BDBM499542 US11020395, Example 138.0

SMILES CO[C@@H]([C@H](C)S(=O)(=O)Nc1nnc(C2CCC2)n1-c1c(OC)cccc1OC)c1cnc(C)cn1

InChI Key InChIKey=AXKYIAPDCRBQJE-BTYIYWSLSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 499542   

TargetApelin receptor(Homo sapiens (Human))
Amgen

US Patent
LigandPNGBDBM499542(US11020395, Example 138.0)
Affinity DataEC50:  27nMAssay Description:The human APJ receptor was cloned by polymerase chain reaction and the gene encoding the receptor was subcloned in pFLAG-CMV™-3 expression vector (Si...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent