BDBM50065520 4-[2-Pyridin-2-yl-5-(thiophen-3-ylmethoxy)-phenoxy]-4-o-tolyl-butyric acid::CHEMBL92965

SMILES Cc1ccccc1C(CCC(O)=O)Oc1cc(OCc2ccsc2)ccc1-c1ccccn1

InChI Key InChIKey=BRFPHZRJHAJJMA-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50065520   

TargetEndothelin receptor type B(RAT)
Rh£Ne-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065520(4-[2-Pyridin-2-yl-5-(thiophen-3-ylmethoxy)-phenoxy...)
Affinity DataIC50:  1.00E+4nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat cerebellum Endothelin B receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Rh£Ne-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50065520(4-[2-Pyridin-2-yl-5-(thiophen-3-ylmethoxy)-phenoxy...)
Affinity DataIC50:  40nMAssay Description:In vitro inhibition of [125I]ET1 binding to rat A10 cell Endothelin A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed