BDBM29983 arylpyrazole, 28

SMILES Cc1c(CN[C@H]2CC[C@@H](F)C2)nn(c1-c1ccc(C)nc1)-c1ncccc1Cl

InChI Key InChIKey=BUSSQQRPMMHCBN-SJORKVTESA-N

Data  2 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 29983   

TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Banyu Pharmaceutical

LigandPNGBDBM29983(arylpyrazole, 28)
Affinity DataIC50:  2.90E+4nMAssay Description:Binding affinity to the hERG K+ channel was measured by displacement of [35S]-radiolabeled MK499 in membranes derived from HEK 293 cells stably trans...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Banyu Pharmaceutical

LigandPNGBDBM29983(arylpyrazole, 28)
Affinity DataIC50:  2.5nM EC50:  1nMAssay Description:Compounds were tested for their inhibitory effects on ligand binding to the human ORL1 receptor. Bound and free radioligands are separated by filtra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed