BDBM50015784 1-Ethyl-7-methoxy-[1,2,4]triazolo[4,3-a]quinoxalin-4-ylamine::CHEMBL431376

SMILES CCc1nnc2c(N)nc3cc(OC)ccc3n12

InChI Key InChIKey=BKXFREWVIYPFIN-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50015784   

TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015784(1-Ethyl-7-methoxy-[1,2,4]triazolo[4,3-a]quinoxalin...)
Affinity DataIC50:  36nMAssay Description:Evaluated for the binding affinity towards the Adenosine A2 receptor in corpora striata of rats using [3H]NECA as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015784(1-Ethyl-7-methoxy-[1,2,4]triazolo[4,3-a]quinoxalin...)
Affinity DataIC50:  140nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed