BDBM50011236 CHEMBL344314::Isoquinoline-5-sulfonic acid (2-amino-ethyl)-amide::Isoquinolinesulfonamide, H-9::N-(2-aminoethyl)isoquinoline-5-sulfonamide
SMILES NCCNS(=O)(=O)c1cccc2cnccc12
InChI Key InChIKey=DCVZSHVZGVWQKV-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 8 hits for monomerid = 50011236
Affinity DataIC50: 1.10E+5nMpH: 7.4 T: 2°CAssay Description:Casein kinase activities were determined under the conditions as described by Huang et al (1982).More data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+5nMpH: 7.4 T: 2°CAssay Description:Casein kinase activities were determined under the conditions as described by Huang et al (1982).More data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+4nMpH: 7.4 T: 2°CAssay Description:Casein kinase activities were determined under the conditions as described by Huang et al (1982).More data for this Ligand-Target Pair
TargetO94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Ura Cnrs 1309
Curated by ChEMBL
Ura Cnrs 1309
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of protein kinase C (PKC)More data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase II inhibitor 2(Bos taurus (Bovine))
Nagoya University School Of Medicine
Nagoya University School Of Medicine
Affinity DataIC50: 5.80E+4nMpH: 7.4 T: 2°CAssay Description:Casein kinase activities were determined under the conditions as described by Huang et al (1982).More data for this Ligand-Target Pair
TargetMO15-related protein kinase Pfmrk(Plasmodium falciparum)
Institute Of Research
Curated by ChEMBL
Institute Of Research
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of Plasmodium falciparum PfmrkMore data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit gamma(Homo sapiens (Human))
Ura Cnrs 1309
Curated by ChEMBL
Ura Cnrs 1309
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of cAMP-dependent protein kinase (PKA).More data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bos taurus)
Nagoya University School Of Medicine
Nagoya University School Of Medicine
Affinity DataIC50: 3.60E+3nMpH: 7.4 T: 2°CAssay Description:Casein kinase activities were determined under the conditions as described by Huang et al (1982).More data for this Ligand-Target Pair