BDBM368240 US10227338, Example 21::US10227338, Example 52
SMILES CNC1CCN(C1)c1ccccc1Nc1cc(F)c(cc1Cl)S(=O)(=O)Nc1cscn1
InChI Key InChIKey=SGUPKIRVVDCQRR-UHFFFAOYSA-N
Data 4 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 368240
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Daewoong Pharmaceutical
US Patent
Daewoong Pharmaceutical
US Patent
Affinity DataIC50: 66nMAssay Description:In order to measure the sodium ion channel blocking effect, an IonFlux16 Auto patch clamp system (Fluxion, Inc.) and a plate for exclusive use were u...More data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Daewoong Pharmaceutical
US Patent
Daewoong Pharmaceutical
US Patent
Affinity DataIC50: >1.00E+4nMAssay Description:In order to measure the sodium ion channel blocking effect, an IonFlux16 Auto patch clamp system (Fluxion, Inc.) and a plate for exclusive use were u...More data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
Daewoong Pharmaceutical
US Patent
Daewoong Pharmaceutical
US Patent
Affinity DataIC50: >3.00E+3nMAssay Description:In order to measure the sodium ion channel blocking effect, an IonFlux16 Auto patch clamp system (Fluxion, Inc.) and a plate for exclusive use were u...More data for this Ligand-Target Pair
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Daewoong Pharmaceutical
US Patent
Daewoong Pharmaceutical
US Patent
Affinity DataIC50: 61nMAssay Description:In order to measure the sodium ion channel blocking effect, an IonFlux16 Auto patch clamp system (Fluxion, Inc.) and a plate for exclusive use were u...More data for this Ligand-Target Pair