BDBM50122699 2'-Imidazol-1-ylmethyl-4'-oxazol-2-yl-biphenyl-2-sulfonic acid (3,4-dimethyl-isoxazol-5-yl)-amide::CHEMBL30009

SMILES Cc1noc(NS(=O)(=O)c2ccccc2-c2ccc(cc2Cn2ccnc2)-c2ncco2)c1C

InChI Key InChIKey=KAIWKTKPOCNWMM-UHFFFAOYSA-N

Data  2 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50122699   

TargetEndothelin-1 receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50122699(2'-Imidazol-1-ylmethyl-4'-oxazol-2-yl-biphenyl-2-s...)
Affinity DataKi:  0.300nMAssay Description:Inhibitory activity against human endothelin A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50122699(2'-Imidazol-1-ylmethyl-4'-oxazol-2-yl-biphenyl-2-s...)
Affinity DataKi:  4.30E+3nMAssay Description:Inhibitory activity against human endothelin B receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed