BDBM23918 3-amidinophenylalanine deriv., 60::4-amino-N-(3-{[(2S)-1-[4-(2-aminoethyl)piperidin-1-yl]-3-(3-carbamimidoylphenyl)-1-oxopropan-2-yl]sulfamoyl}phenyl)butanamide

SMILES NCCCC(=O)Nc1cccc(c1)S(=O)(=O)N[C@@H](Cc1cccc(c1)C(N)=N)C(=O)N1CCC(CCN)CC1

InChI Key InChIKey=JFUQGOKQNWYPFR-DEOSSOPVSA-N

Data  5 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 23918   

TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Curacyte Chemistry

LigandPNGBDBM23918(3-amidinophenylalanine deriv., 60 | 4-amino-N-(3-{...)
Affinity DataKi:  3.90nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Curacyte Chemistry

LigandPNGBDBM23918(3-amidinophenylalanine deriv., 60 | 4-amino-N-(3-{...)
Affinity DataKi:  2.50E+3nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Curacyte Chemistry

LigandPNGBDBM23918(3-amidinophenylalanine deriv., 60 | 4-amino-N-(3-{...)
Affinity DataKi:  8.00E+3nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
Curacyte Chemistry

LigandPNGBDBM23918(3-amidinophenylalanine deriv., 60 | 4-amino-N-(3-{...)
Affinity DataKi:  2.10E+4nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Bos taurus)
Curacyte Chemistry

LigandPNGBDBM23918(3-amidinophenylalanine deriv., 60 | 4-amino-N-(3-{...)
Affinity DataKi:  2.30E+4nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed