BDBM50011628 4-(2-Chloro-phenyl)-2-iodo-9-methyl-6H-1-thia-5,7,8,9a-tetraaza-cyclopenta[e]azulene::CHEMBL20359

SMILES Cc1nnc2CN=C(c3cc(I)sc3-n12)c1ccccc1Cl

InChI Key InChIKey=KJZJHABCRCESGN-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50011628   

TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011628(4-(2-Chloro-phenyl)-2-iodo-9-methyl-6H-1-thia-5,7,...)
Affinity DataIC50:  370nMAssay Description:PAF-antagonist activity determined in dog platelets by PAF-binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011628(4-(2-Chloro-phenyl)-2-iodo-9-methyl-6H-1-thia-5,7,...)
Affinity DataIC50:  370nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed