BDBM499339 N-(cyclopropylsulfonyl)-4-((3- (6-((tetrahydro-2H-pyran-4- yl)methoxy)pyridin-3- yl)phenoxy)methyl)benzamide::US11020381, Example 29

SMILES O=C(NS(=O)(=O)C1CC1)c1ccc(COc2cccc(c2)-c2ccc(OCC3CCOCC3)nc2)cc1

InChI Key InChIKey=VBUAUOXOJQAZLT-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 499339   

TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Raqualia Pharma

US Patent
LigandPNGBDBM499339(N-(cyclopropylsulfonyl)-4-((3- (6-((tetrahydro-2H-...)
Affinity DataIC50: <500nMAssay Description:This screen is used to determine the effects of compounds on human Nav1.7 channels, utilizing electrical field stimulation (EFS) system in 96-well pl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent