BDBM193783 US9670208, Example 563 2-cyclopropyl-1-(7-(2-((1-methyl-1H-pyrazol-5-yl)amino)pyrimidin-4-yl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl)propan-2-ol

SMILES Cn1nccc1Nc1nccc(n1)-c1ccn2c(CC(C)(O)C3CC3)nnc2c1

InChI Key InChIKey=YSUHBTDQGGGTSK-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 193783   

TargetMitogen-activated protein kinase 1 [8-360](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM193783(US9670208, Example 563 2-cyclopropyl-1-(7-(2-((1-m...)
Affinity DataIC50:  661nMpH: 7.3Assay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent