BDBM50049788 1-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-3-[4-methyl-3-(1H-tetrazol-5-ylamino)-phenyl]-urea::CHEMBL170275

SMILES CN1c2ccccc2C(=N[C@@H](NC(=O)Nc2ccc(C)c(Nc3nnn[nH]3)c2)C1=O)c1ccccc1

InChI Key InChIKey=HCOILVMPQWKLPU-QFIPXVFZSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50049788   

TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50049788(1-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of [125 I]BH CCK-8S binding to Cholecystokinin type B receptor in guinea pig cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Neuroscience Research Centre

Curated by ChEMBL
LigandPNGBDBM50049788(1-((R)-1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of [125 I]BH CCK-8S binding to Cholecystokinin type A receptor in pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed