BDBM50146360 CHEMBL328573::Dimethyl-[(2S,3aR)-1-(2,3,3a,8-tetrahydro-1-oxa-12b-aza-dibenzo[e,h]azulen-2-yl)methyl]-amine
SMILES CN(C)C[C@@H]1C[C@H]2N(O1)c1ccccc1Cc1ccccc21
InChI Key InChIKey=BTSCZNWXJQSJIE-QFBILLFUSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 41 hits for monomerid = 50146360
Affinity DataKi: 0.640nMAssay Description:Ability to displace [3H]-pyrilamine from human cloned histamine H1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Ability to displace [3H]- mesulergine from human cloned 5-hydroxytryptamine 2C receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Ability to displace [125I]-R91150 from human cloned 5-hydroxytryptamine 2A receptor expressed in L929 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 537nMAssay Description:Binding affinity against Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 372nMAssay Description:Binding affinity against Alpha-2A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 661nMAssay Description:Binding affinity against 5-HT1D receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 871nMAssay Description:Binding affinity against Dopamine receptor D2LMore data for this Ligand-Target Pair
Affinity DataIC50: 977nMAssay Description:Binding affinity against 5-HT1A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.86E+3nMAssay Description:Binding affinity against Alpha-3A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Binding affinity against Dopamine receptor D3More data for this Ligand-Target Pair
Affinity DataIC50: 6.80nMAssay Description:Binding affinity against Histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Binding affinity against 5-HT2C receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 132nMAssay Description:Binding affinity against Dopamine receptor D4More data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Binding affinity against 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 537nMAssay Description:Binding affinity for human cloned Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Binding affinity for human cloned Dopamine receptor D3More data for this Ligand-Target Pair
Affinity DataIC50: 977nMAssay Description:Binding affinity for human cloned 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 132nMAssay Description:Binding affinity for human cloned Dopamine receptor D4More data for this Ligand-Target Pair
Affinity DataIC50: 372nMAssay Description:Binding affinity for human cloned Alpha-2A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 661nMAssay Description:Binding affinity for human cloned 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 661nMAssay Description:Binding affinity for human cloned 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 537nMAssay Description:Binding affinity for human cloned Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+3nMAssay Description:Binding affinity for human cloned 5-hydroxytryptamine 2A receptor expressed in L929 cells using [125I]R91150 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 871nMAssay Description:Binding affinity for human cloned Dopamine receptor D2LMore data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+3nMAssay Description:Binding affinity for human cloned Histamine H1 receptor expressed in CHO cells using [3H]pyrilamine as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Binding affinity for human cloned Dopamine receptor D3More data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+3nMAssay Description:Binding affinity for human cloned 5-hydroxytryptamine 2C receptor expressed in CHO cells using [3H]mesulergine as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 977nMAssay Description:Binding affinity for human cloned 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 132nMAssay Description:Binding affinity for human cloned Dopamine receptor D4More data for this Ligand-Target Pair
Affinity DataIC50: 372nMAssay Description:Binding affinity for human cloned Alpha-2A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 195nMAssay Description:Binding affinity for rat Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataIC50: 1.86E+3nMAssay Description:Binding affinity for human cloned Alpha-2C adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.86E+3nMAssay Description:Binding affinity for human cloned Alpha-2C adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 2C receptor expressed in CHO cells by [3H]mesulergine displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 195nMAssay Description:Binding affinity for rat Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataIC50: 871nMAssay Description:Binding affinity for human cloned Dopamine receptor D2LMore data for this Ligand-Target Pair
Affinity DataIC50: 6.80nMAssay Description:Binding affinity at human cloned Histamine H1 receptor expressed in CHO cells by [3H]pyrilamine displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Binding affinity for human cloned 5-hydroxytryptamine 2A receptor expressed in L929 cells using [125I]R91150 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Binding affinity for human cloned 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 6.80nMAssay Description:Binding affinity for human cloned 5-hydroxytryptamine 2A receptor expressed in L929 cells using [125I]R91150 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Binding affinity at human cloned 5-hydroxytryptamine 2A receptor expressed in L929 cells by [125I]R91150 displacement.More data for this Ligand-Target Pair