BDBM50068234 5'-Chloro-1H,1''H-[3,3':3',3''-terindol]-2'(1'H)-one (4c)::CHEMBL2011865
SMILES Clc1ccc2NC(=O)C(c2c1)(c1c[nH]c2ccccc12)c1c[nH]c2ccccc12
InChI Key InChIKey=KQTQQJVFFASAJD-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 8 hits for monomerid = 50068234
Affinity DataKi: 670nMAssay Description:Displacement of [3H]LSD from human cloned 5-HT6R expressed in HEK293 cells using seven compounds concentrationsMore data for this Ligand-Target Pair
Affinity DataKi: 720nMAssay Description:Displacement of [3H]LSD from human cloned 5-HT6R expressed in HEK293 cells at 0.1 and 1 uMMore data for this Ligand-Target Pair
Affinity DataKi: 2.45E+3nMAssay Description:Displacement of [3H]-8-OH-DPAT from human cloned 5-HT1A receptor expressed in HEK293 cells at 0.1 and 1 uMMore data for this Ligand-Target Pair
Affinity DataKi: 1.58E+4nMAssay Description:Displacement of [3H]-ketanserin from human cloned 5-HT2A receptor expressed in CHO-K1 cells using seven compounds concentrationsMore data for this Ligand-Target Pair
Affinity DataKi: 1.81E+4nMAssay Description:Displacement of [3H]-5-CT from human cloned 5-HT7R expressed in HEK293 cells at 0.1 and 1 uMMore data for this Ligand-Target Pair
Affinity DataKi: 1.83E+4nMAssay Description:Displacement of [3H]-ketanserin from human cloned 5-HT2A receptor expressed in CHO-K1 cells at 0.1 and 1 uMMore data for this Ligand-Target Pair
TargetProbable maltase-glucoamylase 2(Homo sapiens)
Babasaheb Bhimrao Ambedkar University (A Central University)
Curated by ChEMBL
Babasaheb Bhimrao Ambedkar University (A Central University)
Curated by ChEMBL
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of alpha-glucosidase (unknown origin) using p-nitrophenyl-alpha-d-glucopyranoside as substrate preincubated for 15 mins followed by substr...More data for this Ligand-Target Pair
Affinity DataIC50: 5.05E+4nMpH: 6.8 T: 2°CAssay Description:The α-glucosidase inhibition assay had been carried out using baker's yeast α-glucosidase (EC 3.2.1.20) and p-nitrophenyl α-d-gluco...More data for this Ligand-Target Pair