BDBM438835 N-{[5-(Ethylsulfonyl)pyridin-2-yl]methyl}-1″-(1R)-1-[2-(trifluoromethyl)pyrimidin-5-yl]ethyl-4′H-dispiro[cyclopropane-1,5′-thieno[2,3-c]pyran-7′,4″-piperidine]-2′-carboxamide::US10603320, Example 7
SMILES CCS(=O)(=O)c1ccc(CNC(=O)c2cc3CC4(CC4)OC4(CCN(CC4)[C@H](C)c4cnc(nc4)C(F)(F)F)c3s2)nc1
InChI Key InChIKey=GPFKJSWERRLMSX-GOSISDBHSA-N
Data 3 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 438835
Affinity DataKi: 6.40nMAssay Description:His-tagged human RAR-related orphan receptor alpha (hRORa), human RAR-related orphan receptor beta (hRORb), and human RAR-related orphan receptor gam...More data for this Ligand-Target Pair
Affinity DataKi: 3.46E+3nMAssay Description:His-tagged human RAR-related orphan receptor alpha (hRORa), human RAR-related orphan receptor beta (hRORb), and human RAR-related orphan receptor gam...More data for this Ligand-Target Pair
Affinity DataKi: >1.25E+4nMAssay Description:His-tagged human RAR-related orphan receptor alpha (hRORa), human RAR-related orphan receptor beta (hRORb), and human RAR-related orphan receptor gam...More data for this Ligand-Target Pair