BDBM50095646 CHEMBL410795::H-DTyr-Val-Met-Gly-His-Phe-Arg-Trp-Asp-Arg-Phe-Gly-OH::H-Tyr-DVal-Met-Gly-His-Phe-Arg-Trp-Asp-Arg-Phe-Gly-OH::H-Tyr-Val-DMet-Gly-His-Phe-Arg-Trp-Asp-Arg-Phe-Gly-OH::H-Tyr-Val-Met-Gly-DHis-Phe-Arg-Trp-Asp-Arg-Phe-Gly-OH::H-Tyr-Val-Met-Gly-His-DPhe-Arg-Trp-Asp-Arg-Phe-Gly-OH::H-Tyr-Val-Met-Gly-His-Phe-Arg-DTrp-Asp-Arg-Phe-Gly-OH::H-Tyr-Val-Met-Gly-His-Phe-Arg-Trp-Asp-Arg-DPhe-Gly-OH::H-Tyr-Val-Met-Gly-His-Phe-Arg-Trp-Asp-Arg-Phe-Gly-OH( gama-melanocyte-stimulating hormone(MSH))::H-Tyr-Val-Met-Gly-His-Phe-Arg-Trp-Asp-DArg-Phe-Gly-OH::H-Tyr-Val-Met-Gly-His-Phe-Arg-Trp-DAsp-Arg-Phe-Gly-OH::H-Tyr-Val-Met-Gly-His-Phe-DArg-Trp-Asp-Arg-Phe-Gly-OH

SMILES CSCC[C@H](NC(=O)[C@@H](NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(C)C)C(=O)NCC(=O)N[C@@H](Cc1cnc[nH]1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@H](CC(O)=O)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](Cc1ccccc1)C(=O)NCC(O)=O

InChI Key InChIKey=GZWUQPQBOGLSIM-BQLCFHTJSA-N

Data  3 IC50  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50095646   

TargetMelanocortin receptor 5(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50095646(CHEMBL410795 | H-DTyr-Val-Met-Gly-His-Phe-Arg-Trp-...)
Affinity DataEC50:  550nMAssay Description:Effective concentration required for intracellular cAMP accumulation by Melanocortin 5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50095646(CHEMBL410795 | H-DTyr-Val-Met-Gly-His-Phe-Arg-Trp-...)
Affinity DataEC50:  940nMAssay Description:Effective concentration required for intracellular cAMP accumulation by Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50095646(CHEMBL410795 | H-DTyr-Val-Met-Gly-His-Phe-Arg-Trp-...)
Affinity DataIC50:  1.10E+3nMAssay Description:Binding affinity for Human Melanocortin 4 receptor expressed in L-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50095646(CHEMBL410795 | H-DTyr-Val-Met-Gly-His-Phe-Arg-Trp-...)
Affinity DataEC50:  250nMAssay Description:Effective concentration required for intracellular cAMP accumulation against Melanocortin 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50095646(CHEMBL410795 | H-DTyr-Val-Met-Gly-His-Phe-Arg-Trp-...)
Affinity DataIC50:  540nMAssay Description:Effective concentration required for intracellular cAMP accumulation by Melanocortin 5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50095646(CHEMBL410795 | H-DTyr-Val-Met-Gly-His-Phe-Arg-Trp-...)
Affinity DataIC50:  1.00E+3nMAssay Description:Binding affinity for Human Melanocortin 3 receptor expressed in L-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed