BDBM50158891 CHEMBL3785194

SMILES Fc1ccc(nc1)-c1cc(ccc1O[C@@H]1CCOc2cc(ccc12)S(=O)(=O)Nc1nccs1)C(F)(F)F

InChI Key InChIKey=HIWLPNGXXFNDGE-OAQYLSRUSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50158891   

TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50158891(CHEMBL3785194)
Affinity DataIC50:  4nMAssay Description:Inhibition of Nav1.7 (unknown origin) overexpressed in HEK293 cells preincubated for 15 to 20 mins followed by depolarization with 10 to 30 uM veratr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed