BDBM50041147 (S)-2-Amino-3-(4-hydroxy-phenyl)-N-((5S,8S,17aR)-5-naphthalen-2-ylmethyl-4,7,14,17-tetraoxo-hexadecahydro-3a,6,13,16-tetraaza-cyclopentacyclohexadecen-8-yl)-propionamide::CHEMBL274012
SMILES N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@H]1CCCCNC(=O)CNC(=O)[C@H]2CCCN2C(=O)[C@H](Cc2ccc3ccccc3c2)NC1=O
InChI Key InChIKey=HXRSYJPZHHJNPY-GCXHJFECSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50041147
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Binding affinity for mu opioid receptors by displacement of [3H]-DAMGO from rat brain membrane binding siteMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montreal
Curated by ChEMBL
Clinical Research Institute Of Montreal
Curated by ChEMBL
Affinity DataKi: 63nMAssay Description:Binding affinity for delta opioid receptors was determined by displacement of [3H]DSLET from rat brain membrane binding siteMore data for this Ligand-Target Pair
Affinity DataIC50: 609nMAssay Description:In vitro inhibition of electrically evoked contractions of the guinea pig ileum (GPI)More data for this Ligand-Target Pair