BDBM224632 US9328111, 5
SMILES Cc1ccc2c3c(n[nH]c2=O)c2CCCCc2[nH]c13
InChI Key InChIKey=NZZXITVESFGTFK-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 224632
Affinity DataIC50: 70.7nMpH: 8.0Assay Description:PARP1 enzymatic assay was conducted using a method modified from HT F Homogeneous PARP Inhibition Assay Kit (Trevigen). 8.8 nM PARP1 was pre-incubate...More data for this Ligand-Target Pair