BDBM50170654 (+-)-cis-4-(3-(4-tert-butylphenyl)-2-methylpropyl)-2,6-dimethylmorpholine::(2R,6S)-4-[3-(4-tert-butylphenyl)-2-methylpropyl]-2,6-dimethylmorpholine::CHEMBL372700::cis-2,6-dimethyl-4-(3-(4-(1,1-dimethylethyl)phenyl)-2-methylpropyl)morpholine::cis-4-(3-(4-(1,1-dimethylethyl)phenyl)-2-methylpropyl)-2,6-dimethylmorpholine::cis-4-(3-(p-tert-butylphenyl)-2-methylpropyl)-2,6-dimethylmorpholine::cis-fenpropimorph::fenpropimorph::fenpropimorph cis-form::fenpropimorphe
SMILES CC(CN1C[C@H](C)O[C@H](C)C1)Cc1ccc(cc1)C(C)(C)C
InChI Key InChIKey=RYAUSSKQMZRMAI-ALOPSCKCSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 16 hits for monomerid = 50170654
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.00500nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma 1 receptor in guinea pig brain microsomesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.00500nMAssay Description:Displacement of (+)-[3H]-pentazocine from sigma 1 receptor in guinea pig whole brain microsomesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.00500nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma 1 receptor in guinea pigMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University Of Innsbruck
Curated by ChEMBL
University Of Innsbruck
Curated by ChEMBL
Affinity DataKi: 0.0100nMAssay Description:Affinity for sigma receptor type 1 of guinea pig using [3H]ifenprodil or (+)-[3H]pentazocine radioligandMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.0110nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma 1 receptor in guinea pig liver microsomesMore data for this Ligand-Target Pair
Affinity DataKi: 0.0110nMAssay Description:Displacement of [3H]-pentazocine from sigma 1 opioid receptor in rat liver homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.0110nMAssay Description:Displacement of (+)-[3H]-pentazocine from sigma 1 receptor in guinea pig liver microsomesMore data for this Ligand-Target Pair
Affinity DataKi: 0.0500nMAssay Description:Affinity for ERG2 of Sacchromyces cerevisiae using [3H]ifenprodil or (+)-[3H]pentazocine radioligandMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University Of Innsbruck
Curated by ChEMBL
University Of Innsbruck
Curated by ChEMBL
Affinity DataKi: 0.0800nMAssay Description:Displacement of (+)-[3H]pentazocine from sigma 1 receptor expressed in Saccharomyces cerevisiae WA0More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
University Of Wisconsin School Of Medicine And Public Health
Curated by ChEMBL
Affinity DataKi: 0.0800nMAssay Description:Displacement of (+)-[3H]-pentazocine from recombinant guinea pig His6-tagged sigma 1 receptor expressed in Saccharomyces cerevisiae WAO microsomesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University Of Innsbruck
Curated by ChEMBL
University Of Innsbruck
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Displacement of (+)-[3H]-pentazocine from recombinant human sigma 1 receptor expressed in baculovirus infected Sf9 insect cell membranes after 90 min...More data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Homo sapiens (Human))
University Of Innsbruck
Curated by ChEMBL
University Of Innsbruck
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Affinity for human EMP expressed in ERG2 deficient strain of Sacchromyces cerevisiae using [3H]ifenprodil or (+)-[3H]pentazocine as radioligandMore data for this Ligand-Target Pair
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
Virginia Commonwealth University
Curated by ChEMBL
Virginia Commonwealth University
Curated by ChEMBL
Affinity DataKi: 854nMAssay Description:Displacement of (+)-[3H]-ditolylguanidine from recombinant rat sigma 2 receptor expressed in rat PC12 cell membranes after 90 mins in presence of sig...More data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of Zea mays (maize) cycloeucalenol-obtusifolial isomeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of Zea mays (maize) delta8,delta7-sterol isomeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Inhibition of Zea mays (maize) microsomal delta 8,14-steroid 14-reductase using delta 8,14-cholestadienol as substrate after 90 min by GC analysisMore data for this Ligand-Target Pair