BDBM50001462 3-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-propionylamino}-indane-2-carbonyl)-amino]-N-{1-[1-(carbamoylmethyl-carbamoyl)-2-methyl-propylcarbamoyl]-2-methyl-propyl}-succinamic acid::CHEMBL124435::H-Tyr-D-Ala-Aic-Asp-Val-Val-Gly-NH2
SMILES CC(C)[C@H](NC(=O)[C@@H](NC(=O)[C@H](CC(O)=O)NC(=O)C1(Cc2ccccc2C1)NC(=O)[C@@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(C)C)C(=O)NCC(N)=O
InChI Key InChIKey=QZYUFPDOTMWDCQ-UZHHEQFGSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 8 hits for monomerid = 50001462
Affinity DataKi: 0.200nMAssay Description:Binding affinity was determined on delta [3H]-DPDPE site in rat brain synaptosomes by radioreceptor assayMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibition of [3H]- ]DSLET binding to Opioid receptor delta 1 from rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 56nMAssay Description:Binding affinity was determined on mu [3H]-DAGO site in rat brain synaptosomes by radioreceptor assayMore data for this Ligand-Target Pair
Affinity DataKi: 207nMAssay Description:Inhibition of [3H]- ]DAMGO binding to Opioid receptor mu 1 from rat brain membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 290nMAssay Description:Inhibition of electrically evoked contractions in Guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0803nMAssay Description:Inhibition of electrically evoked contractions in mouse vas deferensMore data for this Ligand-Target Pair
Affinity DataIC50: 0.410nMAssay Description:Tested for inhibition of amplification of electrically induced twitch in mouse vas deferens (MVD)More data for this Ligand-Target Pair
Affinity DataIC50: 369nMAssay Description:Tested for inhibition of amplification of electrically induced twitch in guinea pig ileum (GPI)More data for this Ligand-Target Pair