BDBM50069107 CHEMBL356792

SMILES [H][C@@](Cc1cccc(c1)C(N)=N)(NS(=O)(=O)c1ccc2ccccc2c1)C(=O)N1CCN(CC1)c1ccccc1

InChI Key InChIKey=FVLGQHJQXSNNFU-NDEPHWFRSA-N

Data  6 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50069107   

TargetSerine protease 1(Bos taurus (bovine))
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50069107(CHEMBL356792)
Affinity DataKi:  27nMAssay Description:Binding affinity towards trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50069107(CHEMBL356792)
Affinity DataKi:  520nMAssay Description:Binding affinity towards thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50069107(CHEMBL356792)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of matripase (unknown origin) using Boc-QAR-AMC as substrate incubated for 30 mins prior to substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease hepsin(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50069107(CHEMBL356792)
Affinity DataKi:  7.00E+3nMAssay Description:Inhibition of hepsin (unknown origin) using Boc-QAR-AMC as substrate after 30 mins prior to substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor activator(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50069107(CHEMBL356792)
Affinity DataKi:  1.82E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged HGFA (unknown origin) expressed in baculovirus-infected Sf9 cells using Boc-QLR-AMC as substrate incu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50069107(CHEMBL356792)
Affinity DataKi:  2.69E+4nMAssay Description:Binding affinity towards Coagulation factor XaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed