BDBM50094886 CHEMBL3589468

SMILES COc1ccc(\C=C(\C(=O)N2CC(=O)Nc3ccccc23)c2ccccc2)cc1

InChI Key InChIKey=WQITZMVRSQPEBE-HMMYKYKNSA-N

Data  2 IC50

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50094886   

TargetBromodomain-containing protein 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094886(CHEMBL3589468)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD2(2) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50094886(CHEMBL3589468)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of HTRF binding to N-terminal His-tagged BRD4(1) (unknown origin) using biotinylated tetra-acetylated histone H4 peptide and Cryptate-labe...More data for this Ligand-Target Pair