC(CC1)Oc1ccc2c(c1)n(Cc1ccc3ccc(cc3c1)C(N)=N)c1ccccc21
InChI Key InChIKey=DZLGSWPXZYDHBD-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 17281
Affinity DataKi: 1.60nM ΔG°: -11.9kcal/molepH: 7.5 T: 2°CAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:In vitro inhibition of human Coagulation factor X.More data for this Ligand-Target Pair
Affinity DataKi: 36nM ΔG°: -10.0kcal/molepH: 7.5 T: 2°CAssay Description:The enzyme activities were determined kinetically as the initial rate of cleavage of a peptide p-nitroanilide. Km for enzyme and substrate was determ...More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:In vitro inhibition of human Coagulation factor II.More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:In vitro inhibition of bovine trypsin.More data for this Ligand-Target Pair