BDBM327895 (4-(4- fluorobenzyl)piperazin- 1-yl)(6-(4- phenoxyphenylamino) pyridin-3-yl)methanone::US10377742, Compound 34::US9663496, Compound 34

SMILES Fc1ccc(CN2CCN(CC2)C(=O)c2ccc(Nc3ccc(Oc4ccccc4)cc3)nc2)cc1

InChI Key InChIKey=SCZKOAZZRCYNFT-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 327895   

Target5'-AMP-activated protein kinase catalytic subunit alpha-2(Homo sapiens (Human))
Rigel Pharmaceuticals

US Patent
LigandPNGBDBM327895((4-(4- fluorobenzyl)piperazin- 1-yl)(6-(4- phenoxy...)
Affinity DataEC50:  3.00E+3nMAssay Description:Compounds were assayed for their ability to activate AMPK using an enzyme-linked immunosorbent assay. Reagents and procedures for measuring AMPK acti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5'-AMP-activated protein kinase catalytic subunit alpha-2(Homo sapiens (Human))
Rigel Pharmaceuticals

US Patent
LigandPNGBDBM327895((4-(4- fluorobenzyl)piperazin- 1-yl)(6-(4- phenoxy...)
Affinity DataEC50:  3.00E+3nMAssay Description:Compounds were assayed for their ability to activate AMPK using an enzyme-linked immunosorbent assay. Reagents and procedures for measuring AMPK acti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent