BDBM29501 Pyrazolo[1,5-a]-1,3,5-triazine, 13-26

SMILES CCN(C)c1nc(C)nc2c(c(C)nn12)-c1ccc(OC)nc1C


Data  1 IC50

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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 29501   

TargetCorticotropin-releasing factor receptor 1(Rattus norvegicus (rat))
Bristol-Myers Squibb Co.

LigandPNGBDBM29501(Pyrazolo[1,5-a]-1,3,5-triazine, 13-26)
Show SMILES CCN(C)c1nc(C)nc2c(c(C)nn12)-c1ccc(OC)nc1C
Show InChI InChI=1S/C17H22N6O/c1-7-22(5)17-20-12(4)19-16-15(11(3)21-23(16)17)13-8-9-14(24-6)18-10(13)2/h8-9H,7H2,1-6H3
Affinity DataIC50: 81.6nMpH: 7.2 T: 2°CAssay Description:Naive rats were sacrificed by decapitation, and the brain and pituitary were collected. Slide-mounted brain sections were preincubated in an assay so...More data for this Ligand-Target Pair