BDBM50157901 CHEMBL3780073
SMILES CN1CCN(CC1)c1ccc(NC(=O)c2c(Nc3ccccc3C)cc[nH]c2=O)cc1
InChI Key InChIKey=KGMPHIGFGPMSLD-UHFFFAOYSA-N
Data 2 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50157901
Affinity DataKi: 61nMAssay Description:Inhibition of human EGFR catalytic domain (668 to 1210 residues) T790M/L858R double mutant using Fl-EEPLYWSFPAKKK-CONH2 peptide substrate preincubate...More data for this Ligand-Target Pair
Affinity DataKi: 2.34E+3nMAssay Description:Inhibition of human N-terminal GST-tagged EGFR catalytic domain (669 to 1210 residues) expressed in baculovirus expression system using Fl-EEPLYWSFPA...More data for this Ligand-Target Pair