BDBM437344 1-(5-(1-benzyl-1H-pyrazol-4-yl)-1-methyl-2-oxo-1,2- dihydropyridin-4-yl)-N,N-dimethyl-1H-pyrrole-3-carboxamide::US10617680, Example 78::US11020380, Example 78

SMILES CN(C)C(=O)c1ccn(c1)-c1cc(=O)n(C)cc1-c1cnn(Cc2ccccc2)c1

InChI Key InChIKey=NGCFPHAEVPYKKM-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 437344   

TargetCREB-binding protein(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM437344(1-(5-(1-benzyl-1H-pyrazol-4-yl)-1-methyl-2-oxo-1,2...)
Affinity DataIC50: <500nMAssay Description:The CBP-inhibitory activity of the compounds described herein was determined by calculating the IC50. More specifically, CBP inhibitor activity was a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCREB-binding protein(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM437344(1-(5-(1-benzyl-1H-pyrazol-4-yl)-1-methyl-2-oxo-1,2...)
Affinity DataIC50: <500nMAssay Description:The CBP-inhibitory activity of the compounds described herein was determined by calculating the IC50. More specifically, CBP inhibitor activity was a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent