BDBM50032595 CHEMBL107106::[1-(1-Methyl-2-morpholin-4-yl-ethyl)-1H-indol-3-yl]-naphthalen-1-yl-methanone

SMILES CC(CN1CCOCC1)n1cc(C(=O)c2cccc3ccccc23)c2ccccc12

InChI Key InChIKey=KBBXHAYJCWLNHP-UHFFFAOYSA-N

Data  2 KI  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50032595   

TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Sanofi Research Division

Curated by ChEMBL
LigandPNGBDBM50032595(CHEMBL107106 | [1-(1-Methyl-2-morpholin-4-yl-ethyl...)
Affinity DataKi:  3.80E+7nMAssay Description:Cannabinoid receptor 1 binding affinity by measuring its ability to displace [3H]WIN-55212-2 in rat forebrain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Sanofi Research Division

Curated by ChEMBL
LigandPNGBDBM50032595(CHEMBL107106 | [1-(1-Methyl-2-morpholin-4-yl-ethyl...)
Affinity DataKi:  3.80E+7nMAssay Description:Cannabinoid receptor 1 binding affinity by measuring its ability to displace [3H]WIN-55212-2 in rat forebrain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Sanofi Research Division

Curated by ChEMBL
LigandPNGBDBM50032595(CHEMBL107106 | [1-(1-Methyl-2-morpholin-4-yl-ethyl...)
Affinity DataIC50:  33nMAssay Description:Concentration of compound required to inhibit 50% of [3H]-WIN- 55212 binding to Cannabinoid receptor 1 in rat cerebellum membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Sanofi Research Division

Curated by ChEMBL
LigandPNGBDBM50032595(CHEMBL107106 | [1-(1-Methyl-2-morpholin-4-yl-ethyl...)
Affinity DataIC50:  33nMAssay Description:Concentration of compound required to inhibit 50% of [3H]-WIN- 55212 binding to Cannabinoid receptor 1 in rat cerebellum membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed