BDBM50123658 3-[(R)-((2S,5R)-4-Allyl-2,5-dimethyl-piperazin-1-yl)-(3-hydroxy-phenyl)-methyl]-N-(3-fluoro-phenyl)-N-methyl-benzamide::CHEMBL155892
SMILES C[C@@H]1CN([C@@H](c2cccc(O)c2)c2cccc(c2)C(=O)N(C)c2cccc(F)c2)[C@@H](C)CN1CC=C
InChI Key InChIKey=LZXRQLIIMYJZDA-UETOGOEVSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 8 hits for monomerid = 50123658
Affinity DataKi: 0.180nMAssay Description:Displacement of [3H]DPDPE from mu opioid receptor in albino Sprague-Dawley rat after 90 mins by liquid scintillationMore data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Binding affinity of compound evaluated for Opioid receptor delta 1 isolated from rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Binding affinity of compound evaluated for Opioid receptor delta 1 isolated from rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Binding affinity of compound evaluated for Opioid receptor mu 1 isolated from rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Displacement of [3H]DAMGO from kappa opioid receptor in albino Sprague-Dawley rat after 90 mins by liquid scintillationMore data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Binding affinity of compound evaluated for Opioid receptor mu 1 isolated from rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:Antagonist activity at human delta opioid receptor in CD1 mouse assessed as electrically induced twitchesMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Agonist activity at mu-opioid receptor in guinea pig ileum assessed as inhibition of electrically induced twitchesMore data for this Ligand-Target Pair