BDBM437368 4-ethoxy-1-methyl-5-(1-(4-(1-methyl-1H-pyrazol-4-yl)benzyl)- 1H-pyrazol-4-yl)pyridin-2(1H)-one::US10617680, Example 102::US11020380, Example 102

SMILES CCOc1cc(=O)n(C)cc1-c1cnn(Cc2ccc(cc2)-c2cnn(C)c2)c1

InChI Key InChIKey=AHRNUSRCZJSRKE-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 437368   

TargetCREB-binding protein(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM437368(4-ethoxy-1-methyl-5-(1-(4-(1-methyl-1H-pyrazol-4-y...)
Affinity DataIC50: <500nMAssay Description:The CBP-inhibitory activity of the compounds described herein was determined by calculating the IC50. More specifically, CBP inhibitor activity was a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCREB-binding protein(Homo sapiens (Human))
Celgene Quanticel Research

US Patent
LigandPNGBDBM437368(4-ethoxy-1-methyl-5-(1-(4-(1-methyl-1H-pyrazol-4-y...)
Affinity DataIC50: <500nMAssay Description:The CBP-inhibitory activity of the compounds described herein was determined by calculating the IC50. More specifically, CBP inhibitor activity was a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent