BDBM499443 4-((3-(5-(cyclopropylmethoxy) pyrazin- 2-yl)-4-fluorophenoxy) methyl)-3-fluoro- N-(methylsulfonyl)benzamide::US11020381, Example 139

SMILES CS(=O)(=O)NC(=O)c1ccc(COc2ccc(F)c(c2)-c2cnc(OCC3CC3)cn2)c(F)c1

InChI Key InChIKey=UMXYLADVVAMHQA-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 499443   

TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Raqualia Pharma

US Patent
LigandPNGBDBM499443(4-((3-(5-(cyclopropylmethoxy) pyrazin- 2-yl)-4-flu...)
Affinity DataIC50: <500nMAssay Description:This screen is used to determine the effects of compounds on human Nav1.7 channels, utilizing electrical field stimulation (EFS) system in 96-well pl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent