BDBM50090688 7-Methyl-2-(4-nitro-phenyl)-[1,8]naphthyridin-4-ol::CHEMBL316630

SMILES Cc1ccc2c(O)cc(nc2n1)-c1ccc(cc1)[N+]([O-])=O

InChI Key InChIKey=MGONMXNIZCTIPU-UHFFFAOYSA-N

Data  7 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 7 hits for monomerid = 50090688   

TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50090688(7-Methyl-2-(4-nitro-phenyl)-[1,8]naphthyridin-4-ol...)
Affinity DataKi:  9.90nMAssay Description:Binding affinity against adenosine A1 receptor in bovine cortical membranes using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50090688(7-Methyl-2-(4-nitro-phenyl)-[1,8]naphthyridin-4-ol...)
Affinity DataKi:  10nMAssay Description:Ability to displace the specific binding of [3H]CHA to adenosine A1 receptor from bovine brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50090688(7-Methyl-2-(4-nitro-phenyl)-[1,8]naphthyridin-4-ol...)
Affinity DataKi:  460nMAssay Description:Binding affinity against adenosine A2 receptor in bovine striatal membranes using [3H]-CGS-21,680 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50090688(7-Methyl-2-(4-nitro-phenyl)-[1,8]naphthyridin-4-ol...)
Affinity DataKi:  460nMAssay Description:Ability to displace the specific binding of [3H]-CGS- to adenosine A2A receptor form bovine brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50090688(7-Methyl-2-(4-nitro-phenyl)-[1,8]naphthyridin-4-ol...)
Affinity DataKi:  640nMAssay Description:Binding affinity against adenosine A2 receptor in human striatal membranes using [3H]-CGS-21,680 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50090688(7-Methyl-2-(4-nitro-phenyl)-[1,8]naphthyridin-4-ol...)
Affinity DataKi:  3.10E+3nMAssay Description:Binding affinity against adenosine A1 receptor in human cortical membranes using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50090688(7-Methyl-2-(4-nitro-phenyl)-[1,8]naphthyridin-4-ol...)
Affinity DataKi: >1.00E+4nMAssay Description:Ability to displace the specific binding of [3H](R)-PIA to adenosine A3 receptor from rat testis membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed