BDBM50001915 1-(3-chlorophenyl)piperazine::CHEMBL478::m-Chlorophenylpiperazine::mCPP
SMILES Clc1cccc(c1)N1CCNCC1
InChI Key InChIKey=VHFVKMTVMIZMIK-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 159 hits for monomerid = 50001915
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Affinity DataKi: 4.40nMAssay Description:Binding affinity at rat 5-hydroxytryptamine 1B receptor by [3H]-5-HT displacement.More data for this Ligand-Target Pair
Affinity DataKi: 7.90nMAssay Description:Displacement of [125I]DOI from recombinant human 5-HT2C receptor expressed in HEK293 cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Displacement of [3H]5HT from human 5HT2CMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Affinity for human 5-hydroxytryptamine 2A receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [125I]DOI from recombinant human 5-HT2B receptor expressed in HEK293 cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Emory University
Curated by PDSP Ki Database
Emory University
Curated by PDSP Ki Database
Affinity DataKi: 17nMAssay Description:Displacement of [125I]DOI from human recombinant 5HT2C expressed in HEK293E cellsMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Displacement of [125I]DOI from human recombinant 5HT2C receptor expressed in HEK293E cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Roche Bioscience
Curated by PDSP Ki Database
Roche Bioscience
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 3A(RAT)
Virginia Commonwealth University
Curated by PDSP Ki Database
Virginia Commonwealth University
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Roche Bioscience
Curated by PDSP Ki Database
Roche Bioscience
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Roche Bioscience
Curated by PDSP Ki Database
Roche Bioscience
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Stanford University
Curated by PDSP Ki Database
Stanford University
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Emory University
Curated by PDSP Ki Database
Emory University
Curated by PDSP Ki Database
Affinity DataKi: 23nMAssay Description:Binding affinity at rat 5-hydroxytryptamine 1A receptor by [3H]-WB-4101 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT2B expressed in HEK293E cellsMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Displacement of [125I]LSD from human recombinant 5HT2B receptor expressed in HEK293E cellsMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Agonist activity at 5-HT2A receptor (unknown origin) expressed in HEK293 cells assessed as [3H]inositol phosphate accumulation after 2 hrs by scintil...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A/1B/1D/1F(RAT)
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Inhibition of [3H]5-HT radioligand binding against 5-hydroxytryptamine 1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Binding affinity to 5HT2C (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Displacement of [3H]5HT from human 5HT2BMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Affinity for human 5-hydroxytryptamine 2C receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Binding affinity to 5-HT2AR (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetSerotonin 2 (5-HT2) receptor(RAT)
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Binding affinity at rat 5-hydroxytryptamine 2 receptor by [3H]ketanserin displacement.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Cracow University Of Technology
Curated by ChEMBL
Cracow University Of Technology
Curated by ChEMBL
Affinity DataKi: 42nMAssay Description:Binding affinity to 5-HT1AR (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Displacement of [125I]DOI from human recombinant 5HT2A receptor expressed in HEK293E cellsMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Displacement of [125I]DOI from human recombinant 5HT2A expressed in HEK293E cellsMore data for this Ligand-Target Pair
Affinity DataKi: 54nMAssay Description:Affinity for human 5-hydroxytryptamine 2A receptor expressed in mammalian cell lineMore data for this Ligand-Target Pair
Affinity DataKi: 54nMAssay Description:Displacement of [125I]DOI from human 5HT2AMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Roche Bioscience
Curated by PDSP Ki Database
Roche Bioscience
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 3A/3B/3C/3D/3E(Homo sapiens (Human))
Virginia Commonwealth University
Curated by ChEMBL
Virginia Commonwealth University
Curated by ChEMBL
Affinity DataKi: 62nMAssay Description:Compound was tested for the inhibition of [3H]-GR-65,630 binding to 5-hydroxytryptamine 3 receptor expressed in NG 108-15 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Mcneil Pharmaceutical And Janssen Research Foundation Worldwide
Curated by ChEMBL
Affinity DataKi: 75nMAssay Description:Binding affinity (Ki) to rat cortical membranes at 5-HT1B binding site by using [125 I] ICYP as a radioligand.More data for this Ligand-Target Pair