BDBM50011868 4-(2-Chloro-phenyl)-2-[2-(4-cyclohexyl-phenyl)-ethyl]-9-methyl-6H-1-thia-5,7,8,9a-tetraaza-cyclopenta[e]azulene::CHEMBL432850

SMILES Cc1nnc2CN=C(c3cc(CCc4ccc(cc4)C4CCCCC4)sc3-n12)c1ccccc1Cl

InChI Key InChIKey=KVEJKTJWEFXFDT-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50011868   

TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011868(4-(2-Chloro-phenyl)-2-[2-(4-cyclohexyl-phenyl)-eth...)
Affinity DataIC50:  35nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed