BDBM318043 8-Methyl-2-[4-[(3-methyl- pyrazin-2-yl)methyl]piperazin- 1-yl]-3,5,6,7- tetrahydropyrido[2,3- d]pyrimidin-4-one::US9624218, Example 44
SMILES CN1CCCc2c1nc([nH]c2=O)N1CCN(Cc2nccnc2C)CC1
InChI Key InChIKey=WLVFPFBPOHXOMK-UHFFFAOYSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 318043
Affinity DataIC50: 17.6nMAssay Description:The enzymatic activity of hTNKS1 and hTNKS2 is assessed using an enzyme-linked immunosorbent assay (ELISA) which detects poly ADP ribose incorporated...More data for this Ligand-Target Pair
Affinity DataIC50: 5.83E+3nMAssay Description:The Poly ADP-ribose polymerase 1(PARP1) assay is an ELISA which detects poly ADP ribose incorporated into plate-bound histone protein in a 384-well f...More data for this Ligand-Target Pair
Affinity DataIC50: 12.7nMAssay Description:The enzymatic activity of hTNKS1 and hTNKS2 is assessed using an enzyme-linked immunosorbent assay (ELISA) which detects poly ADP ribose incorporated...More data for this Ligand-Target Pair