BDBM391729 3,5-dibromo-Nalpha-[(2'-oxo-::US10300056, Example 14::US10888561, Example 14

SMILES Oc1c(Br)cc(C[C@@H](NC(=O)N2CCC3(CC2)OC(=O)Nc2ncccc32)C(=O)N[C@@H](CC2CCNCC2)C(=O)N2CCN(CC2)c2ccncc2)cc1Br

InChI Key InChIKey=PIYNZUIYDJFKLR-JSOSNVBQSA-N

Data  2 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 391729   

TargetReceptor activity-modifying protein 1(Homo sapiens (Human))
Heptares Therapeutics

US Patent
LigandPNGBDBM391729(3,5-dibromo-Nalpha-[(2'-oxo- | US10300056, Example...)
Affinity DataKi:  0.0790nMAssay Description:Radioligand binding assay. Human CGRP receptors expressed (consisting of CRLR and RAMP1) in insect Sf21 cell membrane homogenates were re-suspended i...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor activity-modifying protein 1(Homo sapiens (Human))
Heptares Therapeutics

US Patent
LigandPNGBDBM391729(3,5-dibromo-Nalpha-[(2'-oxo- | US10300056, Example...)
Affinity DataKi:  0.0790nMAssay Description:Human CGRP receptors expressed (consisting of CRLR and RAMP1) in insect Sf21 cell membrane homogenates were re-suspended in the binding buffer (10 mM...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent